DK170817B1 - Quinazolinderivater, fremgangsmåder til deres fremstilling samt deres anvendelse som insekticider, acaricider og fungicider - Google Patents

Quinazolinderivater, fremgangsmåder til deres fremstilling samt deres anvendelse som insekticider, acaricider og fungicider Download PDF

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Publication number
DK170817B1
DK170817B1 DK037089A DK37089A DK170817B1 DK 170817 B1 DK170817 B1 DK 170817B1 DK 037089 A DK037089 A DK 037089A DK 37089 A DK37089 A DK 37089A DK 170817 B1 DK170817 B1 DK 170817B1
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DK
Denmark
Prior art keywords
compound
alkyl
formula
phenyl
quinazoline
Prior art date
Application number
DK037089A
Other languages
Danish (da)
English (en)
Other versions
DK37089A (da
DK37089D0 (da
Inventor
Barry Allen Dreikorn
Robert George Suhr
Glen Phil Jourdan
Ian Glaisby Wright
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of DK37089D0 publication Critical patent/DK37089D0/da
Publication of DK37089A publication Critical patent/DK37089A/da
Application granted granted Critical
Publication of DK170817B1 publication Critical patent/DK170817B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/74—Quinazolines; Hydrogenated quinazolines with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached to ring carbon atoms of the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/95—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK037089A 1988-01-29 1989-01-27 Quinazolinderivater, fremgangsmåder til deres fremstilling samt deres anvendelse som insekticider, acaricider og fungicider DK170817B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US15010288A 1988-01-29 1988-01-29
US15010288 1988-01-29

Publications (3)

Publication Number Publication Date
DK37089D0 DK37089D0 (da) 1989-01-27
DK37089A DK37089A (da) 1989-07-30
DK170817B1 true DK170817B1 (da) 1996-01-29

Family

ID=22533128

Family Applications (1)

Application Number Title Priority Date Filing Date
DK037089A DK170817B1 (da) 1988-01-29 1989-01-27 Quinazolinderivater, fremgangsmåder til deres fremstilling samt deres anvendelse som insekticider, acaricider og fungicider

Country Status (21)

Country Link
EP (1) EP0326329B1 (xx)
JP (1) JP2776864B2 (xx)
KR (1) KR0129754B1 (xx)
CN (1) CN1052379C (xx)
AR (1) AR246516A1 (xx)
AT (1) ATE172725T1 (xx)
AU (1) AU632994B2 (xx)
BR (1) BR8900365A (xx)
DE (1) DE68928841T2 (xx)
DK (1) DK170817B1 (xx)
EG (1) EG19187A (xx)
ES (1) ES2121737T3 (xx)
FI (1) FI890421A (xx)
HU (1) HU207643B (xx)
IL (1) IL89027A (xx)
MX (1) MX14663A (xx)
MY (1) MY103804A (xx)
NZ (1) NZ227733A (xx)
PT (1) PT89506B (xx)
TR (1) TR27343A (xx)
ZA (1) ZA89623B (xx)

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* Cited by examiner, † Cited by third party
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IL89029A (en) * 1988-01-29 1993-01-31 Lilly Co Eli Fungicidal quinoline and cinnoline derivatives, compositions containing them, and fungicidal methods of using them
IL89028A0 (en) * 1988-01-29 1989-08-15 Lilly Co Eli Quinoline,quinazoline and cinnoline derivatives
GT198900005A (es) * 1988-01-29 1990-07-17 Quinolinas y cinolinas substituidas.
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CA2015981A1 (en) * 1989-05-10 1990-11-10 Thomas H. Brown Compounds
BR9101256A (pt) * 1990-03-30 1991-11-05 Dowelanco Composto,composicao fungicida,processo fungicida,composicao inseticida ou acaricida e processo inseticida ou acaricida
DE59108699D1 (de) * 1990-08-10 1997-06-12 Ciba Geigy Ag Naphthylalkylaminopyrimidin-Derivate, Verfahren zu ihrer Herstellung und diese enthaltende Schädlingsbekämpfungsmittel
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DE69130830D1 (de) * 1990-11-19 1999-03-11 Du Pont Insektizide, akarizide und fungizide aminopyrimidine
US5227387A (en) * 1991-09-03 1993-07-13 Dowelanco Quinoline nematicidal method
DE4131924A1 (de) * 1991-09-25 1993-07-08 Hoechst Ag Substituierte 4-alkoxypyrimidine, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
US5214144A (en) * 1991-10-07 1993-05-25 Dowelanco Process for the preparation of 4-haloquinazolines
EP0555183A1 (de) * 1992-02-07 1993-08-11 Ciba-Geigy Ag Schädlingsbekämpfungsmittel
EG20596A (en) * 1992-05-28 1999-09-30 Dow Elanco L L S Aqueaus flowable phenazaquin composition
AU4790893A (en) * 1992-08-19 1994-03-15 Dowelanco Pyridylethoxy-, pyridylethylamino-, and pyridylpropyl-derivatives of quinoline and quinazoline as insecticides and fungicides
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TW349094B (en) * 1995-09-05 1999-01-01 Basf Ag Compositions and methods for controlling harmful fungi
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CA2252684A1 (en) * 1996-04-26 1997-11-06 Basf Aktiengesellschaft Fungicide mixtures
WO1997042192A1 (de) * 1996-05-07 1997-11-13 Basf Aktiengesellschaft Imidazo-chinazoline, sie enthaltende mittel und deren verwendung zur bekämpfung von schadpilzen und tierischen schädlingen
DE19647317A1 (de) * 1996-11-15 1998-05-20 Hoechst Schering Agrevo Gmbh Substituierte Stickstoff-Heterocyclen, Verfahren zu ihrer Herstellung und ihre Verwendung als Schädlingsbekämpfungsmittel
AU2001293817A1 (en) * 2000-09-20 2002-04-02 Merck Patent Gmbh 4-amino-quinazolines
DE10055941A1 (de) * 2000-11-10 2002-05-23 Bayer Ag Wirkstoffkombinationen mit insektiziden und akariziden Eigenschaften
KR100415622B1 (ko) * 2002-02-21 2004-01-24 이회선 살비성 화합물 및 해충 표시자
JP4804706B2 (ja) * 2003-05-20 2011-11-02 クミアイ化学工業株式会社 農園芸用殺菌剤組成物
DE10353281A1 (de) 2003-11-14 2005-06-16 Bayer Cropscience Ag Wirkstoffkombination mit insektiziden und akariziden Eigenschaften
JP4630623B2 (ja) * 2004-10-04 2011-02-09 クミアイ化学工業株式会社 農園芸用殺菌剤組成物
EP1844023A1 (en) * 2004-12-31 2007-10-17 Sk Chemicals Co., Ltd. Quinazoline derivatives for the treatment and prevention of diabetes and obesity
WO2007065913A1 (en) * 2005-12-07 2007-06-14 Neurosearch A/S Novel quinazoline-2,4-diamine derivatives and their use as modulators of small-conductance calcium-activated potassium channels
PT2166855T (pt) * 2007-06-07 2018-06-12 Bayer Animal Health Gmbh Controlo de ectoparasitas
EP2008517A1 (de) 2007-06-29 2008-12-31 Bayer CropScience AG Akarizide Wirkstoffkombinationen
DE102007045922A1 (de) 2007-09-26 2009-04-02 Bayer Cropscience Ag Wirkstoffkombinationen mit insektiziden und akariziden Eigenschaften
EP2127522A1 (de) 2008-05-29 2009-12-02 Bayer CropScience AG Wirkstoffkombinationen mit insektiziden und akariziden Eigenschaften
PH12012500097A1 (en) * 2009-07-21 2011-01-27 Shanghai Inst Organic Chem Potent small molecule inhibitors of autophagy, and methods of use thereof
EP2525658B1 (de) 2010-01-22 2017-03-01 Bayer Intellectual Property GmbH Akarizide und/oder insektizide wirkstoffkombinationen
EP2382865A1 (de) 2010-04-28 2011-11-02 Bayer CropScience AG Synergistische Wirkstoffkombinationen
JPWO2012096137A1 (ja) * 2011-01-14 2014-06-09 株式会社エス・ディー・エス バイオテック 農園芸用の有害生物防除剤としてのキナゾリン誘導体
WO2012096115A1 (ja) * 2011-01-14 2012-07-19 株式会社エス・ディー・エス バイオテック 農園芸用の有害生物防除剤としての含フッ素キナゾリン誘導体
CN102210307A (zh) * 2011-05-04 2011-10-12 陕西韦尔奇作物保护有限公司 一种含有喹螨醚的农药组合物
TWI566700B (zh) 2011-07-21 2017-01-21 住友化學股份有限公司 防制病蟲害之組成物
CN102321075B (zh) * 2011-10-11 2013-06-05 华中师范大学 2-（1h-咪唑-1-基）喹唑啉衍生物的制备与杀菌活性
EP2825533B1 (en) 2012-03-13 2016-10-19 Basf Se Fungicidal pyrimidine compounds
CN105722833A (zh) 2013-09-16 2016-06-29 巴斯夫欧洲公司 杀真菌的嘧啶化合物
WO2015036059A1 (en) 2013-09-16 2015-03-19 Basf Se Fungicidal pyrimidine compounds
BR112018006873A2 (pt) 2015-10-05 2018-11-06 The Trustees Of Columbia University In The City Of New York ativadores do fluxo autofágico e fosfolipase d e depuração de agregados de proteína incluindo tau e tratamento de proteinopatias
CN106632282B (zh) * 2016-12-22 2019-09-20 重庆智合生物医药有限公司 1,3-二甲基-7-取代喹唑啉-2,4-二酮含氟酰胺类化合物及其合成方法和应用
US20220235013A1 (en) 2017-03-21 2022-07-28 Bayer Pharma Aktiengesellschaft 2-methyl-quinazolines
CA3097231A1 (en) 2018-04-18 2019-10-24 Bayer Pharma Aktiengesellschaft 2-methyl-aza-quinazolines
US20220071999A1 (en) * 2018-12-21 2022-03-10 University Of Notre Dame Du Lac Design and discovery of bd oxidase inhibitors for the treatment of mycobacterial diseases
CN110194761B (zh) * 2019-07-05 2021-08-20 华东理工大学 喹唑啉基羧酸酯类衍生物及其抗菌用途
WO2022058344A1 (en) 2020-09-18 2022-03-24 Bayer Aktiengesellschaft Pyrido[2,3-d]pyrimidin-4-amines as sos1 inhibitors
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IL89029A (en) * 1988-01-29 1993-01-31 Lilly Co Eli Fungicidal quinoline and cinnoline derivatives, compositions containing them, and fungicidal methods of using them
IL89028A0 (en) * 1988-01-29 1989-08-15 Lilly Co Eli Quinoline,quinazoline and cinnoline derivatives

Also Published As

Publication number Publication date
BR8900365A (pt) 1989-09-19
CN1052379C (zh) 2000-05-17
DE68928841D1 (de) 1998-12-03
EP0326329B1 (en) 1998-10-28
EP0326329A3 (en) 1990-09-12
KR0129754B1 (ko) 1998-04-09
IL89027A0 (en) 1989-08-15
AU632994B2 (en) 1993-01-21
IL89027A (en) 1993-01-31
FI890421A0 (fi) 1989-01-27
AU2874789A (en) 1989-08-03
JP2776864B2 (ja) 1998-07-16
PT89506B (pt) 1994-04-29
AR246516A1 (es) 1994-08-31
DE68928841T2 (de) 1999-08-12
DK37089A (da) 1989-07-30
HUT49791A (en) 1989-11-28
EG19187A (en) 1994-10-30
HU207643B (en) 1993-05-28
EP0326329A2 (en) 1989-08-02
DK37089D0 (da) 1989-01-27
MX14663A (es) 1994-01-31
ZA89623B (en) 1989-12-27
JPH01226877A (ja) 1989-09-11
ES2121737T3 (es) 1998-12-16
MY103804A (en) 1993-09-30
PT89506A (pt) 1989-10-04
FI890421A (fi) 1989-07-30
TR27343A (tr) 1995-01-13
KR890011862A (ko) 1989-08-23
ATE172725T1 (de) 1998-11-15
NZ227733A (en) 1990-08-28
CN1035825A (zh) 1989-09-27

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B1 Patent granted (law 1993)
PUP Patent expired