DK1104765T4 - Fremgangsmåde til fremstilling af N,N,6-trimethyl-2-(4-methylphenyl)-imidazo-[1,2-a]-pyridin-3-acetamid og salte deraf - Google Patents

Fremgangsmåde til fremstilling af N,N,6-trimethyl-2-(4-methylphenyl)-imidazo-[1,2-a]-pyridin-3-acetamid og salte deraf

Info

Publication number
DK1104765T4
DK1104765T4 DK99938403T DK99938403T DK1104765T4 DK 1104765 T4 DK1104765 T4 DK 1104765T4 DK 99938403 T DK99938403 T DK 99938403T DK 99938403 T DK99938403 T DK 99938403T DK 1104765 T4 DK1104765 T4 DK 1104765T4
Authority
DK
Denmark
Prior art keywords
imidazo
acetamide
methylphenyl
trimethyl
pyridine
Prior art date
Application number
DK99938403T
Other languages
Danish (da)
English (en)
Other versions
DK1104765T3 (da
Inventor
Rafael Labriola
Original Assignee
Sint Quimica Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8304817&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK1104765(T4) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sint Quimica Sa filed Critical Sint Quimica Sa
Publication of DK1104765T3 publication Critical patent/DK1104765T3/da
Application granted granted Critical
Publication of DK1104765T4 publication Critical patent/DK1104765T4/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK99938403T 1998-08-06 1999-08-04 Fremgangsmåde til fremstilling af N,N,6-trimethyl-2-(4-methylphenyl)-imidazo-[1,2-a]-pyridin-3-acetamid og salte deraf DK1104765T4 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES009801694A ES2151834B1 (es) 1998-08-06 1998-08-06 Procedimiento para preparar n,n,6-trimetil-2-(4-metilfenil)-imidazo-(1,2-a)-piridina-3-acetamida y sus sales.
PCT/ES1999/000250 WO2000008021A2 (es) 1998-08-06 1999-08-04 Procedimiento para preparar n,n,6- trimetil-2- (4-metilfenil)- imidazo-[1,2-a] -piridina-3- acetamida y sus sales

Publications (2)

Publication Number Publication Date
DK1104765T3 DK1104765T3 (da) 2003-06-30
DK1104765T4 true DK1104765T4 (da) 2008-03-03

Family

ID=8304817

Family Applications (1)

Application Number Title Priority Date Filing Date
DK99938403T DK1104765T4 (da) 1998-08-06 1999-08-04 Fremgangsmåde til fremstilling af N,N,6-trimethyl-2-(4-methylphenyl)-imidazo-[1,2-a]-pyridin-3-acetamid og salte deraf

Country Status (26)

Country Link
US (1) US6407240B1 (hu)
EP (1) EP1104765B2 (hu)
JP (1) JP3544944B2 (hu)
KR (1) KR100492054B1 (hu)
AT (1) ATE234836T1 (hu)
AU (1) AU750302B2 (hu)
CA (1) CA2339594C (hu)
CZ (1) CZ292446B6 (hu)
DE (1) DE69906088T3 (hu)
DK (1) DK1104765T4 (hu)
ES (2) ES2151834B1 (hu)
HK (1) HK1037624A1 (hu)
HR (1) HRP20010158B1 (hu)
HU (1) HUP0102936A3 (hu)
IL (1) IL141133A (hu)
IS (1) IS5839A (hu)
NO (1) NO319780B1 (hu)
NZ (1) NZ510310A (hu)
PL (1) PL195888B1 (hu)
PT (1) PT1104765E (hu)
RS (1) RS50103B (hu)
RU (1) RU2221797C2 (hu)
SI (1) SI1104765T2 (hu)
SK (1) SK283652B6 (hu)
WO (1) WO2000008021A2 (hu)
ZA (1) ZA200101294B (hu)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2151834B1 (es) 1998-08-06 2001-08-16 Sint Quimica Sa Procedimiento para preparar n,n,6-trimetil-2-(4-metilfenil)-imidazo-(1,2-a)-piridina-3-acetamida y sus sales.
AU1873901A (en) * 1999-11-22 2001-06-04 Egis Gyogyszergyar Rt. Process for the preparation of 6-methyl-2-(4-methyl-phenyl)-imidazo(1,2-A)pyrimidine-3- (N,N-dimethyl-acetamide) and intermediates
IT1318624B1 (it) * 2000-07-14 2003-08-27 Dinamite Dipharma S P A In For Processo per la preparazione di 2-fenil-imidazo (1,2-a)piridin-3-acetammidi.
US6596731B2 (en) 2001-03-27 2003-07-22 Hoffmann-La Roche Inc. Substituted imidazo[1,2-A] pyridine derivatives
ATE394398T1 (de) * 2002-07-15 2008-05-15 Scinopharm Taiwan Ltd Verfahren zur herstellung von imidazo(1,2- a)pyridin-3-acetamiden
ES2320758T3 (es) 2002-12-18 2009-05-28 Mallinckrodt Inc. Sintesis de heteroaril acetamidas.
AU2005262622A1 (en) * 2004-06-22 2006-01-19 Mallinckrodt Inc. Synthesis of heteroaryl acetamides from reaction mixtures having reduced water content
EP1948655A1 (en) * 2005-10-03 2008-07-30 Mallinckrodt, Inc. Process for preparing zolpidem hemitartrate and tartrate polymorphs
EP1803722A1 (en) * 2006-01-03 2007-07-04 Ferrer Internacional, S.A. Imidazo[1,2-a]pyridin-3-yl-acetic acid hydrazides, processes for their preparation and pharmaceutical uses thereof
US20080145425A1 (en) * 2006-12-15 2008-06-19 Pliva Research & Development Limited Pharmaceutical composition of zolpidem
CN103360387B (zh) * 2012-03-28 2016-12-14 江苏豪森药业集团有限公司 一种制备化合物唑吡坦的方法
CN104610253B (zh) * 2015-01-26 2016-11-16 郑州大学 2‑三氟甲基‑2‑羟基‑2‑(2‑芳基吡啶并[1,2‑α]咪唑)乙酸酯类化合物
CN114105974A (zh) * 2020-08-27 2022-03-01 鲁南制药集团股份有限公司 一种唑吡坦的制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2600650B1 (fr) * 1986-06-27 1988-09-09 Synthelabo Procede de preparation d'imidazopyridines et composes intermediaires
ES2151834B1 (es) 1998-08-06 2001-08-16 Sint Quimica Sa Procedimiento para preparar n,n,6-trimetil-2-(4-metilfenil)-imidazo-(1,2-a)-piridina-3-acetamida y sus sales.

Also Published As

Publication number Publication date
CZ2001360A3 (cs) 2001-12-12
EP1104765A2 (en) 2001-06-06
IL141133A (en) 2005-11-20
RU2221797C2 (ru) 2004-01-20
CZ292446B6 (cs) 2003-09-17
US6407240B1 (en) 2002-06-18
ES2151834B1 (es) 2001-08-16
RS50103B (sr) 2009-01-22
AU750302B2 (en) 2002-07-18
DE69906088D1 (de) 2003-04-24
HUP0102936A2 (hu) 2002-01-28
HRP20010158A2 (en) 2002-02-28
ES2151834A1 (es) 2001-01-01
ATE234836T1 (de) 2003-04-15
SK1592001A3 (en) 2001-12-03
IS5839A (is) 2001-02-05
HUP0102936A3 (en) 2002-09-30
DE69906088T2 (de) 2003-12-24
WO2000008021A3 (es) 2000-07-06
NO20010613L (no) 2001-02-05
CA2339594C (en) 2005-05-03
SI1104765T1 (en) 2003-08-31
SK283652B6 (sk) 2003-11-04
EP1104765B2 (en) 2007-11-14
NO319780B1 (no) 2005-09-12
ES2195598T5 (es) 2008-05-01
PT1104765E (pt) 2003-08-29
DK1104765T3 (da) 2003-06-30
KR20010072173A (ko) 2001-07-31
ES2195598T3 (es) 2003-12-01
EP1104765B1 (en) 2003-03-19
DE69906088T3 (de) 2008-04-30
YU8301A (sh) 2003-10-31
JP3544944B2 (ja) 2004-07-21
NZ510310A (en) 2002-11-26
SI1104765T2 (sl) 2008-04-30
ZA200101294B (en) 2002-02-15
HRP20010158B1 (en) 2003-12-31
AU5291299A (en) 2000-02-28
HK1037624A1 (en) 2002-02-15
CA2339594A1 (en) 2000-02-17
PL346158A1 (en) 2002-01-28
NO20010613D0 (no) 2001-02-05
WO2000008021A2 (es) 2000-02-17
IL141133A0 (en) 2002-02-10
KR100492054B1 (ko) 2005-05-31
PL195888B1 (pl) 2007-11-30
JP2002522437A (ja) 2002-07-23

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