UY32126A - Composición farmacéutica sólida - Google Patents

Composición farmacéutica sólida

Info

Publication number
UY32126A
UY32126A UY0001032126A UY32126A UY32126A UY 32126 A UY32126 A UY 32126A UY 0001032126 A UY0001032126 A UY 0001032126A UY 32126 A UY32126 A UY 32126A UY 32126 A UY32126 A UY 32126A
Authority
UY
Uruguay
Prior art keywords
pharmaceutical composition
solid pharmaceutical
dissolution
superior
stability
Prior art date
Application number
UY0001032126A
Other languages
English (en)
Inventor
Tanoue Yutaka
Nomura Junya
Hirata Kazuhiro
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42059801&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY32126(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of UY32126A publication Critical patent/UY32126A/es

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    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
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    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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  • Physical Education & Sports Medicine (AREA)
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  • Urology & Nephrology (AREA)
  • Obesity (AREA)
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  • Addiction (AREA)
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  • Reproductive Health (AREA)

Abstract

La presente invención provee una preparación sólida que contiene el compuesto (I) o una de sus sales correspondientes, un agente der control de pH y un antagonista de calcio, la cual es superior en las propiedades de disolución, estabilidad y similares
UY0001032126A 2008-09-25 2009-09-16 Composición farmacéutica sólida UY32126A (es)

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CO6361934A2 (es) 2012-01-20
IL211886A0 (en) 2011-06-30
EP2332535A4 (en) 2013-11-27
US20110229567A1 (en) 2011-09-22
AU2009297522A1 (en) 2010-04-01
CA2738147A1 (en) 2010-04-01
GEP20146063B (en) 2014-03-25
KR20110063557A (ko) 2011-06-10
TW201014850A (en) 2010-04-16
NZ592225A (en) 2012-06-29
CN104306975A (zh) 2015-01-28
WO2010035806A1 (ja) 2010-04-01
AR073380A1 (es) 2010-11-03
ZA201102715B (en) 2012-07-25
CR20110209A (es) 2011-05-27
PE20110844A1 (es) 2011-12-05
CA2738147C (en) 2016-10-11
US9173849B2 (en) 2015-11-03
CN102223884B (zh) 2015-05-06
BRPI0918955A2 (pt) 2015-12-01
MA32721B1 (fr) 2011-10-02
CL2011000625A1 (es) 2011-07-08
JPWO2010035806A1 (ja) 2012-02-23
UA102271C2 (en) 2013-06-25
EA201170483A1 (ru) 2011-10-31
MX2011003261A (es) 2011-04-21
JP5570426B2 (ja) 2014-08-13
EP2332535A1 (en) 2011-06-15
ECSP11011001A (es) 2011-05-31
CN102223884A (zh) 2011-10-19

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