DK0705272T3 - Særlig fremgangsmåde til fremstilling af 17beta-substituerede 4-azaandrostanderivater - Google Patents

Særlig fremgangsmåde til fremstilling af 17beta-substituerede 4-azaandrostanderivater

Info

Publication number
DK0705272T3
DK0705272T3 DK93913459T DK93913459T DK0705272T3 DK 0705272 T3 DK0705272 T3 DK 0705272T3 DK 93913459 T DK93913459 T DK 93913459T DK 93913459 T DK93913459 T DK 93913459T DK 0705272 T3 DK0705272 T3 DK 0705272T3
Authority
DK
Denmark
Prior art keywords
cir
general formula
group
substituted
preparing
Prior art date
Application number
DK93913459T
Other languages
Danish (da)
English (en)
Inventor
Judit Horvath
Janos Szeles
Laszlo Kollar
Zoltan Tuba
Gabor Balogh
Original Assignee
Richter Gedeon Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszet filed Critical Richter Gedeon Vegyeszet
Application granted granted Critical
Publication of DK0705272T3 publication Critical patent/DK0705272T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK93913459T 1993-06-24 1993-06-24 Særlig fremgangsmåde til fremstilling af 17beta-substituerede 4-azaandrostanderivater DK0705272T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/HU1993/000039 WO1995000531A1 (en) 1993-06-24 1993-06-24 NOVEL PROCESS FOR PREPARING 17β-SUBSTITUTED 4-AZAANDROSTANE DERIVATIVES

Publications (1)

Publication Number Publication Date
DK0705272T3 true DK0705272T3 (da) 2002-05-27

Family

ID=10982846

Family Applications (1)

Application Number Title Priority Date Filing Date
DK93913459T DK0705272T3 (da) 1993-06-24 1993-06-24 Særlig fremgangsmåde til fremstilling af 17beta-substituerede 4-azaandrostanderivater

Country Status (14)

Country Link
EP (1) EP0705272B1 (enExample)
JP (1) JP3253088B2 (enExample)
KR (1) KR100279567B1 (enExample)
AT (1) ATE215092T1 (enExample)
AU (1) AU681585B2 (enExample)
CA (1) CA2166090C (enExample)
DE (1) DE69331763T2 (enExample)
DK (1) DK0705272T3 (enExample)
ES (1) ES2173889T3 (enExample)
FI (1) FI956236A0 (enExample)
PT (1) PT705272E (enExample)
RU (1) RU2109746C1 (enExample)
UA (1) UA41933C2 (enExample)
WO (1) WO1995000531A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU212459B (en) * 1992-10-02 1996-06-28 Richter Gedeon Vegyeszet Process for producing new 17-beta-substituted 4-aza-androstane-derivatives and pharmaceutical compositions containing them
ES2153789B1 (es) 1999-07-05 2001-10-16 Raga Consultores S L Procedimiento para la obtencion de 178-(n-terc-butlcarbamoil)-3-ona-4-aza-esteroides
CN1784236A (zh) 2003-05-07 2006-06-07 麦克公司 雄激素受体调节剂及其使用方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU527030B2 (en) * 1978-04-13 1983-02-10 Merck & Co., Inc. 4-aza-17-substituted-5a-androstan-3-ones
SU930914A1 (ru) * 1980-03-07 1985-05-30 Институт биоорганической химии АН БССР Способ получени спин-меченых производных 8-аза-16-оксастероидов
IL74365A (en) * 1984-02-27 1990-07-26 Merck & Co Inc 17beta-(n-t.-butylcarbamoyl)-4-aza-5alpha-androst-1-en-3-one and pharmaceutical compositions containing it
US5120847A (en) * 1990-08-27 1992-06-09 Merck & Co., Inc. Process for iodinating or brominating the α-methylenic carbon of a secondary amide
GB9216329D0 (en) * 1992-07-31 1992-09-16 Erba Carlo Spa 17beta-substituted 4-aza-5alpha-androstan-3-one derivatives
GB9216284D0 (en) * 1992-07-31 1992-09-16 Erba Carlo Spa Fluorinated 17beta-substituted 4-aza-5alpha-androstane-3-one derivatives

Also Published As

Publication number Publication date
AU681585B2 (en) 1997-09-04
AU4352693A (en) 1995-01-17
WO1995000531A1 (en) 1995-01-05
RU2109746C1 (ru) 1998-04-27
KR100279567B1 (ko) 2001-03-02
FI115837B (enExample) 2005-07-29
KR960703133A (ko) 1996-06-19
EP0705272A1 (en) 1996-04-10
JP3253088B2 (ja) 2002-02-04
EP0705272B1 (en) 2002-03-27
CA2166090A1 (en) 1995-01-05
FI956236A7 (fi) 1995-12-22
DE69331763T2 (de) 2002-10-02
PT705272E (pt) 2002-07-31
CA2166090C (en) 2006-01-24
ATE215092T1 (de) 2002-04-15
DE69331763D1 (de) 2002-05-02
ES2173889T3 (es) 2002-11-01
UA41933C2 (uk) 2001-10-15
JPH08511796A (ja) 1996-12-10
FI956236A0 (fi) 1995-12-22

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