DK171276B1 - 1-Substituerede 7-(N-diazabicycloalkyl)-6-fluor-1,4-dihydro-4-oxo-quinolin-3-carboxylsyre-forbindelser, disse forbindelser til anvendelse som lægemidler og antibaktielle præparater indeholdende disse forbindelser - Google Patents

1-Substituerede 7-(N-diazabicycloalkyl)-6-fluor-1,4-dihydro-4-oxo-quinolin-3-carboxylsyre-forbindelser, disse forbindelser til anvendelse som lægemidler og antibaktielle præparater indeholdende disse forbindelser Download PDF

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Publication number
DK171276B1
DK171276B1 DK445886A DK445886A DK171276B1 DK 171276 B1 DK171276 B1 DK 171276B1 DK 445886 A DK445886 A DK 445886A DK 445886 A DK445886 A DK 445886A DK 171276 B1 DK171276 B1 DK 171276B1
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Prior art keywords
compounds
oxo
carboxylic acid
dihydro
diazabicyclo
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DK445886A
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Danish (da)
English (en)
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DK445886D0 (da
DK445886A (da
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Martin Raymond Jefson
Paul Robert Mcguirk
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Pfizer
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Publication of DK445886A publication Critical patent/DK445886A/da
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Publication of DK171276B1 publication Critical patent/DK171276B1/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
  • Materials For Photolithography (AREA)
DK445886A 1985-09-18 1986-09-17 1-Substituerede 7-(N-diazabicycloalkyl)-6-fluor-1,4-dihydro-4-oxo-quinolin-3-carboxylsyre-forbindelser, disse forbindelser til anvendelse som lægemidler og antibaktielle præparater indeholdende disse forbindelser DK171276B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US77747185A 1985-09-18 1985-09-18
US77747185 1985-09-18

Publications (3)

Publication Number Publication Date
DK445886D0 DK445886D0 (da) 1986-09-17
DK445886A DK445886A (da) 1987-05-27
DK171276B1 true DK171276B1 (da) 1996-08-19

Family

ID=25110350

Family Applications (1)

Application Number Title Priority Date Filing Date
DK445886A DK171276B1 (da) 1985-09-18 1986-09-17 1-Substituerede 7-(N-diazabicycloalkyl)-6-fluor-1,4-dihydro-4-oxo-quinolin-3-carboxylsyre-forbindelser, disse forbindelser til anvendelse som lægemidler og antibaktielle præparater indeholdende disse forbindelser

Country Status (42)

Country Link
US (3) US4775668A (el)
EP (1) EP0215650B1 (el)
JP (1) JPH0798819B2 (el)
KR (1) KR870000961B1 (el)
CN (1) CN1014789B (el)
AT (1) ATE72245T1 (el)
AU (1) AU576302B2 (el)
BG (2) BG49275A3 (el)
CA (1) CA1340734C (el)
CY (1) CY1774A (el)
CZ (1) CZ277825B6 (el)
DD (1) DD259190A5 (el)
DE (2) DE19675019I2 (el)
DK (1) DK171276B1 (el)
EG (1) EG18184A (el)
ES (1) ES2001428A6 (el)
FI (1) FI87565C (el)
GR (1) GR862363B (el)
HK (1) HK132795A (el)
HU (1) HU200462B (el)
IE (1) IE58966B1 (el)
IL (1) IL80033A (el)
IN (1) IN166416B (el)
LU (1) LU90356I2 (el)
MA (1) MA20770A1 (el)
MW (1) MW5886A1 (el)
MX (1) MX173358B (el)
MY (1) MY102518A (el)
NO (1) NO170335C (el)
NZ (1) NZ217614A (el)
OA (1) OA08410A (el)
PH (2) PH24048A (el)
PL (1) PL149987B1 (el)
PT (1) PT83388B (el)
SG (1) SG28094G (el)
SK (1) SK667886A3 (el)
SU (1) SU1482531A3 (el)
UA (1) UA6340A1 (el)
YU (1) YU45024B (el)
ZA (1) ZA867063B (el)
ZM (1) ZM8586A1 (el)
ZW (1) ZW19386A1 (el)

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US20050234095A1 (en) 2004-03-25 2005-10-20 Wenge Xie Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof
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Also Published As

Publication number Publication date
EP0215650A2 (en) 1987-03-25
IL80033A0 (en) 1986-12-31
AU576302B2 (en) 1988-08-18
NZ217614A (en) 1989-11-28
HUT43070A (en) 1987-09-28
EG18184A (en) 1992-12-30
NO863718L (no) 1987-03-19
FI863756A0 (fi) 1986-09-17
YU161786A (en) 1987-10-31
NO170335C (no) 1992-10-07
FI863756A (fi) 1987-03-19
AU6276886A (en) 1987-03-19
IE862479L (en) 1987-03-18
FI87565C (fi) 1993-01-25
PT83388B (pt) 1989-05-12
PL261410A1 (en) 1987-11-16
PL149987B1 (en) 1990-04-30
CZ277825B6 (en) 1993-06-16
ZW19386A1 (en) 1986-12-10
DK445886D0 (da) 1986-09-17
SU1482531A3 (ru) 1989-05-23
MW5886A1 (en) 1987-12-09
SK278605B6 (en) 1997-11-05
CZ667886A3 (en) 1993-02-17
EP0215650A3 (en) 1987-12-02
BG61091B2 (bg) 1996-10-31
JPH0798819B2 (ja) 1995-10-25
NO170335B (no) 1992-06-29
SG28094G (en) 1994-10-28
NO863718D0 (no) 1986-09-17
MX173358B (es) 1994-02-23
MA20770A1 (fr) 1987-04-01
KR870003106A (ko) 1987-04-15
OA08410A (fr) 1988-06-30
LU90356I2 (fr) 1999-04-26
FI87565B (fi) 1992-10-15
CN1014789B (zh) 1991-11-20
PT83388A (en) 1986-10-01
DE3683711D1 (de) 1992-03-12
IE58966B1 (en) 1993-12-01
MX3751A (es) 1993-09-01
US4775668A (en) 1988-10-04
JPS62103083A (ja) 1987-05-13
EP0215650B1 (en) 1992-01-29
HK132795A (en) 1995-09-01
DE19675019I2 (de) 2004-01-29
YU45024B (en) 1991-06-30
US5091383A (en) 1992-02-25
US4861779A (en) 1989-08-29
ATE72245T1 (de) 1992-02-15
ZA867063B (en) 1988-04-27
IN166416B (el) 1990-05-05
ZM8586A1 (en) 1987-03-27
PH24048A (en) 1990-03-05
SK667886A3 (en) 1997-11-05
ES2001428A6 (es) 1988-05-16
MY102518A (en) 1992-07-31
DD259190A5 (de) 1988-08-17
KR870000961B1 (ko) 1987-05-14
CN86106385A (zh) 1987-06-03
IL80033A (en) 1992-05-25
GR862363B (en) 1987-01-19
DK445886A (da) 1987-05-27
HU200462B (en) 1990-06-28
BG49275A3 (en) 1991-09-16
PH25338A (en) 1991-04-30
UA6340A1 (uk) 1994-12-29
CY1774A (en) 1995-10-20
CA1340734C (en) 1999-09-14

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