EA200900136A1 - Пирролопиримидины для фармацевтических композиций - Google Patents

Пирролопиримидины для фармацевтических композиций

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Publication number
EA200900136A1
EA200900136A1 EA200900136A EA200900136A EA200900136A1 EA 200900136 A1 EA200900136 A1 EA 200900136A1 EA 200900136 A EA200900136 A EA 200900136A EA 200900136 A EA200900136 A EA 200900136A EA 200900136 A1 EA200900136 A1 EA 200900136A1
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EA
Eurasian Patent Office
Prior art keywords
pharmaceutical compositions
pyrrophyrimidines
pyrrolopyrimidine compounds
relates
present
Prior art date
Application number
EA200900136A
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English (en)
Inventor
Штефан Йэкель
Таня Ройтер
Стивен Мерфин
Томас Стивен Коултер
Стивен Тейлор
Original Assignee
Девелоджен Акциенгезельшафт
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Publication date
Application filed by Девелоджен Акциенгезельшафт filed Critical Девелоджен Акциенгезельшафт
Publication of EA200900136A1 publication Critical patent/EA200900136A1/ru

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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Abstract

В заявке описаны новые пирролопиримидины и фармацевтические композиции, включающие указанные пирролопиримидины. В заявке также описано применение пирролопиримидинов, предлагаемых в настоящем изобретении, для приготовления фармацевтических композиций, предназначенных для профилактики и/или лечения заболеваний, на которые можно воздействовать путем ингибирования активности киназы Mnk1 и/или Mnk2 (Mnk2a или Mnk2b) и/или их вариантов.
EA200900136A 2006-07-10 2007-07-10 Пирролопиримидины для фармацевтических композиций EA200900136A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06014297A EP1889847A1 (en) 2006-07-10 2006-07-10 Pyrrolopyrimidines for pharmaceutical compositions
PCT/EP2007/006109 WO2008006547A2 (en) 2006-07-10 2007-07-10 Pyrrolopyrimidines for pharmaceutical compositions

Publications (1)

Publication Number Publication Date
EA200900136A1 true EA200900136A1 (ru) 2009-06-30

Family

ID=37496429

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200900136A EA200900136A1 (ru) 2006-07-10 2007-07-10 Пирролопиримидины для фармацевтических композиций

Country Status (16)

Country Link
US (1) US8697713B2 (ru)
EP (2) EP1889847A1 (ru)
JP (1) JP5331951B2 (ru)
KR (1) KR20090039757A (ru)
CN (1) CN101511837A (ru)
AT (1) ATE526331T1 (ru)
AU (1) AU2007271928A1 (ru)
BR (1) BRPI0712882A2 (ru)
CA (1) CA2690277A1 (ru)
CO (1) CO6150162A2 (ru)
EA (1) EA200900136A1 (ru)
IL (1) IL196391A0 (ru)
MX (1) MX2009000333A (ru)
NO (1) NO20090029L (ru)
WO (1) WO2008006547A2 (ru)
ZA (1) ZA200810785B (ru)

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