DOP2005000025A - Compuestos de heteroaril- y fenilsulfamoilo sustituidos - Google Patents

Compuestos de heteroaril- y fenilsulfamoilo sustituidos

Info

Publication number
DOP2005000025A
DOP2005000025A DO2005P000025A DO2005000025A DOP2005000025A DO P2005000025 A DOP2005000025 A DO P2005000025A DO 2005P000025 A DO2005P000025 A DO 2005P000025A DO 2005000025 A DO2005000025 A DO 2005000025A DO P2005000025 A DOP2005000025 A DO P2005000025A
Authority
DO
Dominican Republic
Prior art keywords
fenilsulfamoil
heteroaril
substituted compounds
compounds
heteroarilaminopirazolic
Prior art date
Application number
DO2005P000025A
Other languages
English (en)
Inventor
John Gordon Allen
Karin Briner
Michael Philip Cohen
Christopher Stanley Galka
Sarah Lynne Hellman
Maria Angeles Martinez
Mathew Robert Reinhard
Michael John Rodriguez
Roger Ryan Rotar
Michael Wade Tidwell
Andrew Caerwyn Williams
Deyi Zhang
Steven Armen Boyd
Richard Gerard Conway
Arundhati S Deo
Wai-Man Lee
Christopher Stephen Siedem
Ajay Singh
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34960729&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DOP2005000025(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of DOP2005000025A publication Critical patent/DOP2005000025A/es

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    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C311/21—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
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    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
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    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
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    • C07C323/23—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C323/46—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having at least one of the nitrogen atoms, not being part of nitro or nitroso groups, further bound to other hetero atoms
    • C07C323/49—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having at least one of the nitrogen atoms, not being part of nitro or nitroso groups, further bound to other hetero atoms to sulfur atoms
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    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
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    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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Abstract

LA PRESENTE INVENCION SE REFIERE A COMPUESTOS HETEROARILAMINOPIRAZOLICOS, A COMPOSICIONES FARMACEUTICAS Y A METODOS PARA EL TRATAMIENTO DE LA DIABETES Y TRASTORNOS RELACIONADOS.
DO2005P000025A 2004-03-10 2005-02-23 Compuestos de heteroaril- y fenilsulfamoilo sustituidos DOP2005000025A (es)

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US11/012,139 US7262318B2 (en) 2004-03-10 2004-12-16 Substituted heteroaryl- and phenylsulfamoyl compounds

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KR20070001173A (ko) 2007-01-03
MA28461B1 (fr) 2007-03-01
BRPI0508555A (pt) 2007-08-07
AR048260A1 (es) 2006-04-12
AP2006003714A0 (en) 2006-08-31
SV2005002047A (es) 2005-12-13
EP1725524A1 (en) 2006-11-29
NL1028519C2 (nl) 2006-06-22
IL177631A0 (en) 2006-12-31
EA200601442A1 (ru) 2007-02-27
CA2559035A1 (en) 2005-10-06
ECSP066834A (es) 2006-12-29
AU2005225628A1 (en) 2005-10-06
AU2005225628B2 (en) 2008-09-11
NO20064615L (no) 2006-12-07
PE20051147A1 (es) 2006-01-28
US20060258723A1 (en) 2006-11-16
PA8625701A1 (es) 2006-01-25
TW200610525A (en) 2006-04-01
US7262318B2 (en) 2007-08-28
WO2005092845A1 (en) 2005-10-06
UY28794A1 (es) 2005-10-31
DOP2005000034A (es) 2005-12-15
US20050228015A1 (en) 2005-10-13
NL1028519A1 (nl) 2005-09-13
JP2007528387A (ja) 2007-10-11

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