DZ2680A1 - Dérivé de thiazolidinedione nouveau procédé pour sa préparation et composition pharmaceutique le contenant. - Google Patents

Dérivé de thiazolidinedione nouveau procédé pour sa préparation et composition pharmaceutique le contenant.

Info

Publication number
DZ2680A1
DZ2680A1 DZ980290A DZ980290A DZ2680A1 DZ 2680 A1 DZ2680 A1 DZ 2680A1 DZ 980290 A DZ980290 A DZ 980290A DZ 980290 A DZ980290 A DZ 980290A DZ 2680 A1 DZ2680 A1 DZ 2680A1
Authority
DZ
Algeria
Prior art keywords
preparation
pharmaceutical composition
composition containing
novel process
thiazolidinedione derivative
Prior art date
Application number
DZ980290A
Other languages
English (en)
French (fr)
Inventor
Paul David James Blackler
Michael John Sasse
David C Lee
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Application granted granted Critical
Publication of DZ2680A1 publication Critical patent/DZ2680A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Obesity (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DZ980290A 1997-12-16 1998-12-15 Dérivé de thiazolidinedione nouveau procédé pour sa préparation et composition pharmaceutique le contenant. DZ2680A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9726568.0A GB9726568D0 (en) 1997-12-16 1997-12-16 Novel pharmaceutical

Publications (1)

Publication Number Publication Date
DZ2680A1 true DZ2680A1 (fr) 2005-02-20

Family

ID=10823694

Family Applications (1)

Application Number Title Priority Date Filing Date
DZ980290A DZ2680A1 (fr) 1997-12-16 1998-12-15 Dérivé de thiazolidinedione nouveau procédé pour sa préparation et composition pharmaceutique le contenant.

Country Status (37)

Country Link
US (2) US7045633B2 (sr)
EP (1) EP1045847A1 (sr)
JP (1) JP2002508372A (sr)
KR (1) KR100549143B1 (sr)
CN (3) CN101412714A (sr)
AP (1) AP1441A (sr)
AR (2) AR017213A1 (sr)
AU (1) AU2272399A (sr)
BG (1) BG64905B1 (sr)
BR (1) BR9813604A (sr)
CA (1) CA2314965A1 (sr)
CO (1) CO4990927A1 (sr)
CZ (1) CZ299970B6 (sr)
DZ (1) DZ2680A1 (sr)
EA (1) EA002355B1 (sr)
EG (2) EG21417A (sr)
GB (1) GB9726568D0 (sr)
HR (1) HRP20000405A2 (sr)
HU (1) HUP0100500A3 (sr)
ID (1) ID24744A (sr)
IL (1) IL136381A (sr)
IN (1) IN190821B (sr)
MA (1) MA26582A1 (sr)
MY (1) MY135770A (sr)
NO (1) NO317253B1 (sr)
NZ (1) NZ504704A (sr)
OA (1) OA11634A (sr)
PE (1) PE20000057A1 (sr)
PL (1) PL341147A1 (sr)
RS (1) RS50079B (sr)
SK (1) SK286197B6 (sr)
TR (2) TR200001798T2 (sr)
TW (1) TW467913B (sr)
UA (1) UA63980C2 (sr)
UY (2) UY25305A1 (sr)
WO (1) WO1999031094A1 (sr)
ZA (1) ZA9811505B (sr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9909041D0 (en) * 1999-04-20 1999-06-16 Smithkline Beecham Plc Novel pharmaceutical
US20040248945A1 (en) 1999-04-23 2004-12-09 Smithkline Beecham P.L.C. Thiazolidinedione derivative and its use as antidiabetic
DZ3164A1 (fr) * 1999-04-23 2000-11-02 Smithkline Beecham Plc Nouvel agent pharmaceutique.
CZ20013799A3 (cs) 1999-04-23 2002-04-17 Smithkline Beecham Plc Nový léčivý přípravek
GB0014005D0 (en) * 2000-06-08 2000-08-02 Smithkline Beecham Plc Novel pharmaceutical
GB0021784D0 (en) * 2000-09-05 2000-10-18 Smithkline Beecham Plc Novel pharmaceutical
GB0021978D0 (en) * 2000-09-07 2000-10-25 Smithkline Beecham Plc Novel pharmaceutical
WO2003050112A1 (en) * 2001-12-13 2003-06-19 Smithkline Beecham Plc Toluenesulfonate hydrates of a thiazolidinedione derivative
AU2002352391A1 (en) * 2001-12-13 2003-06-23 Smithkline Beecham Plc A 5(-4-(2-(n-methyl-n-(2-pyridil)amino)ethoxy)benzyl)thiazolidine-2,4-dione (i) 10-camphorsulphonic acid salt and use against diabetes mellitus
GB0129876D0 (en) * 2001-12-13 2002-02-06 Smithkline Beecham Plc Novel pharmaceutical
WO2003053962A1 (en) * 2001-12-20 2003-07-03 Smithkline Beecham Plc 5- (4- (2- (n-methyl-n- (2-pyridyl) amino) ethoxy) benzyl) thiazolidine-2, 4-dione malic acid salt and use against diabetes mellitus
GB0130511D0 (en) * 2001-12-20 2002-02-06 Smithkline Beecham Plc Novel pharmaceutical
GB2405403A (en) * 2003-08-29 2005-03-02 Cipla Ltd Rosiglitazone maleate of particular polymorphic forms and methods of preparing rosiglitazone free base
ITMI20041537A1 (it) * 2004-07-28 2004-10-28 Chemi Spa Nuova forma polimorfa del rosiglitazone maleato
CZ298424B6 (cs) * 2005-05-24 2007-09-26 Zentiva, A. S. Zpusob krystalizace rosiglitazonu a jeho derivátuze smesných rozpouštedel
EP2184055A1 (en) 2008-11-07 2010-05-12 LEK Pharmaceuticals d.d. Process for preparing solid dosage forms of rosiglitazone maleate

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR240698A1 (es) * 1985-01-19 1990-09-28 Takeda Chemical Industries Ltd Procedimiento para preparar compuestos de 5-(4-(2-(5-etil-2-piridil)-etoxi)benzil)-2,4-tiazolidindiona y sus sales
US4812570A (en) * 1986-07-24 1989-03-14 Takeda Chemical Industries, Ltd. Method for producing thiazolidinedione derivatives
ES2137915T3 (es) 1987-09-04 2000-01-01 Beecham Group Plc Derivados de tiazolidindiona sustituida.
GB8820389D0 (en) * 1988-08-26 1988-09-28 Beecham Group Plc Novel compounds
GB9124513D0 (en) 1991-11-19 1992-01-08 Smithkline Beecham Plc Novel process
WO1994005669A1 (en) 1992-08-28 1994-03-17 Merck & Co., Inc. Cationic-2-heteroarylphenyl-carbapenem antibacterial agents
GB9218830D0 (en) * 1992-09-05 1992-10-21 Smithkline Beecham Plc Novel compounds
US5741803A (en) 1992-09-05 1998-04-21 Smithkline Beecham Plc Substituted thiazolidinedionle derivatives
TW245716B (sr) * 1992-12-28 1995-04-21 Takeda Pharm Industry Co
DE4404198A1 (de) 1994-02-10 1995-08-17 Henkel Kgaa 2-Fluor-6-nitroaniline
GB9726563D0 (en) 1997-12-16 1998-02-11 Smithkline Beecham Plc Novel pharmaceutical
US20020137940A1 (en) 1997-12-16 2002-09-26 Smithkline Beecham P.L.C. 5-[4-[2-(N-methyl-N-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2, 4-dione, maleic acid salt, hydrate as pharmaceutical
US6664278B2 (en) * 1997-12-16 2003-12-16 Smithkline Beecham P.L.C. Hydrate of 5-[4-[2-(N-methyl-N-(2-pyridil)amino)ethoxy]benzyl]thiazolidine-2,4-dione maleic acid salt
GB9726566D0 (en) 1997-12-16 1998-02-11 Smithkline Beecham Plc Novel pharmaceutical
CZ432299A3 (cs) * 1998-06-02 2000-08-16 Smithkline Beecham Plc Kompozice obsahující 5-[4-[2-(N-methyl-N-(2- pyridyI)amino)ethoxy]benzyl]thiazolidin-2,4-dion
CO5170421A1 (es) 1999-04-23 2002-06-27 Smithkline Beecham Plc Nuevo compuesto farmaceutico maleico
CZ20013799A3 (cs) 1999-04-23 2002-04-17 Smithkline Beecham Plc Nový léčivý přípravek
DZ3164A1 (fr) 1999-04-23 2000-11-02 Smithkline Beecham Plc Nouvel agent pharmaceutique.

Also Published As

Publication number Publication date
CN101412713A (zh) 2009-04-22
IN190821B (sr) 2003-08-23
JP2002508372A (ja) 2002-03-19
WO1999031094A1 (en) 1999-06-24
YU36200A (sh) 2003-12-31
TR199802626A2 (xx) 1999-10-21
CA2314965A1 (en) 1999-06-24
US7045633B2 (en) 2006-05-16
RS50079B (sr) 2009-01-22
EG21417A (en) 2001-10-31
BG104595A (en) 2001-02-28
NO20003068D0 (no) 2000-06-15
UY25305A1 (es) 2000-12-29
BG64905B1 (bg) 2006-08-31
HUP0100500A3 (en) 2002-08-28
EG23694A (en) 2007-05-15
NO20003068L (no) 2000-06-15
CN1281454A (zh) 2001-01-24
AP1441A (en) 2005-07-30
MY135770A (en) 2008-06-30
CO4990927A1 (es) 2000-12-26
NO317253B1 (no) 2004-09-27
KR100549143B1 (ko) 2006-02-03
HUP0100500A2 (hu) 2002-05-29
EA200000655A1 (ru) 2000-12-25
US20060189659A1 (en) 2006-08-24
SK286197B6 (sk) 2008-05-06
ZA9811505B (en) 2000-11-06
HRP20000405A2 (en) 2000-12-31
EP1045847A1 (en) 2000-10-25
GB9726568D0 (en) 1998-02-11
IL136381A0 (en) 2001-06-14
US20040097553A1 (en) 2004-05-20
PL341147A1 (en) 2001-03-26
PE20000057A1 (es) 2000-03-09
UA63980C2 (en) 2004-02-16
BR9813604A (pt) 2000-10-10
NZ504704A (en) 2003-03-28
AR017430A1 (es) 2001-09-05
TR199802626A3 (tr) 1999-10-21
CZ299970B6 (cs) 2009-01-07
KR20010033142A (ko) 2001-04-25
CN101412714A (zh) 2009-04-22
CZ20002205A3 (cs) 2000-11-15
SK9102000A3 (en) 2001-01-18
TW467913B (en) 2001-12-11
UY25310A1 (es) 1999-07-19
AU2272399A (en) 1999-07-05
OA11634A (en) 2004-11-22
TR200001798T2 (tr) 2000-11-21
ID24744A (id) 2000-08-03
EA002355B1 (ru) 2002-04-25
AR017213A1 (es) 2001-08-22
AP2000001830A0 (en) 2000-06-30
MA26582A1 (fr) 2004-12-20
IL136381A (en) 2003-09-17

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