DK1940821T3 - Nye vanilloid-receptorligander og deres anvendelse til fremstilling af lægemidler. - Google Patents

Nye vanilloid-receptorligander og deres anvendelse til fremstilling af lægemidler.

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Publication number
DK1940821T3
DK1940821T3 DK06806372.6T DK06806372T DK1940821T3 DK 1940821 T3 DK1940821 T3 DK 1940821T3 DK 06806372 T DK06806372 T DK 06806372T DK 1940821 T3 DK1940821 T3 DK 1940821T3
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Prior art keywords
drugs
manufacture
receptor ligands
vanilloid receptor
novel vanilloid
Prior art date
Application number
DK06806372.6T
Other languages
English (en)
Inventor
Hyung Chul Ryu
Robert Frank
Thomas Christoph
Derek John Saunders
Jeewoo Lee
Gregor Bahrenberg
Vry Jean De
Bernd Sundermann
Klaus Schiene
Original Assignee
Gruenenthal Gmbh
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Filing date
Publication date
Priority claimed from DE200510050408 external-priority patent/DE102005050408A1/de
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Application granted granted Critical
Publication of DK1940821T3 publication Critical patent/DK1940821T3/da

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    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
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KR20080067674A (ko) 2008-07-21
CN103382176A (zh) 2013-11-06
EP1940821B1 (de) 2013-03-20
WO2007045462A2 (de) 2007-04-26
EP2388258A1 (de) 2011-11-23

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