DE60028538T2 - Kondensierte heterocyclische verbindungen und ihre verwendung zur behandlung von neurodegenerativen erkrankungen - Google Patents
Kondensierte heterocyclische verbindungen und ihre verwendung zur behandlung von neurodegenerativen erkrankungen Download PDFInfo
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- DE60028538T2 DE60028538T2 DE60028538T DE60028538T DE60028538T2 DE 60028538 T2 DE60028538 T2 DE 60028538T2 DE 60028538 T DE60028538 T DE 60028538T DE 60028538 T DE60028538 T DE 60028538T DE 60028538 T2 DE60028538 T2 DE 60028538T2
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- tetrahydropyridine
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- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Psychology (AREA)
- Ophthalmology & Optometry (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA199900061 | 1999-01-19 | ||
| DK9900061 | 1999-01-19 | ||
| PCT/DK2000/000012 WO2000043397A1 (en) | 1999-01-19 | 2000-01-13 | Fused heterocyclic compounds and their use in the treatment of neurodegenerative diseases |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE60028538D1 DE60028538D1 (de) | 2006-07-20 |
| DE60028538T2 true DE60028538T2 (de) | 2007-06-21 |
Family
ID=8089290
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE60028538T Expired - Lifetime DE60028538T2 (de) | 1999-01-19 | 2000-01-13 | Kondensierte heterocyclische verbindungen und ihre verwendung zur behandlung von neurodegenerativen erkrankungen |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US6576641B2 (enExample) |
| EP (1) | EP1147113B1 (enExample) |
| JP (1) | JP2002535334A (enExample) |
| CN (1) | CN1147490C (enExample) |
| AT (1) | ATE328887T1 (enExample) |
| AU (1) | AU776276B2 (enExample) |
| CA (1) | CA2353903A1 (enExample) |
| DE (1) | DE60028538T2 (enExample) |
| NZ (1) | NZ512289A (enExample) |
| WO (1) | WO2000043397A1 (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1432708B1 (en) * | 2001-09-24 | 2005-11-30 | Bayer Pharmaceuticals Corporation | Preparation and use of 1,5,6,7-tetrahydropyrrolo 3,2-c]pyridine derivatives for treatment of obesity |
| KR100553398B1 (ko) * | 2004-03-12 | 2006-02-16 | 한미약품 주식회사 | 티에노[3,2-ｃ]피리딘 유도체의 제조 방법 및 이에사용되는 중간체 |
| CN104193761B (zh) | 2009-12-04 | 2017-10-17 | 桑诺维恩药品公司 | 多环化合物及其使用方法 |
| BR112019001407A2 (pt) | 2016-07-29 | 2019-07-09 | Sunovion Pharmaceuticals Inc. | compostos e composições e usos dos mesmos |
| SG10202100724UA (en) | 2016-07-29 | 2021-03-30 | Sunovion Pharmaceuticals Inc | Compounds and compositions and uses thereof |
| EP3582815A1 (en) | 2017-02-16 | 2019-12-25 | Sunovion Pharmaceuticals Inc. | Methods of treating schizophrenia |
| MX2020000523A (es) | 2017-08-02 | 2020-08-20 | Sunovion Pharmaceuticals Inc | Compuestos de isocromano y usos de los mismos. |
| SG11202007823PA (en) | 2018-02-16 | 2020-09-29 | Sunovion Pharmaceuticals Inc | Salts, crystal forms, and production methods thereof |
| JP7703449B2 (ja) | 2019-03-14 | 2025-07-07 | スミトモ・ファーマ・アメリカ・インコーポレイテッド | イソクロマニル化合物の塩およびその結晶体、ならびにそれらの製造方法、治療用途および医薬組成物 |
| KR20230003503A (ko) | 2020-04-14 | 2023-01-06 | 선오비온 파마슈티컬스 인코포레이티드 | 신경학적 및 정신의학적 장애의 치료를 위한 (S)-(4,5-디히드로-7H-티에노[2,3-c]피란-7-일)-N-메틸메탄아민 |
| KR20240101561A (ko) | 2021-10-14 | 2024-07-02 | 인사이트 코포레이션 | Kras의 저해제로서의 퀴놀린 화합물 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2395028A2 (fr) * | 1977-06-22 | 1979-01-19 | Centre Etd Ind Pharma | Derives pyridiniques, leur preparation et leurs application therapeutique |
| FR2566775B1 (fr) | 1984-06-27 | 1986-10-31 | Synthelabo | Derives de tetrahydro-4,5,6,7 furo ou 1h-pyrrolo(2,3-c)pyridine, leur preparation et leur application en therapeutique |
| FR2570701B1 (fr) * | 1984-09-27 | 1987-05-22 | Synthelabo | Derives de furo(3,2-c)pyridines, leur preparation et leur application en therapeutique |
| FR2635977B1 (fr) * | 1988-09-07 | 1992-05-15 | Synthelabo | Utilisation de derives de tetrahydro-4,5,6,7 furopyridines pour obtenir des medicaments destines au traitement de l'obesite |
| GB8921465D0 (en) * | 1989-09-22 | 1989-11-08 | Fujisawa Pharmaceutical Co | Bicyclic amine compound and a process for the preparation thereof |
| FR2652579B1 (fr) * | 1989-10-02 | 1992-01-24 | Sanofi Sa | Derives d'hydroxy-2 thiophene et furanne condenses avec un cycle azote, sur procede de preparation et leur application en therapeutique. |
| FI101150B (fi) * | 1991-09-09 | 1998-04-30 | Sankyo Co | Menetelmä lääkeaineina käyttökelpoisten tetrahydrotienopyridiinin johd annaisten valmistamiseksi |
| AU3619795A (en) * | 1994-10-11 | 1996-05-02 | Takeda Chemical Industries Ltd. | Substituted heterobicyclic alkyl amines and their use as squalene oxide cyclase inhibitors |
| EP0863878B1 (en) * | 1995-09-11 | 2003-01-08 | Aventis Pharmaceuticals Inc. | Cyclic nitrones and pharmaceutical compositions containing them |
-
2000
- 2000-01-13 NZ NZ512289A patent/NZ512289A/xx not_active IP Right Cessation
- 2000-01-13 CN CNB008027080A patent/CN1147490C/zh not_active Expired - Fee Related
- 2000-01-13 DE DE60028538T patent/DE60028538T2/de not_active Expired - Lifetime
- 2000-01-13 WO PCT/DK2000/000012 patent/WO2000043397A1/en not_active Ceased
- 2000-01-13 AT AT00900497T patent/ATE328887T1/de not_active IP Right Cessation
- 2000-01-13 JP JP2000594813A patent/JP2002535334A/ja active Pending
- 2000-01-13 CA CA002353903A patent/CA2353903A1/en not_active Abandoned
- 2000-01-13 AU AU30333/00A patent/AU776276B2/en not_active Ceased
- 2000-01-13 EP EP00900497A patent/EP1147113B1/en not_active Expired - Lifetime
-
2001
- 2001-06-07 US US09/875,019 patent/US6576641B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US20020013336A1 (en) | 2002-01-31 |
| CN1147490C (zh) | 2004-04-28 |
| CA2353903A1 (en) | 2000-07-27 |
| US6576641B2 (en) | 2003-06-10 |
| AU776276B2 (en) | 2004-09-02 |
| WO2000043397A1 (en) | 2000-07-27 |
| AU3033300A (en) | 2000-08-07 |
| EP1147113A1 (en) | 2001-10-24 |
| EP1147113B1 (en) | 2006-06-07 |
| ATE328887T1 (de) | 2006-06-15 |
| JP2002535334A (ja) | 2002-10-22 |
| DE60028538D1 (de) | 2006-07-20 |
| CN1336929A (zh) | 2002-02-20 |
| NZ512289A (en) | 2003-06-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8364 | No opposition during term of opposition |