DK1392667T3 - Fremgangsmåde til fremstilling af biperiden - Google Patents

Fremgangsmåde til fremstilling af biperiden

Info

Publication number
DK1392667T3
DK1392667T3 DK02743054T DK02743054T DK1392667T3 DK 1392667 T3 DK1392667 T3 DK 1392667T3 DK 02743054 T DK02743054 T DK 02743054T DK 02743054 T DK02743054 T DK 02743054T DK 1392667 T3 DK1392667 T3 DK 1392667T3
Authority
DK
Denmark
Prior art keywords
biperiden
mixture
hept
piperidino
cyclo
Prior art date
Application number
DK02743054T
Other languages
Danish (da)
English (en)
Inventor
Peter Klein
Marco Thyes
Markus Grosse
Klaus Dieter Weber
Original Assignee
Farmaceutico S I T Specialita
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmaceutico S I T Specialita filed Critical Farmaceutico S I T Specialita
Application granted granted Critical
Publication of DK1392667T3 publication Critical patent/DK1392667T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/084Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/088Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/10Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms
    • C07D295/104Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms with the ring nitrogen atoms and the doubly bound oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/108Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms with the ring nitrogen atoms and the doubly bound oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Steroid Compounds (AREA)
  • Separation By Low-Temperature Treatments (AREA)
  • Crystals, And After-Treatments Of Crystals (AREA)
  • Superconductors And Manufacturing Methods Therefor (AREA)
DK02743054T 2001-05-18 2002-05-17 Fremgangsmåde til fremstilling af biperiden DK1392667T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10124451A DE10124451A1 (de) 2001-05-18 2001-05-18 Verfahren zur Herstellung von Biperiden
PCT/EP2002/005496 WO2002094800A1 (fr) 2001-05-18 2002-05-17 Procede de production de biperidene

Publications (1)

Publication Number Publication Date
DK1392667T3 true DK1392667T3 (da) 2007-10-22

Family

ID=7685403

Family Applications (1)

Application Number Title Priority Date Filing Date
DK02743054T DK1392667T3 (da) 2001-05-18 2002-05-17 Fremgangsmåde til fremstilling af biperiden

Country Status (14)

Country Link
US (1) US7030247B2 (fr)
EP (1) EP1392667B1 (fr)
JP (1) JP4338978B2 (fr)
KR (1) KR100849756B1 (fr)
CN (1) CN1240692C (fr)
AT (1) ATE365726T1 (fr)
BR (1) BRPI0209853C1 (fr)
CY (1) CY1106888T1 (fr)
DE (2) DE10124451A1 (fr)
DK (1) DK1392667T3 (fr)
ES (1) ES2290317T3 (fr)
IL (2) IL158926A0 (fr)
PT (1) PT1392667E (fr)
WO (1) WO2002094800A1 (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10124451A1 (de) 2001-05-18 2002-11-21 Abbott Gmbh & Co Kg Verfahren zur Herstellung von Biperiden
ES2250678T3 (es) 2001-05-18 2006-04-16 Laboratorio Farmaceutico S.I.T. Specialita' Igienico Terapeutiche S.R.L. Procedimiento para la preparacion de biperideno i.
KR100975396B1 (ko) * 2007-11-23 2010-08-11 윤중원 분수용 안전노즐
CN101508628B (zh) * 2009-03-30 2011-12-28 南昌航空大学 一种1-苯基-1-(二环[2.2.1]-5-庚烯-2)-乙醇的制备方法
CN106187948B (zh) * 2016-08-02 2019-02-22 安徽省逸欣铭医药科技有限公司 盐酸比哌立登制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2789110A (en) * 1953-03-14 1957-04-16 Knoll Ag Amino alcohols substituted by bicycloalkyl residues and a process of making same
DE1005067B (de) * 1953-03-14 1957-03-28 Knoll Ag Verfahren zur Herstellung von bicyclisch substituierten Aminopropanolen
JPH11189729A (ja) 1997-12-26 1999-07-13 Chemiprokasei Kaisha Ltd 色素兼紫外線安定剤およびそれを含む高分子組成物
DE10124451A1 (de) 2001-05-18 2002-11-21 Abbott Gmbh & Co Kg Verfahren zur Herstellung von Biperiden
DE10124449A1 (de) * 2001-05-18 2002-11-21 Abbott Gmbh & Co Kg Verfahren zur Herstellung von Biperiden

Also Published As

Publication number Publication date
BRPI0209853B8 (pt) 2018-12-18
US20040147753A1 (en) 2004-07-29
IL158926A0 (en) 2004-05-12
BR0209853A (pt) 2004-06-15
BRPI0209853B1 (pt) 2018-06-19
CN1525964A (zh) 2004-09-01
DE10124451A1 (de) 2002-11-21
BRPI0209853C1 (pt) 2021-05-25
CY1106888T1 (el) 2012-09-26
JP2004536067A (ja) 2004-12-02
EP1392667A1 (fr) 2004-03-03
KR100849756B1 (ko) 2008-07-31
KR20040007579A (ko) 2004-01-24
EP1392667B1 (fr) 2007-06-27
IL158926A (en) 2011-02-28
CN1240692C (zh) 2006-02-08
PT1392667E (pt) 2007-10-09
WO2002094800A1 (fr) 2002-11-28
ATE365726T1 (de) 2007-07-15
ES2290317T3 (es) 2008-02-16
JP4338978B2 (ja) 2009-10-07
US7030247B2 (en) 2006-04-18
DE50210384D1 (de) 2007-08-09

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