DK16779A - Fremgangsmaade til fremstilling af betaendoprphinanaloge - Google Patents

Fremgangsmaade til fremstilling af betaendoprphinanaloge

Info

Publication number
DK16779A
DK16779A DK16779A DK16779A DK16779A DK 16779 A DK16779 A DK 16779A DK 16779 A DK16779 A DK 16779A DK 16779 A DK16779 A DK 16779A DK 16779 A DK16779 A DK 16779A
Authority
DK
Denmark
Prior art keywords
betaendoprphin
analog
procedure
preparation
betaendoprphin analog
Prior art date
Application number
DK16779A
Other languages
English (en)
Inventor
C H Li
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DK16779A publication Critical patent/DK16779A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/665Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • C07K14/675Beta-endorphins
    • C07K14/6755Beta-endorphins with at least 1 amino acid in D-form
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12Antidiarrhoeals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
DK16779A 1978-01-16 1979-01-15 Fremgangsmaade til fremstilling af betaendoprphinanaloge DK16779A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/869,555 US4116950A (en) 1978-01-16 1978-01-16 Analogs of human β-endorphin

Publications (1)

Publication Number Publication Date
DK16779A true DK16779A (da) 1979-07-17

Family

ID=25353784

Family Applications (1)

Application Number Title Priority Date Filing Date
DK16779A DK16779A (da) 1978-01-16 1979-01-15 Fremgangsmaade til fremstilling af betaendoprphinanaloge

Country Status (17)

Country Link
US (1) US4116950A (da)
EP (1) EP0003028B1 (da)
JP (1) JPS54100399A (da)
AT (1) ATA29679A (da)
AU (1) AU4324879A (da)
BE (1) BE873464A (da)
CA (1) CA1102312A (da)
DE (1) DE2901478A1 (da)
DK (1) DK16779A (da)
FR (1) FR2414497A1 (da)
GB (1) GB2012772B (da)
IL (1) IL56404A (da)
LU (1) LU80790A1 (da)
NL (1) NL7900093A (da)
PH (1) PH15501A (da)
SE (1) SE7900346L (da)
ZA (1) ZA7986B (da)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4396606A (en) * 1979-11-05 1983-08-02 Addiction Research Foundation Novel polypeptide analgesics
US4250087A (en) * 1979-12-10 1981-02-10 Hoffmann-La Roche Inc. Carboxyl terminus analogs of β-endorphin
US4316895A (en) * 1980-01-03 1982-02-23 Kimball Charles D Endorphins having placental or pancreatic origin
US4438104A (en) 1980-01-03 1984-03-20 Endorphin, Inc. Endorphins having placental or pancreatic origin
US4313937A (en) * 1980-08-12 1982-02-02 Tsutomu Oyama Method for producing long-lasting analgesic effects of β-endorphin
DE3152892T1 (de) * 1981-06-16 1983-09-08 John C. 98199 Seattle Wash. Houck Aus placenta oder pancreas gewonnene endorphine
US4422968A (en) * 1982-09-13 1983-12-27 The Regents Of The University Of California β-Endorphin analogs

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4038222A (en) * 1976-03-17 1977-07-26 Hoffman-La Roche Inc. Untriakontapeptide with opiate activity
US4081434A (en) * 1977-03-11 1978-03-28 Hoffmann-La Roche Inc. Novel analogs of β-endorphin

Also Published As

Publication number Publication date
IL56404A0 (en) 1979-03-12
BE873464A (fr) 1979-07-16
LU80790A1 (de) 1980-02-14
FR2414497A1 (fr) 1979-08-10
GB2012772A (en) 1979-08-01
JPS54100399A (en) 1979-08-08
ATA29679A (de) 1982-04-15
DE2901478A1 (de) 1979-07-19
AU4324879A (en) 1979-07-26
EP0003028A1 (de) 1979-07-25
US4116950A (en) 1978-09-26
EP0003028B1 (de) 1981-08-05
ZA7986B (en) 1980-03-26
PH15501A (en) 1983-02-03
GB2012772B (en) 1982-04-28
CA1102312A (en) 1981-06-02
IL56404A (en) 1981-11-30
NL7900093A (nl) 1979-07-18
SE7900346L (sv) 1979-07-17

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Legal Events

Date Code Title Description
AHS Application shelved for other reasons than non-payment