EA201170483A1 - Твердая фармацевтическая композиция - Google Patents

Твердая фармацевтическая композиция

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Publication number
EA201170483A1
EA201170483A1 EA201170483A EA201170483A EA201170483A1 EA 201170483 A1 EA201170483 A1 EA 201170483A1 EA 201170483 A EA201170483 A EA 201170483A EA 201170483 A EA201170483 A EA 201170483A EA 201170483 A1 EA201170483 A1 EA 201170483A1
Authority
EA
Eurasian Patent Office
Prior art keywords
pharmaceutical composition
solid pharmaceutical
salt
stability
containing compound
Prior art date
Application number
EA201170483A
Other languages
English (en)
Inventor
Казухиро Хирата
Дзуниа Номура
Ютака Таноуе
Original Assignee
Такеда Фармасьютикал Компани Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42059801&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201170483(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Такеда Фармасьютикал Компани Лимитед filed Critical Такеда Фармасьютикал Компани Лимитед
Publication of EA201170483A1 publication Critical patent/EA201170483A1/ru

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    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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Abstract

В данном изобретении представлен твердый препарат, содержащий соединение (I) или его соль, контролирующее рН средство и антагонист кальция, который имеет превосходное свойство высвобождения, стабильность и подобные.
EA201170483A 2008-09-25 2009-09-25 Твердая фармацевтическая композиция EA201170483A1 (ru)

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PCT/JP2009/066690 WO2010035806A1 (ja) 2008-09-25 2009-09-25 固形医薬組成物

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US9173849B2 (en) 2015-11-03
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CN102223884B (zh) 2015-05-06
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JP5570426B2 (ja) 2014-08-13
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CN104306975A (zh) 2015-01-28
CL2011000625A1 (es) 2011-07-08
WO2010035806A1 (ja) 2010-04-01
PE20110844A1 (es) 2011-12-05
CR20110209A (es) 2011-05-27
ECSP11011001A (es) 2011-05-31
UA102271C2 (en) 2013-06-25
EP2332535A1 (en) 2011-06-15
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