DE3001011C2 - Verwendung von Carbostyrilderivaten - Google Patents

Verwendung von Carbostyrilderivaten

Info

Publication number
DE3001011C2
DE3001011C2 DE3001011A DE3001011A DE3001011C2 DE 3001011 C2 DE3001011 C2 DE 3001011C2 DE 3001011 A DE3001011 A DE 3001011A DE 3001011 A DE3001011 A DE 3001011A DE 3001011 C2 DE3001011 C2 DE 3001011C2
Authority
DE
Germany
Prior art keywords
hydroxy
propoxy
dihydrocarbostyril
glaucoma
tert
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
DE3001011A
Other languages
German (de)
English (en)
Other versions
DE3001011A1 (de
Inventor
Kazuyuki Tokushima Nakagawa
Yoichi Ibaragi Osaka Nishinakamura
Nobuyuki Tokushima Tanaka
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Otsuka Pharmaceutical Co Ltd
Original Assignee
Otsuka Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26345304&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE3001011(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from JP54010108A external-priority patent/JPS5951927B2/ja
Priority claimed from JP54070361A external-priority patent/JPS5951928B2/ja
Application filed by Otsuka Pharmaceutical Co Ltd filed Critical Otsuka Pharmaceutical Co Ltd
Publication of DE3001011A1 publication Critical patent/DE3001011A1/de
Application granted granted Critical
Publication of DE3001011C2 publication Critical patent/DE3001011C2/de
Expired legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DE3001011A 1979-01-30 1980-01-12 Verwendung von Carbostyrilderivaten Expired DE3001011C2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP54010108A JPS5951927B2 (ja) 1979-01-30 1979-01-30 緑内障治療剤
JP54070361A JPS5951928B2 (ja) 1979-06-04 1979-06-04 緑内障治療剤

Publications (2)

Publication Number Publication Date
DE3001011A1 DE3001011A1 (de) 1980-08-28
DE3001011C2 true DE3001011C2 (de) 1986-02-06

Family

ID=26345304

Family Applications (1)

Application Number Title Priority Date Filing Date
DE3001011A Expired DE3001011C2 (de) 1979-01-30 1980-01-12 Verwendung von Carbostyrilderivaten

Country Status (15)

Country Link
US (1) US4309432A (US20030220297A1-20031127-C00074.png)
AT (1) AT371340B (US20030220297A1-20031127-C00074.png)
AU (1) AU518814B2 (US20030220297A1-20031127-C00074.png)
CA (1) CA1139669A (US20030220297A1-20031127-C00074.png)
CH (1) CH646057A5 (US20030220297A1-20031127-C00074.png)
DE (1) DE3001011C2 (US20030220297A1-20031127-C00074.png)
DK (1) DK11580A (US20030220297A1-20031127-C00074.png)
ES (1) ES8100268A1 (US20030220297A1-20031127-C00074.png)
FI (1) FI800089A (US20030220297A1-20031127-C00074.png)
FR (1) FR2447721A1 (US20030220297A1-20031127-C00074.png)
GB (1) GB2042338B (US20030220297A1-20031127-C00074.png)
IT (1) IT1141662B (US20030220297A1-20031127-C00074.png)
NL (1) NL191575C (US20030220297A1-20031127-C00074.png)
NO (1) NO800059L (US20030220297A1-20031127-C00074.png)
SE (1) SE451069B (US20030220297A1-20031127-C00074.png)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0056420A1 (en) * 1981-01-15 1982-07-28 Schering Corporation Ophthalmic gel
FR2539413A1 (fr) * 1983-01-17 1984-07-20 Pos Lab Carbostyriloximinopropanolamines utiles comme medicaments et procede pour leur preparation
US4921862A (en) * 1986-05-29 1990-05-01 Syntex (U.S.A.) Inc. Carbostyril derivatives as combined thromboxane synthetase and cyclic-amp phosphodiesterase inhibitors
US4792561A (en) * 1986-05-29 1988-12-20 Syntex (U.S.A.) Inc. Carbostyril derivatives as combined thromboxane synthetase and cyclic-AMP phosphodiesterase inhibitors
DE68920797T2 (de) * 1988-08-10 1995-06-29 Otsuka Pharma Co Ltd Herzmittel.
US5198448A (en) * 1988-08-10 1993-03-30 Otsuka Pharmaceutical Company, Limited Cardiotonics
DE69019774T2 (de) * 1989-03-28 1995-11-09 Nisshin Flour Milling Co Isochinolin-Derivate zur Behandlung des Glaukoms oder der okulären Hypertonie.
FR2676740B1 (fr) * 1991-05-23 1993-11-05 Roussel Uclaf Nouveaux derives sterouides du pregna-4,9(11),17(20)-trie-3-one, leur preparation, leur application a la preparation de composes sterouides de type pregna-4,9(11),16-triene-3,20-dione et nouveaux intermediaires.
US5629345A (en) * 1993-07-23 1997-05-13 Vide Pharmaceuticals Methods and compositions for ATP-sensitive K+ channel inhibition for lowering intraocular pressure
US5965620A (en) * 1993-07-23 1999-10-12 Vide Pharmaceuticals Methods and compositions for ATP-sensitive K+ channel inhibition for lowering intraocular pressure
US5776482A (en) * 1996-03-29 1998-07-07 University Of Iowa Research Foundation Tetrahydroquinoline analogues for use in glaucoma treatment
MY116782A (en) 1997-12-22 2004-03-31 Otsuka Pharma Co Ltd Water-soluble eye drop
CA2671747C (en) * 2006-12-06 2016-03-15 U.S. Borax Inc. Animal feed compositions

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3910924A (en) * 1972-04-13 1975-10-07 Otsuka Pharma Co Ltd 3,4-Dihydrocarbostyril derivatives and a process for preparing the same
JPS517672B2 (US20030220297A1-20031127-C00074.png) * 1972-04-13 1976-03-10
AR207554A1 (es) * 1972-12-02 1976-10-15 Otsuka Pharma Co Ltd Procedimiento para producir derivados de 3-alquil-5-((3,4-dihidro-5-carbostiril)oximetil)-oxazolidinona-(2)
JPS5239035B2 (US20030220297A1-20031127-C00074.png) * 1972-12-14 1977-10-03
US3975391A (en) * 1973-12-26 1976-08-17 Otsuka Pharmaceutical Company Limited 5-[1-Hydroxy-2-(substituted-amino)]ethyl-8-hydroxy-3,4-dihydrocarbostyril derivatives
AU467612B2 (en) * 1973-07-31 1975-12-04 Novel organophosphorous pesticide
JPS5082218A (US20030220297A1-20031127-C00074.png) * 1973-11-10 1975-07-03
US3994901A (en) * 1974-06-13 1976-11-30 Otsuka Pharmaceutical Company Limited 5-[1-Hydroxy-2-(substituted-amino)]alkyl-8-hydroxy-3,4-dihydrocarbostyril derivatives
US4081447A (en) * 1975-04-09 1978-03-28 Abbott Laboratories 5-[2-Hydroxy-3-(3,4-dimethoxy phenethylamino)]-propoxy-3,4-dihydro carbostyril and pharmaceutically acceptable salts thereof
US4210753A (en) * 1976-03-17 1980-07-01 Otsuka Pharmaceutical Co., Ltd. Carbostyril compounds
CH619453A5 (US20030220297A1-20031127-C00074.png) * 1976-03-17 1980-09-30 Otsuka Pharma Co Ltd
DE2719562C2 (de) * 1976-05-08 1986-05-07 Otsuka Pharmaceutical Co. Ltd., Tokio/Tokyo 3, 4-Dihydrocarbostyrilderivate, Verfahren zu deren Herstellung und Arzneimittel, welche diese enthalten
JPS552631A (en) * 1978-06-19 1980-01-10 Otsuka Pharmaceut Co Ltd 3,4-dihydrocarbostyril derivative
JPS5513241A (en) * 1978-07-14 1980-01-30 Otsuka Pharmaceut Co Ltd Remedy for glaucoma

Also Published As

Publication number Publication date
DE3001011A1 (de) 1980-08-28
ATA14480A (de) 1982-11-15
NL8000211A (nl) 1980-08-01
IT1141662B (it) 1986-10-08
FR2447721B1 (US20030220297A1-20031127-C00074.png) 1983-03-11
CH646057A5 (de) 1984-11-15
FR2447721A1 (fr) 1980-08-29
GB2042338A (en) 1980-09-24
NL191575C (nl) 1995-10-03
AU5426579A (en) 1980-08-07
FI800089A (fi) 1980-07-31
SE8000245L (sv) 1980-07-31
SE451069B (sv) 1987-08-31
NL191575B (nl) 1995-06-01
NO800059L (no) 1980-07-31
US4309432A (en) 1982-01-05
ES487642A0 (es) 1980-11-01
IT8005106A0 (it) 1980-01-09
CA1139669A (en) 1983-01-18
AU518814B2 (en) 1981-10-22
ES8100268A1 (es) 1980-11-01
DK11580A (da) 1980-07-31
GB2042338B (en) 1983-11-30
AT371340B (de) 1983-06-27

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Legal Events

Date Code Title Description
OAP Request for examination filed
OD Request for examination
D2 Grant after examination
8328 Change in the person/name/address of the agent

Free format text: SOLF, A., DR.-ING., 8000 MUENCHEN ZAPF, C., DIPL.-ING., PAT.-ANW., 5600 WUPPERTAL

8364 No opposition during term of opposition