DK160560C - Analogifremgangsmaade til fremstilling af acetyleniske derivater af androstenforbindelser samt mellemprodukt til brug derved - Google Patents

Analogifremgangsmaade til fremstilling af acetyleniske derivater af androstenforbindelser samt mellemprodukt til brug derved

Info

Publication number
DK160560C
DK160560C DK292679A DK292679A DK160560C DK 160560 C DK160560 C DK 160560C DK 292679 A DK292679 A DK 292679A DK 292679 A DK292679 A DK 292679A DK 160560 C DK160560 C DK 160560C
Authority
DK
Denmark
Prior art keywords
androsten
analogue
compounds
preparation
intermediate use
Prior art date
Application number
DK292679A
Other languages
Danish (da)
English (en)
Other versions
DK292679A (da
DK160560B (da
Inventor
Jean Georges Teutsch
Roger Deraedt
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of DK292679A publication Critical patent/DK292679A/da
Publication of DK160560B publication Critical patent/DK160560B/da
Application granted granted Critical
Publication of DK160560C publication Critical patent/DK160560C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003—Androstane derivatives
    • C07J1/0033—Androstane derivatives substituted in position 17 alfa and 17 beta
    • C07J1/004—Androstane derivatives substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0048—Alkynyl derivatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003—Androstane derivatives
    • C07J1/0011—Androstane derivatives substituted in position 17 by a keto group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003—Androstane derivatives
    • C07J1/0033—Androstane derivatives substituted in position 17 alfa and 17 beta

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK292679A 1978-07-13 1979-07-12 Analogifremgangsmaade til fremstilling af acetyleniske derivater af androstenforbindelser samt mellemprodukt til brug derved DK160560C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR7820971A FR2430952A1 (fr) 1978-07-13 1978-07-13 Nouveaux derives acetyleniques de l'androst 4-ene, leur procede de preparation et leur application comme medicament
FR7820971 1978-07-13

Publications (3)

Publication Number Publication Date
DK292679A DK292679A (da) 1980-01-14
DK160560B DK160560B (da) 1991-03-25
DK160560C true DK160560C (da) 1991-09-09

Family

ID=9210731

Family Applications (1)

Application Number Title Priority Date Filing Date
DK292679A DK160560C (da) 1978-07-13 1979-07-12 Analogifremgangsmaade til fremstilling af acetyleniske derivater af androstenforbindelser samt mellemprodukt til brug derved

Country Status (24)

Country Link
US (1) US4233297A (ja)
JP (2) JPS5515474A (ja)
AT (1) AT370109B (ja)
AU (1) AU534841B2 (ja)
BE (1) BE877658A (ja)
CA (1) CA1140110A (ja)
CH (2) CH641475A5 (ja)
DE (2) DE2954699C2 (ja)
DK (1) DK160560C (ja)
ES (1) ES8101081A1 (ja)
FR (1) FR2430952A1 (ja)
GB (2) GB2025422B (ja)
GR (1) GR81403B (ja)
HU (1) HU180519B (ja)
IL (1) IL57533A (ja)
IT (1) IT1164697B (ja)
LU (1) LU81497A1 (ja)
MA (1) MA18516A1 (ja)
NL (1) NL7905481A (ja)
OA (1) OA06258A (ja)
PH (1) PH17055A (ja)
PT (1) PT69906A (ja)
SE (1) SE440781B (ja)
ZA (1) ZA793100B (ja)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2547587B1 (fr) * 1983-06-14 1985-10-25 Roussel Uclaf Steroides radioactifs, leur procede de preparation, leur application a la mise en evidence des recepteurs de glucocorticoides et au dosage du nombre de sites de fixation
FR2644788B1 (fr) * 1989-03-22 1995-02-03 Roussel Uclaf Nouveaux steroides 3-ceto comportant une chaine en 17 amino-substituee, leur procede de preparation et les intermediaires de ce procede, leur application comme medicaments et les compositions pharmaceutiques les contenant
JPH02141007U (ja) * 1989-04-26 1990-11-27
KR0181264B1 (ko) * 1989-07-07 1999-03-20 라브리 페르낭 성스테로이드 활성 억제용 안드로겐 유도체
AU680818B2 (en) * 1992-05-21 1997-08-14 Endorecherche Inc. Improved antiandrogens
HUT69408A (en) * 1993-05-17 1995-09-28 Endorecherche Inc Androstane derivatives as antiandrogenes and pharmaceutical compositions containing them and intermediates
CN103145785B (zh) * 2013-03-19 2016-03-02 浙江仙居仙乐药业有限公司 一种醋酸环丙孕酮脱氢物的合成方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2740798A (en) * 1953-05-25 1956-04-03 Searle & Co 11 beta-hydroxy-17-ethynyl testosterone and esters thereof
US3010957A (en) * 1958-11-26 1961-11-28 Schering Corp Ethinyl androstadienes
FR1349113A (fr) * 1959-01-28 1964-01-17 Upjohn Co Procédé de fabrication de 6-fluoro-11 oxygéné-17-bêta-hydroxy-17 alpha-alkynyl inférieur-4-androstène-3-ones et leurs dérivés acylés
US3793308A (en) * 1972-11-08 1974-02-19 Upjohn Co 4-spiro(cyclopropyl)androstenes and process for their production
SE7801152L (sv) * 1977-02-22 1978-08-23 Roussel Uclaf Sett att framstella 17alfa-acetylen-derivat av androst-4-en

Also Published As

Publication number Publication date
NL7905481A (nl) 1980-01-15
ES482387A0 (es) 1980-12-01
ZA793100B (en) 1980-06-25
GR81403B (ja) 1984-12-11
JPS6362515B2 (ja) 1988-12-02
DE2928374C2 (ja) 1991-12-12
IL57533A0 (en) 1979-10-31
IT7949743A0 (it) 1979-07-12
CH642977A5 (fr) 1984-05-15
HU180519B (en) 1983-03-28
JPS5515474A (en) 1980-02-02
JPS6252758B2 (ja) 1987-11-06
LU81497A1 (fr) 1980-02-14
CA1140110A (fr) 1983-01-25
PT69906A (fr) 1979-08-01
ES8101081A1 (es) 1980-12-01
GB2108503A (en) 1983-05-18
OA06258A (fr) 1981-06-30
US4233297A (en) 1980-11-11
BE877658A (fr) 1980-01-14
PH17055A (en) 1984-05-17
CH641475A5 (fr) 1984-02-29
DE2928374A1 (de) 1980-01-31
ATA488979A (de) 1982-07-15
DK292679A (da) 1980-01-14
JPS6345295A (ja) 1988-02-26
GB2108503B (en) 1983-09-14
DE2954699C2 (ja) 1992-04-16
DK160560B (da) 1991-03-25
FR2430952A1 (fr) 1980-02-08
FR2430952B1 (ja) 1980-12-05
IL57533A (en) 1984-01-31
AT370109B (de) 1983-03-10
SE7904431L (sv) 1980-01-14
GB2025422B (en) 1983-05-05
GB2025422A (en) 1980-01-23
SE440781B (sv) 1985-08-19
AU4889479A (en) 1980-01-17
MA18516A1 (fr) 1980-04-01
IT1164697B (it) 1987-04-15
AU534841B2 (en) 1984-02-16

Similar Documents

Publication Publication Date Title
DK150068C (da) Analogifremgangsmaade til fremstilling af aminothiazoler
DK154553C (da) Analogifremgangsmaade til fremstilling af ether- eller thioethermercaptoacylproliner
DK155665C (da) Analogifremgangsmaade til fremstilling af carbostyrilforbindelser
DK46079A (da) Fremgangsmaade til fremstilling af alkylendiaminderivater
DK295979A (da) Acylphosphinoforbindelser fremgangsmaade til fremstilling af disse samt deres anvendelse
DK174278A (da) Fremgangsmaade til fremstilling af somatostatinanaloge samt mellemprodukt til brug ved fremgangsmaaden
DK156001C (da) Analogifremgangsmaade til fremstilling af mercaptosubstituerede 2,3,4,5-tetrahydro-1h-3-benzazepiner
DK154940C (da) Analogifremgangsmaade til fremstilling af tetra- eller pentapeptider
DK157860C (da) Analogifremgangsmaade til fremstilling af benzylimidazolderivater samt farmaceutisk acceptable syreadditionssalte deraf
DK266479A (da) Fremgangsmaade til fremstilling af 3-aminopropoxyarylderivater
DK301477A (da) Fremgangsmaade til stereoselektiv fremstilling af hexahydrodibenzopyranoner samt mellemprodukt til brug ved fremgangsmaaden
DK148477C (da) Analogifremgangsmaade til fremstilling af tetrahydropyridinylindolderivater eller additionssalte deraf
DK157193C (da) Analogifremgangsmaade til fremstilling af carbostyrilforbindelser
DK310779A (da) Fremgangsmaade til fremstilling af pyrimidinonderivater
DK533979A (da) Fremgangsmaade til fremstilling af thiazolylderivater
DK186179A (da) Fremgangsmaade til fremstilling af carbapenemderivater
DK150141C (da) Analogifremgangsmaade til fremstilling af n-(2-thiazolyl)-amider
DK158460C (da) Analogifremgangsmaade til fremstilling af substituerede oxocarboxylsyrer
NO149958C (no) Analogifremgangsmaate til fremstilling av cykloheksenderivater
DK415379A (da) Fremgangsmaade til fremstilling af chromanolderivater
DK160560C (da) Analogifremgangsmaade til fremstilling af acetyleniske derivater af androstenforbindelser samt mellemprodukt til brug derved
DK184579A (da) Estere af substituerede 8-hydroxy-1-phenyl-2,3,4,5-tetrahydro-1h-3-benzazepiner,fremgangsmaade til deres fremstilling samt deres anvendelse
DK267779A (da) Fr&mgangsmaade til fremstilling af n-aralkylamino-propoxycyanopyridiner
DK16779A (da) Fremgangsmaade til fremstilling af betaendoprphinanaloge
DK160281C (da) Fremgangsmaade til fremstilling af steroid-s-thioesterderivater

Legal Events

Date Code Title Description
PUP Patent expired