IT1317886B1 - Procedimento per la preparazione di 9,10-diidro-pirrolo (2,1-b)(1,3)benzotiazepine 9-ammino sostituite. - Google Patents
Procedimento per la preparazione di 9,10-diidro-pirrolo (2,1-b)(1,3)benzotiazepine 9-ammino sostituite.Info
- Publication number
- IT1317886B1 IT1317886B1 IT2000RM000434A ITRM20000434A IT1317886B1 IT 1317886 B1 IT1317886 B1 IT 1317886B1 IT 2000RM000434 A IT2000RM000434 A IT 2000RM000434A IT RM20000434 A ITRM20000434 A IT RM20000434A IT 1317886 B1 IT1317886 B1 IT 1317886B1
- Authority
- IT
- Italy
- Prior art keywords
- preparation
- benzotiazepine
- pyrol
- dihydro
- procedure
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Neurology (AREA)
- Public Health (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Priority Applications (25)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT2000RM000434A IT1317886B1 (it) | 2000-08-01 | 2000-08-01 | Procedimento per la preparazione di 9,10-diidro-pirrolo (2,1-b)(1,3)benzotiazepine 9-ammino sostituite. |
| DK01955529T DK1305318T3 (da) | 2000-08-01 | 2001-07-20 | Fremgangsmåde til fremstilling af 9-amino substitueret 9,10-dihydropyrrolo-[2,1-B][1,3]]benzothiazepiner |
| MXPA03000917A MXPA03000917A (es) | 2000-08-01 | 2001-07-20 | Procedimiento para la preparacion de 9,10-dihidropirrolo (2,1-b)(1,3)benzotiazepinas sustituidas con 9-amino. |
| PCT/IT2001/000391 WO2002010174A1 (en) | 2000-08-01 | 2001-07-20 | Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo [2,1-b][1,3]benzotiazepines |
| HU0301648A HUP0301648A3 (en) | 2000-08-01 | 2001-07-20 | Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo [2,1-b][1,3]benzotiazepines |
| AU7768701A AU7768701A (en) | 2000-08-01 | 2001-07-20 | Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo (2,1-B)(1,3)benzotiazepines |
| ES01955529T ES2215922T3 (es) | 2000-08-01 | 2001-07-20 | Procedimiento para la preparacion de 9,10 dihidropirrolo(2,1-b)(1,3)benzotiacepinas aminosustituidas en la posicion 9'. |
| PL365009A PL202400B1 (pl) | 2000-08-01 | 2001-07-20 | Sposób wytwarzania 9-aminopodstawionych 9,10-dihydropirolo-[2,1-b] [1,3] benzotiazepin |
| HU0301647A HUP0301647A3 (en) | 2000-08-01 | 2001-07-20 | Use fibrates for the preparation of a medicament useful in the treatment of congestive heart failure |
| KR1020037000134A KR100801269B1 (ko) | 2000-08-01 | 2001-07-20 | 9-아미노 치환된 9,10-디하이드로피롤로[2,1-b][1,3]벤조티아제핀의 제조 방법 |
| SI200130086T SI1305318T1 (en) | 2000-08-01 | 2001-07-20 | Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo (2,1-b) (1,3)benzothiazepines |
| CNB018131433A CN100354281C (zh) | 2000-08-01 | 2001-07-20 | 9－氨基取代的9,10－二氢吡咯并[2,1－b][1,3]苯并硫杂氮杂䓬的制备方法 |
| CZ200311A CZ294502B6 (cs) | 2000-08-01 | 2001-07-20 | Způsob přípravy 9-aminosubstituovaných 9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepinů |
| PT01955529T PT1305318E (pt) | 2000-08-01 | 2001-07-20 | Processo para a preparacao de 9, 10-di-hidropirrolo¬2,1-b|¬1,3)benzotiazepinas 9-amino substituidas |
| JP2002515903A JP2004505089A (ja) | 2000-08-01 | 2001-07-20 | ９−アミノ置換９，１０−ジヒドロピロロ［２，１−ｂ］［１，３］ベンゾチアゼピンの調製方法 |
| CA002415050A CA2415050C (en) | 2000-08-01 | 2001-07-20 | Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepines |
| EP01955529A EP1305318B1 (en) | 2000-08-01 | 2001-07-20 | Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo [2,1-b] [1,3]benzothiazepines |
| TR2004/00821T TR200400821T4 (tr) | 2000-08-01 | 2001-07-20 | 9-Amino-İkameli 9,10-Dihidropirolo [2,1] [1,3] benzotiyazepinlerin hazırlanması için yöntem |
| AU2001277687A AU2001277687B2 (en) | 2000-08-01 | 2001-07-20 | Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo [2,1-B][1,3]benzotiazepines |
| US10/343,629 US7078521B2 (en) | 2000-08-01 | 2001-07-20 | Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo[2,1-b][1,3]benzotiazepines |
| BR0112974-0A BR0112974A (pt) | 2000-08-01 | 2001-07-20 | Processo para a preparação de 9,10-diidropirrolo[2,1-b][1,3]benzotiazepinas 9-amino substituìdas |
| AT01955529T ATE261977T1 (de) | 2000-08-01 | 2001-07-20 | Verfahren zur herstellung von substituerten 9- amino-9,10-dihdropyrrolo(2,1-b)(1, 3)benzothiazepinen |
| DE60102385T DE60102385T2 (de) | 2000-08-01 | 2001-07-20 | Verfahren zur herstellung von substituerten 9-amino-9,10-dihdropyrrolo[2,1-b][1,3]benzothiazepinen |
| SK126-2003A SK287190B6 (sk) | 2000-08-01 | 2001-07-20 | Spôsob prípravy 9-aminosubstituovaných 9,10-dihydropyrol [2,1-B][1,3] benzodiazepínov |
| HK04100774A HK1059775A1 (en) | 2000-08-01 | 2004-02-06 | Process for the preparation of 9-amino substitued 9,10-dihydropyrrolo |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT2000RM000434A IT1317886B1 (it) | 2000-08-01 | 2000-08-01 | Procedimento per la preparazione di 9,10-diidro-pirrolo (2,1-b)(1,3)benzotiazepine 9-ammino sostituite. |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| ITRM20000434A0 ITRM20000434A0 (it) | 2000-08-01 |
| ITRM20000434A1 ITRM20000434A1 (it) | 2002-02-01 |
| IT1317886B1 true IT1317886B1 (it) | 2003-07-15 |
Family
ID=11454867
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IT2000RM000434A IT1317886B1 (it) | 2000-08-01 | 2000-08-01 | Procedimento per la preparazione di 9,10-diidro-pirrolo (2,1-b)(1,3)benzotiazepine 9-ammino sostituite. |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US7078521B2 (it) |
| EP (1) | EP1305318B1 (it) |
| JP (1) | JP2004505089A (it) |
| KR (1) | KR100801269B1 (it) |
| CN (1) | CN100354281C (it) |
| AT (1) | ATE261977T1 (it) |
| AU (2) | AU7768701A (it) |
| BR (1) | BR0112974A (it) |
| CA (1) | CA2415050C (it) |
| CZ (1) | CZ294502B6 (it) |
| DE (1) | DE60102385T2 (it) |
| DK (1) | DK1305318T3 (it) |
| ES (1) | ES2215922T3 (it) |
| HK (1) | HK1059775A1 (it) |
| HU (2) | HUP0301648A3 (it) |
| IT (1) | IT1317886B1 (it) |
| MX (1) | MXPA03000917A (it) |
| PL (1) | PL202400B1 (it) |
| PT (1) | PT1305318E (it) |
| SI (1) | SI1305318T1 (it) |
| SK (1) | SK287190B6 (it) |
| TR (1) | TR200400821T4 (it) |
| WO (1) | WO2002010174A1 (it) |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1301965B1 (it) * | 1998-07-28 | 2000-07-20 | Sigma Tau Ind Farmaceuti | Pirrolo (2,1-b)(1,3) benzotiazepine con attivita' antipsicoticaatipica. |
-
2000
- 2000-08-01 IT IT2000RM000434A patent/IT1317886B1/it active
-
2001
- 2001-07-20 EP EP01955529A patent/EP1305318B1/en not_active Expired - Lifetime
- 2001-07-20 PT PT01955529T patent/PT1305318E/pt unknown
- 2001-07-20 DK DK01955529T patent/DK1305318T3/da active
- 2001-07-20 JP JP2002515903A patent/JP2004505089A/ja not_active Withdrawn
- 2001-07-20 CA CA002415050A patent/CA2415050C/en not_active Expired - Fee Related
- 2001-07-20 AU AU7768701A patent/AU7768701A/xx active Pending
- 2001-07-20 KR KR1020037000134A patent/KR100801269B1/ko not_active IP Right Cessation
- 2001-07-20 HU HU0301648A patent/HUP0301648A3/hu unknown
- 2001-07-20 CZ CZ200311A patent/CZ294502B6/cs not_active IP Right Cessation
- 2001-07-20 AT AT01955529T patent/ATE261977T1/de not_active IP Right Cessation
- 2001-07-20 MX MXPA03000917A patent/MXPA03000917A/es active IP Right Grant
- 2001-07-20 BR BR0112974-0A patent/BR0112974A/pt not_active Application Discontinuation
- 2001-07-20 SK SK126-2003A patent/SK287190B6/sk not_active IP Right Cessation
- 2001-07-20 PL PL365009A patent/PL202400B1/pl not_active IP Right Cessation
- 2001-07-20 ES ES01955529T patent/ES2215922T3/es not_active Expired - Lifetime
- 2001-07-20 AU AU2001277687A patent/AU2001277687B2/en not_active Ceased
- 2001-07-20 US US10/343,629 patent/US7078521B2/en not_active Expired - Fee Related
- 2001-07-20 CN CNB018131433A patent/CN100354281C/zh not_active Expired - Fee Related
- 2001-07-20 SI SI200130086T patent/SI1305318T1/xx unknown
- 2001-07-20 DE DE60102385T patent/DE60102385T2/de not_active Expired - Lifetime
- 2001-07-20 TR TR2004/00821T patent/TR200400821T4/xx unknown
- 2001-07-20 HU HU0301647A patent/HUP0301647A3/hu unknown
- 2001-07-20 WO PCT/IT2001/000391 patent/WO2002010174A1/en active IP Right Grant
-
2004
- 2004-02-06 HK HK04100774A patent/HK1059775A1/xx not_active IP Right Cessation
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