EA002819B1 - Циклическое пептидное соединение и его применение, бициклопептидное соединение, пептидное соединение и его применение, фармацевтическая композиция - Google Patents

Циклическое пептидное соединение и его применение, бициклопептидное соединение, пептидное соединение и его применение, фармацевтическая композиция Download PDF

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Publication number
EA002819B1
EA002819B1 EA199901025A EA199901025A EA002819B1 EA 002819 B1 EA002819 B1 EA 002819B1 EA 199901025 A EA199901025 A EA 199901025A EA 199901025 A EA199901025 A EA 199901025A EA 002819 B1 EA002819 B1 EA 002819B1
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EA
Eurasian Patent Office
Prior art keywords
amino acid
cyclo
acre
peptide
equivalent amino
Prior art date
Application number
EA199901025A
Other languages
English (en)
Russian (ru)
Other versions
EA199901025A1 (ru
Inventor
Стефен М. Кондон
Изабелль Мориз
Original Assignee
Авентис Фармасьютикалз Продактс Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Авентис Фармасьютикалз Продактс Инк. filed Critical Авентис Фармасьютикалз Продактс Инк.
Publication of EA199901025A1 publication Critical patent/EA199901025A1/ru
Publication of EA002819B1 publication Critical patent/EA002819B1/ru

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/34Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/12Drugs for disorders of the metabolism for electrolyte homeostasis
    • A61P3/14Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/18Drugs for disorders of the endocrine system of the parathyroid hormones
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575Hormones
    • C07K14/635Parathyroid hormone, i.e. parathormone; Parathyroid hormone-related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Rheumatology (AREA)
  • Zoology (AREA)
  • Molecular Biology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Toxicology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
EA199901025A 1997-05-14 1998-05-13 Циклическое пептидное соединение и его применение, бициклопептидное соединение, пептидное соединение и его применение, фармацевтическая композиция EA002819B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US4647297P 1997-05-14 1997-05-14
PCT/US1998/009843 WO1998051324A1 (en) 1997-05-14 1998-05-13 Peptide parathyroid hormone analogs

Publications (2)

Publication Number Publication Date
EA199901025A1 EA199901025A1 (ru) 2000-06-26
EA002819B1 true EA002819B1 (ru) 2002-10-31

Family

ID=21943653

Family Applications (1)

Application Number Title Priority Date Filing Date
EA199901025A EA002819B1 (ru) 1997-05-14 1998-05-13 Циклическое пептидное соединение и его применение, бициклопептидное соединение, пептидное соединение и его применение, фармацевтическая композиция

Country Status (20)

Country Link
US (2) US6472505B1 (https=)
EP (1) EP0986395A4 (https=)
JP (1) JP2001517957A (https=)
KR (1) KR100351213B1 (https=)
CN (1) CN1261281A (https=)
AP (1) AP9901686A0 (https=)
AU (1) AU746461B2 (https=)
BG (1) BG103957A (https=)
BR (1) BR9808786A (https=)
CA (1) CA2290443A1 (https=)
EA (1) EA002819B1 (https=)
HU (1) HUP0003349A3 (https=)
IL (1) IL132901A0 (https=)
NO (1) NO995568L (https=)
OA (1) OA11216A (https=)
PL (1) PL336803A1 (https=)
SK (1) SK151599A3 (https=)
UA (1) UA62967C2 (https=)
WO (1) WO1998051324A1 (https=)
ZA (1) ZA984077B (https=)

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Also Published As

Publication number Publication date
PL336803A1 (en) 2000-07-17
AP9901686A0 (en) 1999-12-31
EP0986395A4 (en) 2004-12-01
HUP0003349A3 (en) 2001-12-28
NO995568L (no) 1999-12-29
AU7386798A (en) 1998-12-08
WO1998051324A1 (en) 1998-11-19
US20020132973A1 (en) 2002-09-19
CA2290443A1 (en) 1998-11-19
NO995568D0 (no) 1999-11-12
BG103957A (bg) 2000-04-28
OA11216A (en) 2003-07-10
JP2001517957A (ja) 2001-10-09
ZA984077B (en) 1998-11-24
BR9808786A (pt) 2000-07-11
CN1261281A (zh) 2000-07-26
IL132901A0 (en) 2001-03-19
EA199901025A1 (ru) 2000-06-26
AU746461B2 (en) 2002-05-02
KR20010012568A (ko) 2001-02-15
UA62967C2 (en) 2004-01-15
EP0986395A1 (en) 2000-03-22
HUP0003349A2 (hu) 2001-01-29
US6472505B1 (en) 2002-10-29
SK151599A3 (en) 2000-09-12
KR100351213B1 (ko) 2002-09-05

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