DK3313832T3 - 3-tetrazolyl-benzen-1,2-disulfonamidderivater som metallo-beta- lactamase-hæmmere - Google Patents

3-tetrazolyl-benzen-1,2-disulfonamidderivater som metallo-beta- lactamase-hæmmere Download PDF

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DK3313832T3
DK3313832T3 DK16734151.0T DK16734151T DK3313832T3 DK 3313832 T3 DK3313832 T3 DK 3313832T3 DK 16734151 T DK16734151 T DK 16734151T DK 3313832 T3 DK3313832 T3 DK 3313832T3
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disulphonamide
metallo
tetrazolyl
beta
benzene
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DK16734151.0T
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Inventor
Frank Bennett
Jinlong Jiang
Alexander Pasternak
Shuzhi Dong
Xin Gu
Jack D Scott
Haiqun Tang
Zhiqiang Zhao
Yuhua Huang
Dexi Yang
Katherine Young
Li Xiao
Zhibo Zhang
Jianmin Fu
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Merck Sharp & Dohme
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid, pantothenic acid
    • A61K31/198—Alpha-aminoacids, e.g. alanine, edetic acids [EDTA]
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