EA200970326A1 - Алкильные производные в качестве метаботропных рецепторов глутамата - Google Patents

Алкильные производные в качестве метаботропных рецепторов глутамата

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Publication number
EA200970326A1
EA200970326A1 EA200970326A EA200970326A EA200970326A1 EA 200970326 A1 EA200970326 A1 EA 200970326A1 EA 200970326 A EA200970326 A EA 200970326A EA 200970326 A EA200970326 A EA 200970326A EA 200970326 A1 EA200970326 A1 EA 200970326A1
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EA
Eurasian Patent Office
Prior art keywords
receptors
metabotropic
glutamat
alkyl derivatives
compounds
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EA200970326A
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English (en)
Inventor
Анн-Софи Бесси
Кристелль Боле
Беатрис Бонне
Марк Эппинг-Джордан
Николя Порье
Сония-Мария Поли
Жан-Филип Роше
Ив Толлон
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Аддекс Фарма Са
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Application filed by Аддекс Фарма Са filed Critical Аддекс Фарма Са
Publication of EA200970326A1 publication Critical patent/EA200970326A1/ru

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Abstract

Настоящее изобретение относится к соединениям формулы I, где W, n, Х и W' определены в описании изобретения; соединения согласно настоящему изобретению являются модуляторами метаботропных рецепторов глутамата подтипа 5 (mGluR5), полезными в лечении заболеваний центральной нервной системы, регулируемых рецепторами mGluR5.
EA200970326A 2004-06-17 2005-06-17 Алкильные производные в качестве метаботропных рецепторов глутамата EA200970326A1 (ru)

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Application Number Priority Date Filing Date Title
GBGB0413605.7A GB0413605D0 (en) 2004-06-17 2004-06-17 Novel compounds

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EA200970326A1 true EA200970326A1 (ru) 2009-12-30

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EA200970326A EA200970326A1 (ru) 2004-06-17 2005-06-17 Алкильные производные в качестве метаботропных рецепторов глутамата
EA200700047A EA012206B1 (ru) 2004-06-17 2005-06-17 Алкильные производные в качестве метаботропных рецепторов глутамата

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US (3) US8101637B2 (ru)
EP (2) EP1765795B1 (ru)
JP (2) JP5053840B2 (ru)
KR (1) KR101200175B1 (ru)
CN (2) CN101001846B (ru)
AU (1) AU2005254808B2 (ru)
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CA (1) CA2570987C (ru)
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EA (2) EA200970326A1 (ru)
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