DE2660626C2 - 3-Amino-2-hydroxy-4-phenyl-butansäure-Derivate und Verfahren zu ihrer Herstellung - Google Patents

3-Amino-2-hydroxy-4-phenyl-butansäure-Derivate und Verfahren zu ihrer Herstellung

Info

Publication number
DE2660626C2
DE2660626C2 DE2660626A DE2660626A DE2660626C2 DE 2660626 C2 DE2660626 C2 DE 2660626C2 DE 2660626 A DE2660626 A DE 2660626A DE 2660626 A DE2660626 A DE 2660626A DE 2660626 C2 DE2660626 C2 DE 2660626C2
Authority
DE
Germany
Prior art keywords
ahpa
amino
hydroxy
acid
ethyl acetate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
DE2660626A
Other languages
German (de)
English (en)
Inventor
Takaaki Fujisawa Kanagawa Aoyagi
Rinzo Nishizawa
Tetsushi Tokio/Tokyo Saino
Tomohisa Asaki Saitama Takita
Hamao Tokio/Tokyo Umezawa
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Microbial Chemistry Research Foundation
Original Assignee
Microbial Chemistry Research Foundation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Microbial Chemistry Research Foundation filed Critical Microbial Chemistry Research Foundation
Application granted granted Critical
Publication of DE2660626C2 publication Critical patent/DE2660626C2/de
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DE2660626A 1975-07-22 1976-07-19 3-Amino-2-hydroxy-4-phenyl-butansäure-Derivate und Verfahren zu ihrer Herstellung Expired DE2660626C2 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB30632/75A GB1510477A (en) 1975-07-22 1975-07-22 Peptides and to amino acid intermediates thereof

Publications (1)

Publication Number Publication Date
DE2660626C2 true DE2660626C2 (de) 1985-07-11

Family

ID=10310676

Family Applications (2)

Application Number Title Priority Date Filing Date
DE2632396A Expired DE2632396C2 (de) 1975-07-22 1976-07-19 Bestatin-Analoga, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Präparate
DE2660626A Expired DE2660626C2 (de) 1975-07-22 1976-07-19 3-Amino-2-hydroxy-4-phenyl-butansäure-Derivate und Verfahren zu ihrer Herstellung

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DE2632396A Expired DE2632396C2 (de) 1975-07-22 1976-07-19 Bestatin-Analoga, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Präparate

Country Status (12)

Country Link
JP (2) JPS52136118A (cs)
AU (1) AU506003B2 (cs)
CA (1) CA1104156A (cs)
CH (1) CH630892A5 (cs)
CS (2) CS201034B2 (cs)
DE (2) DE2632396C2 (cs)
DK (1) DK149110C (cs)
FR (1) FR2318863A1 (cs)
GB (1) GB1510477A (cs)
HU (1) HU183048B (cs)
NL (1) NL7608064A (cs)
SE (3) SE431642B (cs)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2725732C2 (de) 1977-06-07 1983-01-05 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai, Tokyo Bestatin-Analoga, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Präparate
DE2760007C2 (cs) * 1977-06-07 1988-10-06 Microbial Chem Res Found
JPS6026099B2 (ja) * 1977-09-21 1985-06-21 財団法人微生物化学研究会 ペプチド、その酸附加塩およびその製造法
DE2954076C2 (cs) * 1978-11-25 1988-02-25 Nippon Kayaku K.K., Tokio/Tokyo, Jp
US4370318A (en) * 1980-07-07 1983-01-25 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai Bestatin-related compounds as immunopotentiator
JPS5767516A (en) * 1980-09-24 1982-04-24 Microbial Chem Res Found Novel analgesic agent
JPH0810855Y2 (ja) * 1989-07-20 1996-03-29 タナシン電機株式会社 オートリバース式テープレコーダ
DE69420524T2 (de) * 1993-06-29 2000-02-17 Kaneka Corp., Osaka Verfahren zur herstellung von derivaten von 3-amin-2-hydroxy-4-phenylbuttersäure und 1-nitro-4-phenyl-2-butanol zwischenprodukte
CA2236117C (en) * 1996-02-08 2004-11-16 Nippon Kayaku Kabushiki Kaisha Process for producing optically active cyanohydrins
BR9910092A (pt) * 1998-05-01 2002-01-22 Abbott Lab Inibidores de beta-aminoácido substituìdo de metionina aminopeptidase-2
US6242494B1 (en) 1998-05-01 2001-06-05 Abbott Laboratories Substituted β-amino acid inhibitors of methionine aminopeptidase-2

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5439477B2 (cs) * 1974-07-01 1979-11-28

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
NICHTS-ERMITTELT *

Also Published As

Publication number Publication date
DE2632396A1 (de) 1977-02-03
DE2632396C2 (de) 1982-11-25
DK149110B (da) 1986-01-27
GB1510477A (en) 1978-05-10
CS201033B2 (en) 1980-10-31
AU506003B2 (en) 1979-12-13
SE452318B (sv) 1987-11-23
CH630892A5 (en) 1982-07-15
FR2318863B1 (cs) 1980-10-31
SE8306145D0 (sv) 1983-11-09
SE8306145L (sv) 1983-11-09
CA1104156A (en) 1981-06-30
FR2318863A1 (fr) 1977-02-18
DK331276A (da) 1977-01-23
JPS5758338B2 (cs) 1982-12-09
CS201034B2 (en) 1980-10-31
SE8001959L (sv) 1980-03-13
JPS5823654A (ja) 1983-02-12
JPS52136118A (en) 1977-11-14
SE7606736L (sv) 1977-01-23
DK149110C (da) 1986-09-08
AU1591276A (en) 1978-01-19
JPS6050780B2 (ja) 1985-11-11
SE431642B (sv) 1984-02-20
HU183048B (en) 1984-04-28
NL7608064A (nl) 1977-01-25

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