DZ3042A1 - Dérivés d'isothiazole nouveaux, procédé pour leur préparation et compositions pharmaceutiques les contenant. - Google Patents

Dérivés d'isothiazole nouveaux, procédé pour leur préparation et compositions pharmaceutiques les contenant.

Info

Publication number
DZ3042A1
DZ3042A1 DZ000085A DZ000085A DZ3042A1 DZ 3042 A1 DZ3042 A1 DZ 3042A1 DZ 000085 A DZ000085 A DZ 000085A DZ 000085 A DZ000085 A DZ 000085A DZ 3042 A1 DZ3042 A1 DZ 3042A1
Authority
DZ
Algeria
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
isothiazole derivatives
new
Prior art date
Application number
DZ000085A
Other languages
English (en)
Inventor
Thomas George Gant
Mark Cari Noe
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of DZ3042A1 publication Critical patent/DZ3042A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
    • C07D275/03—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/44—Oxygen and nitrogen or sulfur and nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
DZ000085A 1999-05-19 2000-05-17 Dérivés d'isothiazole nouveaux, procédé pour leur préparation et compositions pharmaceutiques les contenant. DZ3042A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US13493399P 1999-05-19 1999-05-19

Publications (1)

Publication Number Publication Date
DZ3042A1 true DZ3042A1 (fr) 2004-03-27

Family

ID=22465672

Family Applications (1)

Application Number Title Priority Date Filing Date
DZ000085A DZ3042A1 (fr) 1999-05-19 2000-05-17 Dérivés d'isothiazole nouveaux, procédé pour leur préparation et compositions pharmaceutiques les contenant.

Country Status (21)

Country Link
US (1) US6380214B1 (fr)
EP (1) EP1187826B1 (fr)
JP (2) JP3692041B2 (fr)
AR (1) AR029634A1 (fr)
AT (1) ATE349440T1 (fr)
AU (1) AU4137400A (fr)
BR (1) BR0010746A (fr)
CA (1) CA2374247C (fr)
CO (1) CO5170417A1 (fr)
DE (1) DE60032601T2 (fr)
DZ (1) DZ3042A1 (fr)
ES (1) ES2276681T3 (fr)
GT (1) GT200000069A (fr)
HN (1) HN2000000051A (fr)
MA (1) MA26733A1 (fr)
MX (1) MXPA01011920A (fr)
PA (1) PA8494101A1 (fr)
PE (1) PE20010152A1 (fr)
TN (1) TNSN00104A1 (fr)
UY (1) UY26143A1 (fr)
WO (1) WO2000071532A1 (fr)

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WO2001057034A1 (fr) 2000-02-07 2001-08-09 Bristol-Myers Squibb Co. Inhibiteurs 3-aminopyrazole des kinases dependantes des cyclines
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US7102009B2 (en) 2001-01-12 2006-09-05 Amgen Inc. Substituted amine derivatives and methods of use
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SE0102617D0 (sv) * 2001-07-25 2001-07-25 Astrazeneca Ab Novel compounds
SE0102616D0 (sv) * 2001-07-25 2001-07-25 Astrazeneca Ab Novel compounds
US6924276B2 (en) 2001-09-10 2005-08-02 Warner-Lambert Company Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors
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US20030216396A1 (en) 2002-02-11 2003-11-20 Bayer Corporation Pyridine, quinoline, and isoquinoline N-oxides as kinase inhibitors
US6989451B2 (en) * 2002-06-04 2006-01-24 Valeant Research & Development Heterocyclic compounds and uses thereof
AU2003232551A1 (en) * 2002-06-13 2003-12-31 Qlt Inc. Methods of using isothiazole derivatives to treat cancer or inflammation
AU2003248896B2 (en) * 2002-07-09 2010-04-22 Fasgen, Llc Methods of treating microbial infections in humans and animals
SG169236A1 (en) * 2002-07-09 2011-03-30 Fasgen Inc Novel compunds, pharmaceutical compositions containing same, and methods of use for same
AU2003281664A1 (en) * 2002-07-25 2004-02-16 Pfizer Products Inc. Isothiazole derivatives useful as anticancer agents
US7626031B2 (en) * 2002-11-15 2009-12-01 Symphony Evolution, Inc. Substituted 3-(diarylmethylene)indolin-2-ones and methods of their use
PT1569929E (pt) 2002-12-10 2010-06-18 Virochem Pharma Inc Compostos e métodos para o tratamento ou prevenção de infecções por flavivírus
SE0300091D0 (sv) * 2003-01-15 2003-01-15 Astrazeneca Ab Novel compounds
SE0300092D0 (sv) * 2003-01-15 2003-01-15 Astrazeneca Ab Novel compounds
WO2004078723A1 (fr) * 2003-03-07 2004-09-16 Santen Pharmaceutical Co. Ltd. Nouveau compose comprenant un groupe 4-pyridylalkylthio utilise comme substitutif
CA2526617C (fr) 2003-05-20 2015-04-28 Bayer Pharmaceuticals Corporation Diaryl-urees presentant une activite d'inhibition des kinases
UA84156C2 (ru) 2003-07-23 2008-09-25 Байер Фармасьютикалс Корпорейшн Фторозамещённая омега-карбоксиарилдифенилмочевина для лечения и профилактики болезней и состояний
JP4626353B2 (ja) * 2004-02-17 2011-02-09 参天製薬株式会社 置換又は無置換アミノ基を導入した４−ピリジルアルキルチオ基を有する新規環式化合物
PL1717229T3 (pl) * 2004-02-17 2011-11-30 Santen Pharmaceutical Co Ltd Nowy cykliczny związek mający grupę 4-pirydyloalkilotiolową z wprowadzoną do niej (nie)podstawioną grupą aminową
ES2368153T3 (es) * 2004-02-17 2011-11-14 Santen Pharmaceutical Co., Ltd. Nuevo compuesto cíclico que presenta un grupo 4-piridilalquiltio que presenta amino (no) sustituido introducido en el mismo.
AU2005223483B2 (en) 2004-03-18 2009-04-23 Zoetis Llc N-(1-arylpyrazol-4l)sulfonamides and their use as parasiticides
EP1751139B1 (fr) 2004-04-30 2011-07-27 Bayer HealthCare LLC Derives de pyrazolyl uree substitues utiles dans le traitement du cancer
BRPI0514667A (pt) * 2004-08-26 2008-06-17 Pfizer Prod Inc processos para a preparação de derivados de isotiazol
JP4585978B2 (ja) * 2005-03-03 2010-11-24 参天製薬株式会社 キノリルアルキルチオ基を有する新規環式化合物
EA016071B1 (ru) * 2005-05-13 2012-01-30 Вирокем Фарма Инк. Соединения и способы лечения или предотвращения флавивирусных инфекций
US7932390B2 (en) 2006-06-29 2011-04-26 Hoffman-La Roche Inc. Substituted thieno[3,2-C]pyridine carboxylic acid derivatives
RS52874B (en) 2006-11-15 2013-12-31 Vertex Pharmaceuticals Incorporated THYOPHEN ANALYSIS FOR THE TREATMENT OR PREVENTION OF FLAVIVIRUS INFECTIONS
EP2116530B1 (fr) * 2007-02-26 2012-11-14 Santen Pharmaceutical Co., Ltd Nouveau dérivé de pyrrole ayant un groupe uréide et un groupe aminocarbonyle comme substituants
WO2008153042A1 (fr) * 2007-06-11 2008-12-18 Kyowa Hakko Kirin Co., Ltd. Agent antitumoral
MX2010001636A (es) 2007-08-14 2010-03-15 Hoffmann La Roche Derivados de pirazolo[3,4-d]-pirimidina como agentes antiproliferativos.
JP2012531433A (ja) * 2009-06-25 2012-12-10 メドリューション リミテッド キナーゼ阻害剤としての置換複素環式化合物とその用法
CN104302640A (zh) 2012-03-16 2015-01-21 埃克希金医药品有限公司 3,5-二氨基吡唑激酶抑制剂
NZ631142A (en) 2013-09-18 2016-03-31 Axikin Pharmaceuticals Inc Pharmaceutically acceptable salts of 3,5-diaminopyrazole kinase inhibitors
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DE3541631A1 (de) * 1985-11-26 1987-05-27 Bayer Ag Selektiv-fungizide verwendung von thienylharnstoff-derivaten
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Also Published As

Publication number Publication date
PA8494101A1 (es) 2003-09-05
DE60032601D1 (de) 2007-02-08
JP3692041B2 (ja) 2005-09-07
CO5170417A1 (es) 2002-06-27
CA2374247A1 (fr) 2000-11-30
MXPA01011920A (es) 2002-05-06
HN2000000051A (es) 2001-02-02
EP1187826A1 (fr) 2002-03-20
CA2374247C (fr) 2008-01-22
GT200000069A (es) 2001-11-08
TNSN00104A1 (fr) 2005-11-10
BR0010746A (pt) 2002-02-13
MA26733A1 (fr) 2004-12-20
AU4137400A (en) 2000-12-12
PE20010152A1 (es) 2001-02-08
UY26143A1 (es) 2000-12-29
ATE349440T1 (de) 2007-01-15
JP2003500401A (ja) 2003-01-07
WO2000071532A1 (fr) 2000-11-30
EP1187826B1 (fr) 2006-12-27
US6380214B1 (en) 2002-04-30
ES2276681T3 (es) 2007-07-01
DE60032601T2 (de) 2007-11-15
AR029634A1 (es) 2003-07-10
JP2005008641A (ja) 2005-01-13

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