DOP2012000154A - COMPUESTOS N-ACILSULFONAMIDA QUE INHIBEN LA ACTIVIDAD DE LAS PROTEINAS ANTIAPOPTOTICAS Bcl2 Y SU USO EN LA FABRICACION DE UN MEDICAMENTO PARA EL TRATAMIENTO DEL CANCER Y DE ENFERMEDADES INMUNES Y AUTOINMUNES - Google Patents

COMPUESTOS N-ACILSULFONAMIDA QUE INHIBEN LA ACTIVIDAD DE LAS PROTEINAS ANTIAPOPTOTICAS Bcl2 Y SU USO EN LA FABRICACION DE UN MEDICAMENTO PARA EL TRATAMIENTO DEL CANCER Y DE ENFERMEDADES INMUNES Y AUTOINMUNES

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Publication number
DOP2012000154A
DOP2012000154A DO2012000154A DO2012000154A DOP2012000154A DO P2012000154 A DOP2012000154 A DO P2012000154A DO 2012000154 A DO2012000154 A DO 2012000154A DO 2012000154 A DO2012000154 A DO 2012000154A DO P2012000154 A DOP2012000154 A DO P2012000154A
Authority
DO
Dominican Republic
Prior art keywords
cancer
compounds
immune
inhibit
activity
Prior art date
Application number
DO2012000154A
Other languages
English (en)
Spanish (es)
Inventor
W Elmore Steven
J Souers Andrew
Bruncko Milan
Song Xiaohong
Wang Xilu
Wang Le
D Wendt Michael
Tao Zhi-Fu
Ding Hong
Hasvold Lisa
Hexamer Laura
J Mcclellan William
H Park Chang
M Petros Andrew
M Sullivan Gerard
T Wang Gary
A Mantei Robert
M Hansen Todd
Dai Yujia
A Doherty George
Kunzer Aaron
Park Cheol-Min
Original Assignee
Abbvie Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42463423&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DOP2012000154(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Abbvie Inc filed Critical Abbvie Inc
Publication of DOP2012000154A publication Critical patent/DOP2012000154A/es

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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/455—Nicotinic acids, e.g. niacin; Derivatives thereof, e.g. esters, amides
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    • A61K31/00—Medicinal preparations containing organic active ingredients
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    • A61K31/635—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
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DO2012000154A 2009-12-04 2012-06-01 COMPUESTOS N-ACILSULFONAMIDA QUE INHIBEN LA ACTIVIDAD DE LAS PROTEINAS ANTIAPOPTOTICAS Bcl2 Y SU USO EN LA FABRICACION DE UN MEDICAMENTO PARA EL TRATAMIENTO DEL CANCER Y DE ENFERMEDADES INMUNES Y AUTOINMUNES DOP2012000154A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US12/631,367 US20100160322A1 (en) 2008-12-04 2009-12-04 Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases

Publications (1)

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DOP2012000154A true DOP2012000154A (es) 2018-06-30

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US (5) US20100160322A1 (enExample)
EP (1) EP2507211B1 (enExample)
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CN (2) CN106397418A (enExample)
AR (1) AR076946A1 (enExample)
AU (1) AU2010326727B2 (enExample)
BR (1) BR112012012918A8 (enExample)
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