DK1042324T3 - Heterocykliske forbindelser til inhibering af mavesyresekretion, fremgangsmåder til deres fremstilling og farmaceutiske præparater deraf - Google Patents

Heterocykliske forbindelser til inhibering af mavesyresekretion, fremgangsmåder til deres fremstilling og farmaceutiske præparater deraf

Info

Publication number
DK1042324T3
DK1042324T3 DK98957270T DK98957270T DK1042324T3 DK 1042324 T3 DK1042324 T3 DK 1042324T3 DK 98957270 T DK98957270 T DK 98957270T DK 98957270 T DK98957270 T DK 98957270T DK 1042324 T3 DK1042324 T3 DK 1042324T3
Authority
DK
Denmark
Prior art keywords
inhibition
preparation
methods
pharmaceutical preparations
heterocyclic compounds
Prior art date
Application number
DK98957270T
Other languages
Danish (da)
English (en)
Inventor
Kosrat Amin
Mikael Dahlstroem
Peter Nordberg
Ingemar Starke
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Application granted granted Critical
Publication of DK1042324T3 publication Critical patent/DK1042324T3/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK98957270T 1997-11-28 1998-11-18 Heterocykliske forbindelser til inhibering af mavesyresekretion, fremgangsmåder til deres fremstilling og farmaceutiske præparater deraf DK1042324T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE9704404A SE9704404D0 (sv) 1997-11-28 1997-11-28 New compounds
PCT/SE1998/002091 WO1999028322A1 (en) 1997-11-28 1998-11-18 Heterocyclic compounds for inhibition of gastric acid secretion, processes for their preparation and pharmaceutical compositions thereof

Publications (1)

Publication Number Publication Date
DK1042324T3 true DK1042324T3 (da) 2003-05-05

Family

ID=20409181

Family Applications (1)

Application Number Title Priority Date Filing Date
DK98957270T DK1042324T3 (da) 1997-11-28 1998-11-18 Heterocykliske forbindelser til inhibering af mavesyresekretion, fremgangsmåder til deres fremstilling og farmaceutiske præparater deraf

Country Status (33)

Country Link
US (1) US6518270B1 (cs)
EP (1) EP1042324B1 (cs)
JP (1) JP2001525322A (cs)
KR (1) KR20010032559A (cs)
CN (1) CN1142933C (cs)
AR (1) AR016972A1 (cs)
AT (1) ATE233263T1 (cs)
AU (1) AU752187C (cs)
BR (1) BR9814755A (cs)
CA (1) CA2311798A1 (cs)
CZ (1) CZ292349B6 (cs)
DE (1) DE69811735T2 (cs)
DK (1) DK1042324T3 (cs)
EE (1) EE04060B1 (cs)
ES (1) ES2191356T3 (cs)
HK (1) HK1030216A1 (cs)
HU (1) HUP0100601A3 (cs)
ID (1) ID24730A (cs)
IL (1) IL136145A0 (cs)
IS (1) IS5486A (cs)
MY (1) MY121032A (cs)
NO (1) NO315704B1 (cs)
NZ (1) NZ504355A (cs)
PL (1) PL340920A1 (cs)
PT (1) PT1042324E (cs)
RU (1) RU2241000C2 (cs)
SE (1) SE9704404D0 (cs)
SK (1) SK283904B6 (cs)
TR (1) TR200001530T2 (cs)
TW (1) TW515798B (cs)
UA (1) UA70932C2 (cs)
WO (1) WO1999028322A1 (cs)
ZA (1) ZA9810468B (cs)

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US20070287726A1 (en) * 2004-08-02 2007-12-13 Altana Pharma Ag 5-Substituted 1H-Pyrrolo [3,2-B] Pyridines
CA2579083C (en) * 2004-09-03 2011-06-14 Yuhan Corporation Pyrrolo[3,2-c]pyridine derivatives and processes for the preparation thereof
ES2426920T3 (es) * 2004-09-03 2013-10-25 Yuhan Corporation Derivados de pirrolo[3,2-B]piridina y procesos para su preparación
AU2005280738B2 (en) 2004-09-03 2010-11-25 Yuhan Corporation Pyrrolo(3,2-c)pyridine derivatives and processes for the preparation thereof
KR100958829B1 (ko) 2004-09-03 2010-05-25 주식회사유한양행 피롤로[2,3-ｃ]피리딘 유도체 및 그의 제조방법
US7777040B2 (en) 2005-05-03 2010-08-17 Cgi Pharmaceuticals, Inc. Certain substituted ureas, as modulators of kinase activity
TW200800213A (en) 2005-09-02 2008-01-01 Abbott Lab Novel imidazo based heterocycles
WO2007067416A2 (en) * 2005-12-05 2007-06-14 Affinium Pharmaceuticals, Inc. Heterocyclylacrylamide compounds as fabi inhibitors and antibacterial agents
WO2007145921A1 (en) * 2006-06-06 2007-12-21 Schering Corporation Imidazopyrazines as protein kinase inhibitors
EP2054422B1 (en) 2006-07-20 2017-06-14 Debiopharm International SA Acrylamide derivatives as fab i inhibitors
EP3255045A1 (en) * 2007-02-16 2017-12-13 Debiopharm International SA Salts, prodrugs and polymorphs of fab i inhibitors
US20090221612A1 (en) 2008-02-13 2009-09-03 Mitchell Scott A Certain substituted amides, method of making, and method of use thereof
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ES2744541T3 (es) 2008-12-08 2020-02-25 Gilead Connecticut Inc Inhibidores de imidazopirazina Syk
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US9562056B2 (en) 2010-03-11 2017-02-07 Gilead Connecticut, Inc. Imidazopyridines Syk inhibitors
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MY176803A (en) 2013-07-30 2020-08-21 Gilead Connecticut Inc Polymorph of syk inhibitors
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Also Published As

Publication number Publication date
EP1042324A1 (en) 2000-10-11
CN1284078A (zh) 2001-02-14
WO1999028322A1 (en) 1999-06-10
BR9814755A (pt) 2000-10-03
AR016972A1 (es) 2001-08-01
CZ20001947A3 (cs) 2000-11-15
HUP0100601A2 (hu) 2001-09-28
RU2241000C2 (ru) 2004-11-27
CN1142933C (zh) 2004-03-24
AU752187C (en) 2003-09-18
CA2311798A1 (en) 1999-06-10
PL340920A1 (en) 2001-03-12
MY121032A (en) 2005-12-30
DE69811735D1 (de) 2003-04-03
EP1042324B1 (en) 2003-02-26
JP2001525322A (ja) 2001-12-11
SE9704404D0 (sv) 1997-11-28
AU1356599A (en) 1999-06-16
IL136145A0 (en) 2001-05-20
SK6742000A3 (en) 2001-03-12
AU752187B2 (en) 2002-09-12
NO20002721D0 (no) 2000-05-26
NZ504355A (en) 2001-12-21
ID24730A (id) 2000-08-03
CZ292349B6 (cs) 2003-09-17
ES2191356T3 (es) 2003-09-01
US6518270B1 (en) 2003-02-11
SK283904B6 (sk) 2004-04-06
EE04060B1 (et) 2003-06-16
DE69811735T2 (de) 2003-12-18
EE200000315A (et) 2001-10-15
ATE233263T1 (de) 2003-03-15
HUP0100601A3 (en) 2002-10-28
UA70932C2 (uk) 2004-11-15
NO315704B1 (no) 2003-10-13
KR20010032559A (ko) 2001-04-25
TW515798B (en) 2003-01-01
ZA9810468B (en) 1999-05-21
HK1030216A1 (en) 2001-04-27
PT1042324E (pt) 2003-06-30
IS5486A (is) 2000-05-10
TR200001530T2 (tr) 2000-11-21
NO20002721L (no) 2000-07-28

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