DK169409B1 - Vanduopløselige, farmaceutisk acceptable salte af substituerede derivater af rapamycin og farmaceutisk præparat indeholdende et sådant salt - Google Patents

Vanduopløselige, farmaceutisk acceptable salte af substituerede derivater af rapamycin og farmaceutisk præparat indeholdende et sådant salt Download PDF

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Publication number
DK169409B1
DK169409B1 DK584886A DK584886A DK169409B1 DK 169409 B1 DK169409 B1 DK 169409B1 DK 584886 A DK584886 A DK 584886A DK 584886 A DK584886 A DK 584886A DK 169409 B1 DK169409 B1 DK 169409B1
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Denmark
Prior art keywords
water
sub
rapamycin
pharmaceutically acceptable
soluble
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DK584886A
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Danish (da)
English (en)
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DK584886D0 (da
DK584886A (da
Inventor
Valentino John Stella
Paul Edwin Kennedy
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Univ Kansas
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Publication of DK584886D0 publication Critical patent/DK584886D0/da
Publication of DK584886A publication Critical patent/DK584886A/da
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Publication of DK169409B1 publication Critical patent/DK169409B1/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
DK584886A 1985-12-06 1986-12-05 Vanduopløselige, farmaceutisk acceptable salte af substituerede derivater af rapamycin og farmaceutisk præparat indeholdende et sådant salt DK169409B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/806,152 US4650803A (en) 1985-12-06 1985-12-06 Prodrugs of rapamycin
US80615285 1985-12-06

Publications (3)

Publication Number Publication Date
DK584886D0 DK584886D0 (da) 1986-12-05
DK584886A DK584886A (da) 1987-06-07
DK169409B1 true DK169409B1 (da) 1994-10-24

Family

ID=25193443

Family Applications (2)

Application Number Title Priority Date Filing Date
DK584886A DK169409B1 (da) 1985-12-06 1986-12-05 Vanduopløselige, farmaceutisk acceptable salte af substituerede derivater af rapamycin og farmaceutisk præparat indeholdende et sådant salt
DK034793A DK170750B1 (da) 1985-12-06 1993-03-25 Vandopløselige, farmaceutisk acceptable salte af i 43-stillingen monosubstitueret rapamycin, fremgangsmåde til fremstilling heraf og injicerbare, farmaceutiske præparater indeholdende et sådant salt.

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK034793A DK170750B1 (da) 1985-12-06 1993-03-25 Vandopløselige, farmaceutisk acceptable salte af i 43-stillingen monosubstitueret rapamycin, fremgangsmåde til fremstilling heraf og injicerbare, farmaceutiske præparater indeholdende et sådant salt.

Country Status (16)

Country Link
US (1) US4650803A (cs)
EP (1) EP0227355B1 (cs)
JP (2) JPH0670066B2 (cs)
KR (2) KR940004072B1 (cs)
AT (1) ATE74134T1 (cs)
AU (1) AU583439B2 (cs)
CA (2) CA1273920A (cs)
DE (1) DE3684574D1 (cs)
DK (2) DK169409B1 (cs)
ES (1) ES2032750T3 (cs)
GB (1) GB2183647A (cs)
GR (1) GR3004530T3 (cs)
HU (1) HU198054B (cs)
IE (1) IE64506B1 (cs)
PT (1) PT83843B (cs)
ZA (1) ZA869181B (cs)

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