DD210040A5 - Verfahren zur herstellung von 4-phenyl-chinazolin-derivaten - Google Patents

Verfahren zur herstellung von 4-phenyl-chinazolin-derivaten Download PDF

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Publication number
DD210040A5
DD210040A5 DD82244148A DD24414882A DD210040A5 DD 210040 A5 DD210040 A5 DD 210040A5 DD 82244148 A DD82244148 A DD 82244148A DD 24414882 A DD24414882 A DD 24414882A DD 210040 A5 DD210040 A5 DD 210040A5
Authority
DD
German Democratic Republic
Prior art keywords
group
reaction
amine
preparation
phenyl
Prior art date
Application number
DD82244148A
Other languages
German (de)
English (en)
Inventor
Andre Hallot
Kathleen Biziere
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of DD210040A5 publication Critical patent/DD210040A5/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • C07D239/84Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Luminescent Compositions (AREA)
  • Pyrrole Compounds (AREA)
  • Peptides Or Proteins (AREA)
DD82244148A 1981-10-21 1982-10-20 Verfahren zur herstellung von 4-phenyl-chinazolin-derivaten DD210040A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8119767A FR2514765A1 (fr) 1981-10-21 1981-10-21 Nouveaux derives de la phenyl-4 quinazoline actifs sur le systeme nerveux central

Publications (1)

Publication Number Publication Date
DD210040A5 true DD210040A5 (de) 1984-05-30

Family

ID=9263248

Family Applications (1)

Application Number Title Priority Date Filing Date
DD82244148A DD210040A5 (de) 1981-10-21 1982-10-20 Verfahren zur herstellung von 4-phenyl-chinazolin-derivaten

Country Status (24)

Country Link
US (1) US4499092A (es)
EP (1) EP0079810B1 (es)
JP (1) JPS5888369A (es)
KR (1) KR880001077B1 (es)
AT (1) ATE17576T1 (es)
AU (1) AU551938B2 (es)
CA (1) CA1236102A (es)
CS (1) CS229692B2 (es)
DD (1) DD210040A5 (es)
DE (1) DE3268699D1 (es)
DK (1) DK156063C (es)
ES (1) ES8307226A1 (es)
FI (1) FI73982C (es)
FR (1) FR2514765A1 (es)
GR (1) GR76535B (es)
HU (1) HU187579B (es)
IE (1) IE53653B1 (es)
IL (1) IL66960A0 (es)
NO (1) NO164167C (es)
NZ (1) NZ202237A (es)
PT (1) PT75667B (es)
SU (1) SU1299511A3 (es)
YU (1) YU43528B (es)
ZA (1) ZA827516B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2521144A1 (fr) * 1982-02-08 1983-08-12 Sanofi Sa Nouveaux derives de la piperazinyl-2 phenyl-4 quinazoline possedant des proprietes antidepressives, methode de preparation desdits composes et medicaments en contenant
WO1994007498A1 (en) * 1992-10-07 1994-04-14 Sumitomo Pharmaceuticals Company, Limited Pharmaceutical composition for inhibiting tumor necrosis factor production
JPH11209350A (ja) 1998-01-26 1999-08-03 Eisai Co Ltd 含窒素複素環誘導体およびその医薬
JP2006525357A (ja) * 2003-04-30 2006-11-09 ジ インスチチュート フォー ファーマシューティカル ディスカバリー、エルエルシー プロテインチロシンホスファターゼ阻害物質としての置換ヘテロアリール類
WO2005042501A1 (en) * 2003-11-03 2005-05-12 Warner-Lambert Company Llc Novel norepinephrine reuptake inhibitors for the treatment of central nervous system disorders
EP1899306B1 (en) 2005-06-27 2008-10-15 F. Hoffmann-Roche AG Chloro-substituted guanidines
US7855194B2 (en) 2006-03-27 2010-12-21 Hoffmann-La Roche Inc. Pyrimidine, quinazoline, pteridine and triazine derivatives
BRPI0719111A8 (pt) 2006-11-22 2019-01-15 Sumitomo Chemical Co agente para inibir a sinalização de citocinina

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA894239A (en) * 1972-02-29 Pfizer Inc. Nitrogen heterocycles
US3305553A (en) * 1965-10-18 1967-02-21 Parke Davis & Co 2-aminoquinazoline derivatives
US3509141A (en) * 1966-09-15 1970-04-28 Ciba Geigy Corp 2-amino-quinazolines
GB1347493A (en) * 1971-02-11 1974-02-27 Aspro Nicholas Ltd Benzazine derivatives
JPS5398997A (en) * 1977-02-09 1978-08-29 Sumitomo Chem Co Ltd Fused pyridine derivertives and process for their preparation

Also Published As

Publication number Publication date
US4499092A (en) 1985-02-12
GR76535B (es) 1984-08-10
SU1299511A3 (ru) 1987-03-23
IE822447L (en) 1983-04-21
FR2514765A1 (fr) 1983-04-22
PT75667B (fr) 1985-01-11
DE3268699D1 (en) 1986-03-06
EP0079810B1 (fr) 1986-01-22
NZ202237A (en) 1985-08-30
KR840001968A (ko) 1984-06-07
NO164167C (no) 1990-09-05
ES516694A0 (es) 1983-07-01
NO164167B (no) 1990-05-28
ES8307226A1 (es) 1983-07-01
FI73982C (fi) 1987-12-10
NO823491L (no) 1983-04-22
AU551938B2 (en) 1986-05-15
AU8962882A (en) 1983-04-28
FR2514765B1 (es) 1984-04-06
EP0079810A1 (fr) 1983-05-25
DK156063C (da) 1989-11-13
FI73982B (fi) 1987-08-31
PT75667A (fr) 1982-11-01
ZA827516B (en) 1983-08-31
JPS5888369A (ja) 1983-05-26
IE53653B1 (en) 1989-01-04
DK156063B (da) 1989-06-19
CA1236102A (en) 1988-05-03
CS229692B2 (en) 1984-06-18
FI823580A0 (fi) 1982-10-20
YU43528B (en) 1989-08-31
HU187579B (en) 1986-01-28
KR880001077B1 (ko) 1988-06-22
DK465182A (da) 1983-04-22
IL66960A0 (en) 1983-02-23
YU223382A (en) 1984-10-31
ATE17576T1 (de) 1986-02-15
FI823580L (fi) 1983-04-22

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