EA025294B1 - Бициклические соединения в качестве модуляторов активности сопряженного с g-белком рецептора s1p - Google Patents
Бициклические соединения в качестве модуляторов активности сопряженного с g-белком рецептора s1p Download PDFInfo
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- EA025294B1 EA025294B1 EA201591409A EA201591409A EA025294B1 EA 025294 B1 EA025294 B1 EA 025294B1 EA 201591409 A EA201591409 A EA 201591409A EA 201591409 A EA201591409 A EA 201591409A EA 025294 B1 EA025294 B1 EA 025294B1
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- C—CHEMISTRY; METALLURGY
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Applications Claiming Priority (2)
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| US201361767531P | 2013-02-21 | 2013-02-21 | |
| PCT/US2014/017534 WO2014130752A2 (en) | 2013-02-21 | 2014-02-21 | Bicyclic compounds |
Publications (2)
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| EA201591409A1 EA201591409A1 (ru) | 2015-12-30 |
| EA025294B1 true EA025294B1 (ru) | 2016-12-30 |
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| EP3022176B8 (en) | 2013-07-15 | 2019-12-25 | The Regents of the University of California | Azacyclic constrained analogs of fty720 |
| UY36274A (es) | 2014-08-20 | 2016-02-29 | Bristol Myers Squibb Company Una Corporación Del Estado De Delaware | Compuestos bicíclicos sustituidos como agonistas selectivos de la actividad del receptor s1p1 acoplado a la proteína g |
| CA2999177A1 (en) | 2015-09-24 | 2017-03-30 | The Regents Of The University Of California | Synthetic sphingolipid-like molecules, drugs, methods of their synthesis and methods of treatment |
| CN110234633A (zh) | 2016-09-02 | 2019-09-13 | 百时美施贵宝公司 | 取代的三环杂环化合物 |
| WO2019032631A1 (en) | 2017-08-09 | 2019-02-14 | Bristol-Myers Squibb Company | Oxime ether compounds |
| WO2019032632A1 (en) | 2017-08-09 | 2019-02-14 | Bristol-Myers Squibb Company | ALKYLPHENYL COMPOUNDS |
| WO2021062168A1 (en) * | 2019-09-25 | 2021-04-01 | The Regents Of The University Of California | Synthetic sphingolipid inspired molecules with heteroaromatic appendages, methods of their synthesis and methods of treatment |
| WO2025083549A1 (en) | 2023-10-16 | 2025-04-24 | Sun Pharma Advanced Research Company Limited | Methods and combinations of inhibitors of il-23 pathway and modulators of s1p signaling pathway for the treatment of autoimmune disorders |
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| WO2008079382A1 (en) * | 2006-12-21 | 2008-07-03 | Abbott Laboratories | Sphingosine-1 -phosphate receptor agonist and antagonist compounds |
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Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2008079382A1 (en) * | 2006-12-21 | 2008-07-03 | Abbott Laboratories | Sphingosine-1 -phosphate receptor agonist and antagonist compounds |
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