DK413783D0 - Fremgangsmade til fremstilling af 20-amino-macrolidderivater eller syreadditionssalte deraf - Google Patents

Fremgangsmade til fremstilling af 20-amino-macrolidderivater eller syreadditionssalte deraf

Info

Publication number
DK413783D0
DK413783D0 DK4137/83A DK413783A DK413783D0 DK 413783 D0 DK413783 D0 DK 413783D0 DK 4137/83 A DK4137/83 A DK 4137/83A DK 413783 A DK413783 A DK 413783A DK 413783 D0 DK413783 D0 DK 413783D0
Authority
DK
Denmark
Prior art keywords
amino
preparing
acid addition
addition salts
macrolide derivatives
Prior art date
Application number
DK4137/83A
Other languages
English (en)
Other versions
DK153555C (da
DK153555B (da
DK413783A (da
Inventor
Manuel Debono
Herbert Andrew Kirst
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of DK413783D0 publication Critical patent/DK413783D0/da
Publication of DK413783A publication Critical patent/DK413783A/da
Publication of DK153555B publication Critical patent/DK153555B/da
Application granted granted Critical
Publication of DK153555C publication Critical patent/DK153555C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Fodder In General (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK413783A 1982-09-13 1983-09-12 Analogifremgangsmaade til fremstilling af 20-amino-derivater af tylosin, desmycosin, macrosin eller lactenocin eller syreadditionssalte deraf DK153555C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US41724782A 1982-09-13 1982-09-13
US41724782 1982-09-13

Publications (4)

Publication Number Publication Date
DK413783D0 true DK413783D0 (da) 1983-09-12
DK413783A DK413783A (da) 1984-03-14
DK153555B DK153555B (da) 1988-07-25
DK153555C DK153555C (da) 1988-12-05

Family

ID=23653182

Family Applications (1)

Application Number Title Priority Date Filing Date
DK413783A DK153555C (da) 1982-09-13 1983-09-12 Analogifremgangsmaade til fremstilling af 20-amino-derivater af tylosin, desmycosin, macrosin eller lactenocin eller syreadditionssalte deraf

Country Status (34)

Country Link
EP (1) EP0103465B1 (da)
JP (1) JPS5973598A (da)
KR (1) KR850000961B1 (da)
AR (1) AR241595A1 (da)
AT (1) AT381707B (da)
AU (1) AU561147B2 (da)
BG (1) BG42675A3 (da)
CA (1) CA1243310A (da)
CS (1) CS259862B2 (da)
CY (1) CY1417A (da)
DD (1) DD210284A5 (da)
DE (1) DE3366097D1 (da)
DK (1) DK153555C (da)
EG (1) EG16287A (da)
ES (2) ES8604596A1 (da)
FI (1) FI73222C (da)
GB (1) GB2127017B (da)
GR (1) GR79067B (da)
HK (1) HK21888A (da)
HU (1) HU194271B (da)
IE (1) IE55916B1 (da)
IL (1) IL69666A (da)
LU (1) LU90240I2 (da)
MY (1) MY8700756A (da)
NL (1) NL950001I2 (da)
NZ (1) NZ205501A (da)
PH (1) PH23242A (da)
PL (2) PL142304B1 (da)
PT (1) PT77335B (da)
RO (1) RO89235A (da)
SG (1) SG99287G (da)
SU (1) SU1375135A3 (da)
UA (1) UA6045A1 (da)
ZA (1) ZA836741B (da)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS59181294A (ja) * 1983-03-30 1984-10-15 Satoshi Omura 抗生物質ptl−448とその誘導体およびそれらの製造方法
US4921947A (en) * 1986-03-31 1990-05-01 Eli Lilly And Company Process for preparing macrolide derivatives
US4820694A (en) * 1986-09-29 1989-04-11 Eli Lilly And Company Modifications of 3-O-demethylmycinose in macrocin and lactenocin
EP0262903A3 (en) * 1986-09-29 1988-11-02 Eli Lilly And Company New acyl derivatives of 20-modified tylosin and desmycosin compounds
US5354708A (en) * 1992-06-04 1994-10-11 Taskar Nikhil R Method of nitrogen doping of II-VI semiconductor compounds during epitaxial growth using an amine
TW226373B (da) * 1992-07-15 1994-07-11 Pfizer
ES2076107B1 (es) * 1993-09-20 1996-04-01 Pfizer Derivados de antibioticos macrolidos de anillos de 16 miembros.
AU3121095A (en) * 1994-09-22 1996-04-09 Pfizer Inc. Antibiotic macrolides
EP0778283A3 (en) * 1995-12-05 1998-01-28 Pfizer Inc. Antibiotic macrolides
US6605599B1 (en) 1997-07-08 2003-08-12 Bristol-Myers Squibb Company Epothilone derivatives
ZA991641B (en) * 1998-03-02 2000-09-01 Lilly Co Eli Treatment of viral disease in swine.
EP2019112A1 (en) 2007-07-26 2009-01-28 Intervet International BV Macrolide solid-state forms
PL2089408T3 (pl) 2006-07-28 2012-03-30 Intervet Int Bv Sposób syntezy makrolidu
WO2009075818A1 (en) * 2007-12-07 2009-06-18 Eisai R & D Management Co., Ltd. Intermediates and methods for making zearalenone macrolide analogs
PL2999707T3 (pl) * 2013-05-23 2018-09-28 Bayer Animal Health Gmbh Pochodne tylozynowe i sposób ich wytwarzania
CN103880903B (zh) * 2014-03-21 2016-06-15 烟台万润药业有限公司 一种泰乐菌素类大环内酯及其衍生物的制备方法
CN117304241B (zh) * 2023-11-30 2024-03-01 中国农业科学院饲料研究所 一种大环内酯类化合物及其制备方法与应用
CN117510561B (zh) * 2023-11-30 2024-04-02 中国农业科学院饲料研究所 一种泰乐菌素衍生物及其制备方法与应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE32839B1 (en) * 1967-12-04 1973-12-28 Lilly Co Eli Urea-antibiotic adducts and process for preparing the same
US4279896A (en) * 1980-06-23 1981-07-21 Schering Corporation Novel 20-imino macrolide antibacterial agents
JPS58146595A (ja) * 1982-02-25 1983-09-01 Satoshi Omura マクロライド系抗生物質

Also Published As

Publication number Publication date
JPS5973598A (ja) 1984-04-25
PL142251B1 (en) 1987-10-31
AU1871083A (en) 1984-03-22
GB8324044D0 (en) 1983-10-12
PT77335A (en) 1983-10-01
DK153555C (da) 1988-12-05
AR241595A1 (es) 1992-09-30
ES548472A0 (es) 1986-06-01
FI833229A (fi) 1984-03-14
SG99287G (en) 1988-09-23
BG42675A3 (en) 1988-01-15
CS665383A2 (en) 1988-04-15
EP0103465B1 (en) 1986-09-10
CA1243310A (en) 1988-10-18
HU194271B (en) 1988-01-28
DK153555B (da) 1988-07-25
PL250619A1 (en) 1985-07-30
PH23242A (en) 1989-06-06
ES525544A0 (es) 1986-02-01
KR850000961B1 (ko) 1985-07-02
FI833229A0 (fi) 1983-09-09
ES8604596A1 (es) 1986-02-01
NZ205501A (en) 1985-09-13
PL243718A1 (en) 1985-04-09
KR840005734A (ko) 1984-11-15
IE832131L (en) 1984-03-13
DK413783A (da) 1984-03-14
GR79067B (da) 1984-10-02
EP0103465A1 (en) 1984-03-21
MY8700756A (en) 1987-12-31
NL950001I1 (nl) 1995-02-16
DD210284A5 (de) 1984-06-06
AU561147B2 (en) 1987-04-30
UA6045A1 (uk) 1994-12-29
FI73222B (fi) 1987-05-29
RO89235A (ro) 1986-03-15
CY1417A (en) 1988-04-22
ZA836741B (en) 1984-04-25
HK21888A (en) 1988-03-31
JPH021840B2 (da) 1990-01-12
IE55916B1 (en) 1991-02-27
IL69666A (en) 1987-10-20
LU90240I2 (fr) 1998-07-06
ES8607336A1 (es) 1986-06-01
AT381707B (de) 1986-11-25
NL950001I2 (nl) 1997-05-01
GB2127017A (en) 1984-04-04
SU1375135A3 (ru) 1988-02-15
CS259862B2 (en) 1988-11-15
FI73222C (fi) 1987-09-10
IL69666A0 (en) 1983-12-30
ATA320683A (de) 1986-04-15
DE3366097D1 (en) 1986-10-16
HUT35272A (en) 1985-06-28
PL142304B1 (en) 1987-10-31
GB2127017B (en) 1986-01-15
PT77335B (en) 1986-05-19
EG16287A (en) 1987-04-30

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Legal Events

Date Code Title Description
CTFF Application for supplementary protection certificate (spc) filed

Spc suppl protection certif: CA 2000 00001

Filing date: 20000104

Extension date: 20050625

PUP Patent expired