DE69021826D1 - Verfahren für 1H-Imidazo[4,5-c]-Chinoline. - Google Patents

Verfahren für 1H-Imidazo[4,5-c]-Chinoline.

Info

Publication number
DE69021826D1
DE69021826D1 DE69021826T DE69021826T DE69021826D1 DE 69021826 D1 DE69021826 D1 DE 69021826D1 DE 69021826 T DE69021826 T DE 69021826T DE 69021826 T DE69021826 T DE 69021826T DE 69021826 D1 DE69021826 D1 DE 69021826D1
Authority
DE
Germany
Prior art keywords
quinolines
imidazo
intermediates
chem
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69021826T
Other languages
English (en)
Other versions
DE69021826T2 (de
Inventor
Jean-Denis Andre
Daniel Jean-Marie Lagain
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Meda AB
Original Assignee
Riker Laboratories Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Riker Laboratories Inc filed Critical Riker Laboratories Inc
Application granted granted Critical
Publication of DE69021826D1 publication Critical patent/DE69021826D1/de
Publication of DE69021826T2 publication Critical patent/DE69021826T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • C07D215/42—Nitrogen atoms attached in position 4
    • C07D215/44—Nitrogen atoms attached in position 4 with aryl radicals attached to said nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • C07D215/42—Nitrogen atoms attached in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Cephalosporin Compounds (AREA)
DE69021826T 1989-10-26 1990-10-26 Verfahren für 1H-Imidazo[4,5-c]-Chinoline. Expired - Lifetime DE69021826T2 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/426,677 US4988815A (en) 1989-10-26 1989-10-26 3-Amino or 3-nitro quinoline compounds which are intermediates in preparing 1H-imidazo[4,5-c]quinolines

Publications (2)

Publication Number Publication Date
DE69021826D1 true DE69021826D1 (de) 1995-09-28
DE69021826T2 DE69021826T2 (de) 1996-04-18

Family

ID=23691769

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69021826T Expired - Lifetime DE69021826T2 (de) 1989-10-26 1990-10-26 Verfahren für 1H-Imidazo[4,5-c]-Chinoline.

Country Status (16)

Country Link
US (3) US4988815A (de)
EP (1) EP0425306B1 (de)
JP (1) JP2945121B2 (de)
KR (1) KR0162897B1 (de)
AT (1) ATE126790T1 (de)
AU (1) AU641693B2 (de)
BR (1) BR9005452A (de)
CA (1) CA2027245C (de)
DE (1) DE69021826T2 (de)
ES (1) ES2075168T3 (de)
HK (1) HK1006569A1 (de)
HU (1) HU210051B (de)
IE (1) IE63419B1 (de)
NO (1) NO175530C (de)
RU (1) RU2083563C1 (de)
ZA (1) ZA908193B (de)

Families Citing this family (212)

* Cited by examiner, † Cited by third party
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US5622965A (en) * 1993-03-12 1997-04-22 State Of Oregon, Acting By And Through The Oregon State Board Of Higher Education, Acting For And On Behalf Of The Oregon Health Sciences University And The University Of Oregon, Eugene Oregon 4-hydroxy-3-nitro-1,2-dihydroquinolin-2-ones and the use thereof as excitatory amino acid and glycine receptor antagonists
US5648516A (en) * 1994-07-20 1997-07-15 Minnesota Mining And Manufacturing Company Fused cycloalkylimidazopyridines
EP0708772B1 (de) * 1993-07-15 2000-08-23 Minnesota Mining And Manufacturing Company IMIDAZO [4,5-c]PYRIDIN-4-AMINE
US5352784A (en) * 1993-07-15 1994-10-04 Minnesota Mining And Manufacturing Company Fused cycloalkylimidazopyridines
US5644063A (en) * 1994-09-08 1997-07-01 Minnesota Mining And Manufacturing Company Imidazo[4,5-c]pyridin-4-amine intermediates
US5693811A (en) * 1996-06-21 1997-12-02 Minnesota Mining And Manufacturing Company Process for preparing tetrahdroimidazoquinolinamines
US5741908A (en) * 1996-06-21 1998-04-21 Minnesota Mining And Manufacturing Company Process for reparing imidazoquinolinamines
JP4101302B2 (ja) * 1997-01-09 2008-06-18 テルモ株式会社 新規アミド誘導体および合成中間体
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US5602256A (en) 1997-02-11
IE903597A1 (en) 1991-05-08
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DE69021826T2 (de) 1996-04-18
US4988815A (en) 1991-01-29
ZA908193B (en) 1991-08-28
NO175530B (no) 1994-07-18
US5578727A (en) 1996-11-26
HK1006569A1 (en) 1999-03-05
AU6392890A (en) 1991-07-04
AU641693B2 (en) 1993-09-30
EP0425306A3 (en) 1992-01-08
NO904625L (no) 1991-04-29
HU906404D0 (en) 1991-04-29
HUT55777A (en) 1991-06-28
ATE126790T1 (de) 1995-09-15
RU2083563C1 (ru) 1997-07-10
NO904625D0 (no) 1990-10-25
KR0162897B1 (ko) 1998-12-01
EP0425306B1 (de) 1995-08-23
IE63419B1 (en) 1995-04-19
JP2945121B2 (ja) 1999-09-06
CA2027245C (en) 1999-08-17
ES2075168T3 (es) 1995-10-01
JPH03206078A (ja) 1991-09-09
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KR910007926A (ko) 1991-05-30
BR9005452A (pt) 1991-09-17

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