DK332583A - N-methyl-11-aza-10-deoxo-10-dihydroerythromycin a, mellemprodukter herfor og fremgangsmaader til fremstilling deraf - Google Patents

N-methyl-11-aza-10-deoxo-10-dihydroerythromycin a, mellemprodukter herfor og fremgangsmaader til fremstilling deraf Download PDF

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Publication number
DK332583A
DK332583A DK332583A DK332583A DK332583A DK 332583 A DK332583 A DK 332583A DK 332583 A DK332583 A DK 332583A DK 332583 A DK332583 A DK 332583A DK 332583 A DK332583 A DK 332583A
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Prior art keywords
dihydroerythromycine
deoxo
aza
intermediates
procedures
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DK332583A
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DK158229B (da
DK332583D0 (da
DK158229C (da
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Gene Michael Bright
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Pfizer
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK332583A 1982-07-19 1983-07-19 Analogifremgangsmaade til fremstilling af 9-deoxo-9a-methyl-9a-aza-9a-homoerythromycin a eller alkanoyl-derivater deraf eller farmaceutisk acceptable syreadditionssalte deraf og n,n'-dioxidet deraf til anvendelse som udgangsmateriale ved fremgangsmaaden DK158229C (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US39940182A 1982-07-19 1982-07-19
US39940182 1982-07-19
US44198182 1982-11-15
US06/441,981 US4474768A (en) 1982-07-19 1982-11-15 N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor

Publications (4)

Publication Number Publication Date
DK332583D0 DK332583D0 (da) 1983-07-19
DK332583A true DK332583A (da) 1984-01-20
DK158229B DK158229B (da) 1990-04-16
DK158229C DK158229C (da) 1990-09-24

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Family Applications (1)

Application Number Title Priority Date Filing Date
DK332583A DK158229C (da) 1982-07-19 1983-07-19 Analogifremgangsmaade til fremstilling af 9-deoxo-9a-methyl-9a-aza-9a-homoerythromycin a eller alkanoyl-derivater deraf eller farmaceutisk acceptable syreadditionssalte deraf og n,n'-dioxidet deraf til anvendelse som udgangsmateriale ved fremgangsmaaden

Country Status (15)

Country Link
US (1) US4474768A (da)
EP (1) EP0101186B1 (da)
JP (1) JPH01193292A (da)
AU (1) AU540056B2 (da)
CA (1) CA1202963A (da)
DE (1) DE3367395D1 (da)
DK (1) DK158229C (da)
FI (1) FI832606A (da)
HU (1) HU196426B (da)
IE (1) IE55365B1 (da)
IL (1) IL69265A (da)
NO (1) NO160261C (da)
NZ (1) NZ204938A (da)
PH (1) PH18054A (da)
PT (1) PT77062B (da)

Families Citing this family (153)

* Cited by examiner, † Cited by third party
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EP0101186A1 (en) 1984-02-22
HU196426B (en) 1988-11-28
CA1202963A (en) 1986-04-08
PT77062B (en) 1986-04-09
FI832606A (fi) 1984-01-20
NO160261C (no) 1989-03-29
PH18054A (en) 1985-03-18
IE55365B1 (en) 1990-08-29
DK158229B (da) 1990-04-16
DE3367395D1 (en) 1986-12-11
DK332583D0 (da) 1983-07-19
IL69265A0 (en) 1983-11-30
EP0101186B1 (en) 1986-11-05
US4474768A (en) 1984-10-02
NO832616L (no) 1984-01-20
DK158229C (da) 1990-09-24
IE831667L (en) 1984-01-19
FI832606A0 (fi) 1983-07-18
IL69265A (en) 1986-08-31
NZ204938A (en) 1986-04-11
AU1692383A (en) 1984-01-26
JPH01193292A (ja) 1989-08-03
AU540056B2 (en) 1984-11-01
PT77062A (en) 1983-08-01
NO160261B (no) 1988-12-19

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