DK149110C - Analogifremgangsmaade til fremstilling af bestatin eller et analogt dipeptid samt alfa-hydroxy-beta-aminocarboxylsyrer til brug som udgangsforbindelser herfor - Google Patents

Analogifremgangsmaade til fremstilling af bestatin eller et analogt dipeptid samt alfa-hydroxy-beta-aminocarboxylsyrer til brug som udgangsforbindelser herfor

Info

Publication number
DK149110C
DK149110C DK331276A DK331276A DK149110C DK 149110 C DK149110 C DK 149110C DK 331276 A DK331276 A DK 331276A DK 331276 A DK331276 A DK 331276A DK 149110 C DK149110 C DK 149110C
Authority
DK
Denmark
Prior art keywords
analogue
bestatine
dipeptide
alfa
beta
Prior art date
Application number
DK331276A
Other languages
English (en)
Other versions
DK149110B (da
DK331276A (da
Inventor
Hamao Umezawa
Takaaki Aoyagi
Tomohisa Takita
Rinzo Nishizawa
Tetsushi Saino
Original Assignee
Microbial Chem Res Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Microbial Chem Res Found filed Critical Microbial Chem Res Found
Publication of DK331276A publication Critical patent/DK331276A/da
Publication of DK149110B publication Critical patent/DK149110B/da
Application granted granted Critical
Publication of DK149110C publication Critical patent/DK149110C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK331276A 1975-07-22 1976-07-22 Analogifremgangsmaade til fremstilling af bestatin eller et analogt dipeptid samt alfa-hydroxy-beta-aminocarboxylsyrer til brug som udgangsforbindelser herfor DK149110C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB3063275 1975-07-22
GB30632/75A GB1510477A (en) 1975-07-22 1975-07-22 Peptides and to amino acid intermediates thereof

Publications (3)

Publication Number Publication Date
DK331276A DK331276A (da) 1977-01-23
DK149110B DK149110B (da) 1986-01-27
DK149110C true DK149110C (da) 1986-09-08

Family

ID=10310676

Family Applications (1)

Application Number Title Priority Date Filing Date
DK331276A DK149110C (da) 1975-07-22 1976-07-22 Analogifremgangsmaade til fremstilling af bestatin eller et analogt dipeptid samt alfa-hydroxy-beta-aminocarboxylsyrer til brug som udgangsforbindelser herfor

Country Status (12)

Country Link
JP (2) JPS52136118A (da)
AU (1) AU506003B2 (da)
CA (1) CA1104156A (da)
CH (1) CH630892A5 (da)
CS (2) CS201034B2 (da)
DE (2) DE2660626C2 (da)
DK (1) DK149110C (da)
FR (1) FR2318863A1 (da)
GB (1) GB1510477A (da)
HU (1) HU183048B (da)
NL (1) NL7608064A (da)
SE (3) SE431642B (da)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2760007C2 (da) * 1977-06-07 1988-10-06 Microbial Chem Res Found
DE2725732C2 (de) 1977-06-07 1983-01-05 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai, Tokyo Bestatin-Analoga, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Präparate
JPS6026099B2 (ja) * 1977-09-21 1985-06-21 財団法人微生物化学研究会 ペプチド、その酸附加塩およびその製造法
CA1182125A (en) * 1978-11-25 1985-02-05 Hamao Umezawa Process for producing threo-3-amino-2- hydroxybutanoyl-aminoacetic acids, as well as novel intermediates therefor and process for producing them
US4370318A (en) * 1980-07-07 1983-01-25 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai Bestatin-related compounds as immunopotentiator
JPS5767516A (en) * 1980-09-24 1982-04-24 Microbial Chem Res Found Novel analgesic agent
JPH0810855Y2 (ja) * 1989-07-20 1996-03-29 タナシン電機株式会社 オートリバース式テープレコーダ
EP0657415B1 (en) * 1993-06-29 1999-09-08 Kaneka Corporation Method of producing 3-amino-2-hydroxy-4-phenyl-butyric acid derivatives and 3-amino-1-nitro-4-phenyl-2-butanol intermediates
CN1073555C (zh) * 1996-02-08 2001-10-24 日本化药株式会社 制备旋光性氰醇的方法
SK16282000A3 (sk) * 1998-05-01 2001-05-10 Abbott Laboratories Substituované beta-aminokyselinové inhibítory metionínaminopeptidázy-2
US6242494B1 (en) 1998-05-01 2001-06-05 Abbott Laboratories Substituted β-amino acid inhibitors of methionine aminopeptidase-2

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5439477B2 (da) * 1974-07-01 1979-11-28

Also Published As

Publication number Publication date
SE7606736L (sv) 1977-01-23
DK149110B (da) 1986-01-27
NL7608064A (nl) 1977-01-25
FR2318863A1 (fr) 1977-02-18
JPS6050780B2 (ja) 1985-11-11
JPS5758338B2 (da) 1982-12-09
SE8306145L (sv) 1983-11-09
CA1104156A (en) 1981-06-30
JPS5823654A (ja) 1983-02-12
CH630892A5 (en) 1982-07-15
DE2632396C2 (de) 1982-11-25
HU183048B (en) 1984-04-28
AU1591276A (en) 1978-01-19
SE8306145D0 (sv) 1983-11-09
FR2318863B1 (da) 1980-10-31
SE452318B (sv) 1987-11-23
SE431642B (sv) 1984-02-20
DE2632396A1 (de) 1977-02-03
GB1510477A (en) 1978-05-10
AU506003B2 (en) 1979-12-13
DE2660626C2 (de) 1985-07-11
SE8001959L (sv) 1980-03-13
DK331276A (da) 1977-01-23
CS201033B2 (en) 1980-10-31
CS201034B2 (en) 1980-10-31
JPS52136118A (en) 1977-11-14

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