DK170202B1 - 1,5-diaryl-3-substituerede pyrazolforbindelser, fremgangsmåde til fremstilling deraf og farmaceutiske præparater indeholdende forbindelserne - Google Patents

1,5-diaryl-3-substituerede pyrazolforbindelser, fremgangsmåde til fremstilling deraf og farmaceutiske præparater indeholdende forbindelserne Download PDF

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Publication number
DK170202B1
DK170202B1 DK273587A DK273587A DK170202B1 DK 170202 B1 DK170202 B1 DK 170202B1 DK 273587 A DK273587 A DK 273587A DK 273587 A DK273587 A DK 273587A DK 170202 B1 DK170202 B1 DK 170202B1
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DK
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Prior art keywords
methoxyphenyl
chlorophenyl
pyrazolyl
pyrazole
ome
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DK273587A
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Danish (da)
English (en)
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DK273587A (da
DK273587D0 (da
Inventor
Michael Paul Wachter
Michael Paul Ferro
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Ortho Pharma Corp
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Application filed by Ortho Pharma Corp filed Critical Ortho Pharma Corp
Publication of DK273587D0 publication Critical patent/DK273587D0/da
Publication of DK273587A publication Critical patent/DK273587A/da
Application granted granted Critical
Publication of DK170202B1 publication Critical patent/DK170202B1/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/14—Antitussive agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40—Unsaturated compounds
    • C07C59/76—Unsaturated compounds containing keto groups
    • C07C59/84—Unsaturated compounds containing keto groups containing six membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40—Unsaturated compounds
    • C07C59/76—Unsaturated compounds containing keto groups
    • C07C59/88—Unsaturated compounds containing keto groups containing halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK273587A 1986-05-29 1987-05-27 1,5-diaryl-3-substituerede pyrazolforbindelser, fremgangsmåde til fremstilling deraf og farmaceutiske præparater indeholdende forbindelserne DK170202B1 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US86799686A 1986-05-29 1986-05-29
US86799686 1986-05-29
US07/042,661 US4826868A (en) 1986-05-29 1987-04-29 1,5-Diaryl-3-substituted pyrazoles pharmaceutical compositions and use
US4266187 1987-04-29

Publications (3)

Publication Number Publication Date
DK273587D0 DK273587D0 (da) 1987-05-27
DK273587A DK273587A (da) 1987-11-30
DK170202B1 true DK170202B1 (da) 1995-06-12

Family

ID=26719497

Family Applications (1)

Application Number Title Priority Date Filing Date
DK273587A DK170202B1 (da) 1986-05-29 1987-05-27 1,5-diaryl-3-substituerede pyrazolforbindelser, fremgangsmåde til fremstilling deraf og farmaceutiske præparater indeholdende forbindelserne

Country Status (21)

Country Link
US (1) US4826868A (de)
EP (1) EP0248594B1 (de)
JP (1) JP2512751B2 (de)
KR (1) KR960007163B1 (de)
CN (1) CN1028227C (de)
AU (1) AU596844B2 (de)
CA (1) CA1337122C (de)
DE (2) DE3788244T2 (de)
DK (1) DK170202B1 (de)
ES (1) ES2059377T3 (de)
FI (1) FI94340C (de)
HK (1) HK14094A (de)
HU (1) HU221300B1 (de)
IE (1) IE63856B1 (de)
IL (1) IL82671A0 (de)
LU (1) LU90829I2 (de)
NL (1) NL300057I2 (de)
NO (2) NO172236C (de)
NZ (1) NZ220353A (de)
PH (1) PH25126A (de)
PT (1) PT84964B (de)

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US4956379A (en) * 1990-02-13 1990-09-11 Bristol-Myers Squibb Company Pyrazole carboxylic acids and esters and inhibition of blood platelet aggregation therewith
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Also Published As

Publication number Publication date
NL300057I1 (nl) 2001-12-01
NO172236B (no) 1993-03-15
HU221300B1 (en) 2002-09-28
PT84964A (en) 1987-06-01
EP0248594A2 (de) 1987-12-09
DE3788244D1 (de) 1994-01-05
FI872379A (fi) 1987-11-30
DK273587A (da) 1987-11-30
CN1028227C (zh) 1995-04-19
NZ220353A (en) 1989-05-29
FI94340C (fi) 1995-08-25
IE63856B1 (en) 1995-06-14
EP0248594B1 (de) 1993-11-24
HUT68247A (en) 1995-06-28
JPS6322080A (ja) 1988-01-29
NO2001016I1 (no) 2001-10-01
DE10199049I1 (de) 2002-01-10
ES2059377T3 (es) 1994-11-16
IE871403L (en) 1987-11-29
HK14094A (en) 1994-03-04
PH25126A (en) 1991-02-19
FI94340B (fi) 1995-05-15
DE3788244T2 (de) 1994-04-14
NO872228L (no) 1987-11-30
AU7360887A (en) 1987-12-10
IL82671A0 (en) 1987-11-30
PT84964B (pt) 1990-02-08
US4826868A (en) 1989-05-02
CN87103953A (zh) 1987-12-09
DK273587D0 (da) 1987-05-27
DE10199049I2 (de) 2003-01-09
NL300057I2 (nl) 2002-01-02
NO172236C (no) 1993-06-23
JP2512751B2 (ja) 1996-07-03
LU90829I2 (fr) 2001-11-12
KR960007163B1 (ko) 1996-05-29
FI872379A0 (fi) 1987-05-28
NO872228D0 (no) 1987-05-27
KR870011100A (ko) 1987-12-21
EP0248594A3 (en) 1988-11-17
AU596844B2 (en) 1990-05-17
CA1337122C (en) 1995-09-26

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