ES516694A0 - Procedimiento de preparacion de derivados de la 4-fenil quinazolina. - Google Patents

Procedimiento de preparacion de derivados de la 4-fenil quinazolina.

Info

Publication number
ES516694A0
ES516694A0 ES516694A ES516694A ES516694A0 ES 516694 A0 ES516694 A0 ES 516694A0 ES 516694 A ES516694 A ES 516694A ES 516694 A ES516694 A ES 516694A ES 516694 A0 ES516694 A0 ES 516694A0
Authority
ES
Spain
Prior art keywords
image
derivatives
procedure
preparation
phenyl quinazoline
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES516694A
Other languages
English (en)
Other versions
ES8307226A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi SA
Original Assignee
Sanofi SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi SA filed Critical Sanofi SA
Publication of ES516694A0 publication Critical patent/ES516694A0/es
Publication of ES8307226A1 publication Critical patent/ES8307226A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • C07D239/84Nitrogen atoms
ES516694A 1981-10-21 1982-10-20 Procedimiento de preparacion de derivados de la 4-fenil quinazolina. Expired ES8307226A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8119767A FR2514765A1 (fr) 1981-10-21 1981-10-21 Nouveaux derives de la phenyl-4 quinazoline actifs sur le systeme nerveux central

Publications (2)

Publication Number Publication Date
ES516694A0 true ES516694A0 (es) 1983-07-01
ES8307226A1 ES8307226A1 (es) 1983-07-01

Family

ID=9263248

Family Applications (1)

Application Number Title Priority Date Filing Date
ES516694A Expired ES8307226A1 (es) 1981-10-21 1982-10-20 Procedimiento de preparacion de derivados de la 4-fenil quinazolina.

Country Status (24)

Country Link
US (1) US4499092A (es)
EP (1) EP0079810B1 (es)
JP (1) JPS5888369A (es)
KR (1) KR880001077B1 (es)
AT (1) ATE17576T1 (es)
AU (1) AU551938B2 (es)
CA (1) CA1236102A (es)
CS (1) CS229692B2 (es)
DD (1) DD210040A5 (es)
DE (1) DE3268699D1 (es)
DK (1) DK156063C (es)
ES (1) ES8307226A1 (es)
FI (1) FI73982C (es)
FR (1) FR2514765A1 (es)
GR (1) GR76535B (es)
HU (1) HU187579B (es)
IE (1) IE53653B1 (es)
IL (1) IL66960A0 (es)
NO (1) NO164167C (es)
NZ (1) NZ202237A (es)
PT (1) PT75667B (es)
SU (1) SU1299511A3 (es)
YU (1) YU43528B (es)
ZA (1) ZA827516B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2521144A1 (fr) * 1982-02-08 1983-08-12 Sanofi Sa Nouveaux derives de la piperazinyl-2 phenyl-4 quinazoline possedant des proprietes antidepressives, methode de preparation desdits composes et medicaments en contenant
US5646154A (en) * 1992-10-07 1997-07-08 Sumitomo Pharmaceuticals Co., Ltd. Pharmaceutical compositions for inhibiting the formation of tumor necrosis factor
JPH11209350A (ja) 1998-01-26 1999-08-03 Eisai Co Ltd 含窒素複素環誘導体およびその医薬
MXPA05011523A (es) * 2003-04-30 2006-01-23 Inst For Pharm Discovery Inc Heteroarilos sustituidos como inhibidores de proteinas de tirosina fosfatasas.
BRPI0415683A (pt) * 2003-11-03 2006-12-19 Warner Lambert Co inibidores da reabsorção de norepinefrina para o tratamento de distúrbios do sistema nervoso central
CA2612460A1 (en) 2005-06-27 2007-01-04 F. Hoffmann-La Roche Ag Chloro-substituted guanidines
US7855194B2 (en) 2006-03-27 2010-12-21 Hoffmann-La Roche Inc. Pyrimidine, quinazoline, pteridine and triazine derivatives
ES2532277T3 (es) 2006-11-22 2015-03-25 Sumitomo Chemical Company, Limited Derivados de quinazolina capaces de inhibir la señalización de citoquinina

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA894239A (en) * 1972-02-29 Pfizer Inc. Nitrogen heterocycles
US3305553A (en) * 1965-10-18 1967-02-21 Parke Davis & Co 2-aminoquinazoline derivatives
US3509141A (en) * 1966-09-15 1970-04-28 Ciba Geigy Corp 2-amino-quinazolines
GB1347493A (en) * 1971-02-11 1974-02-27 Aspro Nicholas Ltd Benzazine derivatives
JPS5398997A (en) * 1977-02-09 1978-08-29 Sumitomo Chem Co Ltd Fused pyridine derivertives and process for their preparation

Also Published As

Publication number Publication date
HU187579B (en) 1986-01-28
NO164167C (no) 1990-09-05
DK156063C (da) 1989-11-13
IL66960A0 (en) 1983-02-23
NO164167B (no) 1990-05-28
NZ202237A (en) 1985-08-30
CS229692B2 (en) 1984-06-18
PT75667B (fr) 1985-01-11
ZA827516B (en) 1983-08-31
CA1236102A (en) 1988-05-03
IE53653B1 (en) 1989-01-04
AU8962882A (en) 1983-04-28
DD210040A5 (de) 1984-05-30
EP0079810A1 (fr) 1983-05-25
EP0079810B1 (fr) 1986-01-22
GR76535B (es) 1984-08-10
FR2514765A1 (fr) 1983-04-22
JPS5888369A (ja) 1983-05-26
SU1299511A3 (ru) 1987-03-23
KR880001077B1 (ko) 1988-06-22
YU223382A (en) 1984-10-31
US4499092A (en) 1985-02-12
DK465182A (da) 1983-04-22
DK156063B (da) 1989-06-19
KR840001968A (ko) 1984-06-07
FR2514765B1 (es) 1984-04-06
IE822447L (en) 1983-04-21
NO823491L (no) 1983-04-22
DE3268699D1 (en) 1986-03-06
FI73982C (fi) 1987-12-10
AU551938B2 (en) 1986-05-15
ATE17576T1 (de) 1986-02-15
ES8307226A1 (es) 1983-07-01
FI823580L (fi) 1983-04-22
FI73982B (fi) 1987-08-31
YU43528B (en) 1989-08-31
FI823580A0 (fi) 1982-10-20
PT75667A (fr) 1982-11-01

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19970203