IS5486A - Heterósýklísk efnasambönd til að hindra magasýruflæði, aðferðir við framleiðslu þeirra og lyfjablöndur er innihalda þau - Google Patents

Heterósýklísk efnasambönd til að hindra magasýruflæði, aðferðir við framleiðslu þeirra og lyfjablöndur er innihalda þau

Info

Publication number
IS5486A
IS5486A IS5486A IS5486A IS5486A IS 5486 A IS5486 A IS 5486A IS 5486 A IS5486 A IS 5486A IS 5486 A IS5486 A IS 5486A IS 5486 A IS5486 A IS 5486A
Authority
IS
Iceland
Prior art keywords
pharmaceutical compositions
compositions containing
production methods
heterocyclic compounds
gastric acid
Prior art date
Application number
IS5486A
Other languages
English (en)
Inventor
Amin Kosrat
Dahlström Mikael
Nordberg Peter
Starke Ingemar
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of IS5486A publication Critical patent/IS5486A/is

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
IS5486A 1997-11-28 2000-05-10 Heterósýklísk efnasambönd til að hindra magasýruflæði, aðferðir við framleiðslu þeirra og lyfjablöndur er innihalda þau IS5486A (is)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE9704404A SE9704404D0 (sv) 1997-11-28 1997-11-28 New compounds
PCT/SE1998/002091 WO1999028322A1 (en) 1997-11-28 1998-11-18 Heterocyclic compounds for inhibition of gastric acid secretion, processes for their preparation and pharmaceutical compositions thereof

Publications (1)

Publication Number Publication Date
IS5486A true IS5486A (is) 2000-05-10

Family

ID=20409181

Family Applications (1)

Application Number Title Priority Date Filing Date
IS5486A IS5486A (is) 1997-11-28 2000-05-10 Heterósýklísk efnasambönd til að hindra magasýruflæði, aðferðir við framleiðslu þeirra og lyfjablöndur er innihalda þau

Country Status (32)

Country Link
US (1) US6518270B1 (is)
EP (1) EP1042324B1 (is)
JP (1) JP2001525322A (is)
KR (1) KR20010032559A (is)
CN (1) CN1142933C (is)
AR (1) AR016972A1 (is)
AT (1) ATE233263T1 (is)
AU (1) AU752187C (is)
BR (1) BR9814755A (is)
CA (1) CA2311798A1 (is)
CZ (1) CZ292349B6 (is)
DE (1) DE69811735T2 (is)
DK (1) DK1042324T3 (is)
EE (1) EE04060B1 (is)
ES (1) ES2191356T3 (is)
HU (1) HUP0100601A3 (is)
ID (1) ID24730A (is)
IL (1) IL136145A0 (is)
IS (1) IS5486A (is)
MY (1) MY121032A (is)
NO (1) NO315704B1 (is)
NZ (1) NZ504355A (is)
PL (1) PL340920A1 (is)
PT (1) PT1042324E (is)
RU (1) RU2241000C2 (is)
SE (1) SE9704404D0 (is)
SK (1) SK283904B6 (is)
TR (1) TR200001530T2 (is)
TW (1) TW515798B (is)
UA (1) UA70932C2 (is)
WO (1) WO1999028322A1 (is)
ZA (1) ZA9810468B (is)

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ES2320984T3 (es) * 2001-04-06 2009-06-01 Affinium Pharmaceuticals, Inc. Inhibidores de fab i.
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US7312341B2 (en) 2002-09-09 2007-12-25 Cgi Pharmaceuticals, Inc. 6-aryl-imidazo[1,2-a] pyrazin-8-ylamines, method of making, and method of use thereof
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AU2003266622A1 (en) * 2002-09-25 2004-04-19 Sankyo Company, Limited Medicinal composition for inhibiting increase in blood gastrin concentration
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WO2005005429A1 (en) 2003-06-30 2005-01-20 Cellular Genomics, Inc. Certain heterocyclic substituted imidazo[1,2-a]pyrazin-8-ylamines and methods of inhibition of bruton’s tyrosine kinase by such compounds
WO2005019220A2 (en) 2003-08-11 2005-03-03 Cellular Genomics Inc. Substituted imidazo[1,2-a]pyrazines as modulators of kinase activity
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ES2515101T3 (es) 2004-06-04 2014-10-29 Debiopharm International Sa Derivados de acrilamida como agentes antibióticos
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US7642269B2 (en) 2004-09-03 2010-01-05 Yuhan Corporation Pyrrolo[3,2-B]pyridine derivatives and processes for the preparation thereof
EP1784404B1 (en) 2004-09-03 2011-11-16 Yuhan Corporation Pyrrolo[2,3-c]pyridine derivatives and processes for the preparation thereof
RU2378275C2 (ru) 2004-09-03 2010-01-10 Юхан Корпорейшн ПРОИЗВОДНЫЕ ПИРРОЛО[3,2-c]ПИРИДИНА И СПОСОБ ИХ ПОЛУЧЕНИЯ
WO2007024294A2 (en) 2005-05-03 2007-03-01 Cgi Pharmaceuticals, Inc. Certain substituted ureas, as modulators of kinase activity
CA2620223A1 (en) 2005-09-02 2007-03-08 Abbott Laboratories Novel imidazo based heterocycles
JP2009518399A (ja) * 2005-12-05 2009-05-07 アフィニウム ファーマシューティカルズ， インク． Ｆａｂｉ阻害剤および抗菌剤としてのヘテロ環アクリルアミド化合物
JP2009539840A (ja) * 2006-06-06 2009-11-19 シェーリング コーポレイション プロテインキナーゼ阻害剤としてのイミダゾピラジン
CA2658506C (en) 2006-07-20 2016-01-26 Affinium Pharmaceuticals, Inc. Acrylamide derivatives as fab 1 inhibitors
WO2008098374A1 (en) 2007-02-16 2008-08-21 Affinium Pharmaceuticals, Inc. Salts, prodrugs and polymorphs of fab i inhibitors
AU2009215191A1 (en) 2008-02-13 2009-08-20 Gilead Connecticut, Inc. 6-aryl-imidaz0[l, 2-a] pyrazine derivatives, method of making, and method of use thereof
US8450321B2 (en) 2008-12-08 2013-05-28 Gilead Connecticut, Inc. 6-(1H-indazol-6-yl)-N-[4-(morpholin-4-yl)phenyl]imidazo-[1,2-A]pyrazin-8-amine, or a pharmaceutically acceptable salt thereof, as a SYK inhibitor
CA2746023C (en) 2008-12-08 2018-03-27 Gilead Connecticut, Inc. Imidazopyrazine syk inhibitors
JP5696052B2 (ja) 2008-12-08 2015-04-08 ギリアード コネチカット， インコーポレイテッド イミダゾピラジンｓｙｋ阻害剤
ES2530449T3 (es) 2010-03-11 2015-03-02 Gilead Connecticut Inc Inhibidores de Syk de imidazopiridinas
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HK1222329A1 (zh) 2013-07-30 2017-06-30 吉利德康涅狄格公司 Syk抑制劑的製劑
US9657023B2 (en) 2013-07-30 2017-05-23 Gilead Connecticut, Inc. Polymorph of Syk inhibitors
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US9290505B2 (en) 2013-12-23 2016-03-22 Gilead Sciences, Inc. Substituted imidazo[1,2-a]pyrazines as Syk inhibitors
KR20170029580A (ko) 2014-07-14 2017-03-15 길리애드 사이언시즈, 인코포레이티드 암을 치료하기 위한 조합물
PT3419628T (pt) 2016-02-26 2021-01-05 Debiopharm Int Sa Medicamento para o tratamento de infeções do pé diabético
US11384082B2 (en) 2017-08-25 2022-07-12 Kronos Bio, Inc. Hydrates of polymorphs of 6-(1H-indazol-6-YL)-N-(4-morpholinophenyl)-2,3-dihydroimidazo[1,2-A]pyrazin-8-amine bisemsylate as Syk inhibitors
ES2944535T3 (es) 2019-02-14 2023-06-22 Debiopharm Int Sa Formulación de afabicina, método para preparar la misma
KR20210131372A (ko) 2019-02-22 2021-11-02 크로노스 바이오, 인코포레이티드 Syk 억제제로서의 축합된 피라진의 고체 형태
KR20220020963A (ko) 2019-06-14 2022-02-21 데비오팜 인터네셔날 에스 에이 바이오필름 관련 박테리아 감염을 치료하기 위한 의약 및 이의 용도

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Also Published As

Publication number Publication date
CA2311798A1 (en) 1999-06-10
CN1284078A (zh) 2001-02-14
ID24730A (id) 2000-08-03
ES2191356T3 (es) 2003-09-01
NO20002721L (no) 2000-07-28
UA70932C2 (uk) 2004-11-15
TR200001530T2 (tr) 2000-11-21
SK6742000A3 (en) 2001-03-12
DE69811735D1 (de) 2003-04-03
TW515798B (en) 2003-01-01
HK1030216A1 (en) 2001-04-27
IL136145A0 (en) 2001-05-20
SE9704404D0 (sv) 1997-11-28
CN1142933C (zh) 2004-03-24
AU752187C (en) 2003-09-18
NO20002721D0 (no) 2000-05-26
BR9814755A (pt) 2000-10-03
SK283904B6 (sk) 2004-04-06
HUP0100601A3 (en) 2002-10-28
EP1042324A1 (en) 2000-10-11
ATE233263T1 (de) 2003-03-15
MY121032A (en) 2005-12-30
NO315704B1 (no) 2003-10-13
EP1042324B1 (en) 2003-02-26
RU2241000C2 (ru) 2004-11-27
NZ504355A (en) 2001-12-21
KR20010032559A (ko) 2001-04-25
HUP0100601A2 (hu) 2001-09-28
WO1999028322A1 (en) 1999-06-10
PT1042324E (pt) 2003-06-30
DE69811735T2 (de) 2003-12-18
CZ292349B6 (cs) 2003-09-17
CZ20001947A3 (cs) 2000-11-15
DK1042324T3 (da) 2003-05-05
JP2001525322A (ja) 2001-12-11
EE04060B1 (et) 2003-06-16
PL340920A1 (en) 2001-03-12
AU752187B2 (en) 2002-09-12
US6518270B1 (en) 2003-02-11
AR016972A1 (es) 2001-08-01
EE200000315A (et) 2001-10-15
ZA9810468B (en) 1999-05-21
AU1356599A (en) 1999-06-16

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