DK0545966T3 - Phospholipidderivater af nucleosider, deres fremstilling samt deres anvendelse som anti-virale lægemidler - Google Patents

Phospholipidderivater af nucleosider, deres fremstilling samt deres anvendelse som anti-virale lægemidler

Info

Publication number
DK0545966T3
DK0545966T3 DK91914553.2T DK91914553T DK0545966T3 DK 0545966 T3 DK0545966 T3 DK 0545966T3 DK 91914553 T DK91914553 T DK 91914553T DK 0545966 T3 DK0545966 T3 DK 0545966T3
Authority
DK
Denmark
Prior art keywords
preparation
nucleosides
viral drugs
phospholipid derivatives
compounds
Prior art date
Application number
DK91914553.2T
Other languages
English (en)
Inventor
Alfred Mertens
Harald Zilch
Dieter Herrmann
Herbert Leinert
Original Assignee
Boehringer Mannheim Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25896049&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK0545966(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Mannheim Gmbh filed Critical Boehringer Mannheim Gmbh
Application granted granted Critical
Publication of DK0545966T3 publication Critical patent/DK0545966T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals
    • C07H19/10—Pyrimidine radicals with the saccharide radical esterified by phosphoric or polyphosphoric acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • C07H19/20—Purine radicals with the saccharide radical esterified by phosphoric or polyphosphoric acids
    • C—CHEMISTRY; METALLURGY
    • C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P19/00—Preparation of compounds containing saccharide radicals
    • C12P19/26—Preparation of nitrogen-containing carbohydrates
    • C12P19/28—N-glycosides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Microbiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Engineering & Computer Science (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DK91914553.2T 1990-08-20 1991-08-14 Phospholipidderivater af nucleosider, deres fremstilling samt deres anvendelse som anti-virale lægemidler DK0545966T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4026265A DE4026265A1 (de) 1990-08-20 1990-08-20 Neue phospholipid-derivate von nucleosiden, deren herstellung sowie deren verwendung als antivirale arzneimittel
US08/661,038 US5756711A (en) 1990-08-20 1996-06-10 Phospholipid derivatives of nucleosides and their use as anti-viral medicaments

Publications (1)

Publication Number Publication Date
DK0545966T3 true DK0545966T3 (da) 1995-05-08

Family

ID=25896049

Family Applications (1)

Application Number Title Priority Date Filing Date
DK91914553.2T DK0545966T3 (da) 1990-08-20 1991-08-14 Phospholipidderivater af nucleosider, deres fremstilling samt deres anvendelse som anti-virale lægemidler

Country Status (15)

Country Link
US (1) US5756711A (da)
EP (1) EP0545966B1 (da)
CN (1) CN1032258C (da)
AT (1) ATE114316T1 (da)
CA (1) CA2090024C (da)
DE (2) DE4026265A1 (da)
DK (1) DK0545966T3 (da)
ES (1) ES2066461T3 (da)
FI (1) FI104176B (da)
HK (1) HK35597A (da)
IE (1) IE64374B1 (da)
NO (1) NO179710C (da)
PT (1) PT98720B (da)
SK (1) SK281826B6 (da)
WO (1) WO1992003462A1 (da)

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Also Published As

Publication number Publication date
DE4026265A1 (de) 1992-02-27
IE912930A1 (en) 1992-02-26
AU8325191A (en) 1992-03-17
SK9293A3 (en) 1993-07-07
CN1059149A (zh) 1992-03-04
WO1992003462A1 (de) 1992-03-05
CA2090024C (en) 2000-05-02
CA2090024A1 (en) 1992-02-21
NO179710C (no) 1996-12-04
PT98720A (pt) 1992-07-31
AU654670B2 (en) 1994-11-17
EP0545966A1 (de) 1993-06-16
EP0545966B1 (de) 1994-11-23
US5756711A (en) 1998-05-26
NO930587L (no) 1993-02-19
FI104176B1 (fi) 1999-11-30
HK35597A (en) 1997-03-27
SK281826B6 (sk) 2001-08-06
IE64374B1 (en) 1995-07-26
ATE114316T1 (de) 1994-12-15
ES2066461T3 (es) 1995-03-01
FI104176B (fi) 1999-11-30
DE59103595D1 (de) 1995-01-05
FI930753A0 (fi) 1993-02-19
PT98720B (pt) 1999-02-26
FI930753A (fi) 1993-02-19
CN1032258C (zh) 1996-07-10
NO930587D0 (no) 1993-02-19
NO179710B (no) 1996-08-26

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