DD144545A5 - Verfahren zur herstellung von neuen tetrahydropyridin-und piperidinderivaten - Google Patents

Verfahren zur herstellung von neuen tetrahydropyridin-und piperidinderivaten Download PDF

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Publication number
DD144545A5
DD144545A5 DD79213724A DD21372479A DD144545A5 DD 144545 A5 DD144545 A5 DD 144545A5 DD 79213724 A DD79213724 A DD 79213724A DD 21372479 A DD21372479 A DD 21372479A DD 144545 A5 DD144545 A5 DD 144545A5
Authority
DD
German Democratic Republic
Prior art keywords
hydrogen
general formula
radical
further substituted
ring
Prior art date
Application number
DD79213724A
Other languages
German (de)
English (en)
Inventor
Romeo Paioni
Walter Schilling
Raymond Bernasconi
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of DD144545A5 publication Critical patent/DD144545A5/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/86—Benzo [b] furans; Hydrogenated benzo [b] furans with an oxygen atom directly attached in position 7
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/91—Dibenzofurans; Hydrogenated dibenzofurans

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DD79213724A 1978-06-22 1979-06-19 Verfahren zur herstellung von neuen tetrahydropyridin-und piperidinderivaten DD144545A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH682378 1978-06-22

Publications (1)

Publication Number Publication Date
DD144545A5 true DD144545A5 (de) 1980-10-22

Family

ID=4315581

Family Applications (1)

Application Number Title Priority Date Filing Date
DD79213724A DD144545A5 (de) 1978-06-22 1979-06-19 Verfahren zur herstellung von neuen tetrahydropyridin-und piperidinderivaten

Country Status (10)

Country Link
US (1) US4259338A (ja)
EP (1) EP0006524A1 (ja)
JP (1) JPS552697A (ja)
AU (1) AU523656B2 (ja)
CA (1) CA1119601A (ja)
DD (1) DD144545A5 (ja)
DK (1) DK259879A (ja)
ES (3) ES481714A1 (ja)
NZ (1) NZ190784A (ja)
ZA (1) ZA793091B (ja)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4495357A (en) * 1981-07-01 1985-01-22 The Upjohn Company Pyridyl-substituted-benzofurans
US4490531A (en) * 1981-07-01 1984-12-25 The Upjohn Company Pyridyl-substituted-benzofurans
US4455427A (en) * 1981-07-01 1984-06-19 The Upjohn Company Pyridyl-substituted-benzofurans
US4447620A (en) * 1982-06-08 1984-05-08 The Upjohn Company Imidazolyl-substituted benzothiophenes
US4452986A (en) * 1982-06-08 1984-06-05 The Upjohn Company Imidazolyl-substituted benzofurans
GB2128993B (en) * 1982-10-08 1986-01-15 Ciba Geigy Ag Benzofurans
US4611059A (en) * 1982-10-12 1986-09-09 The Upjohn Company Pyridyl-substituted benzothiophenes
US4855435A (en) * 1982-10-12 1989-08-08 The Upjohn Company Pyridyl-substituted benzothiophenes
EP0398413A1 (en) * 1989-05-16 1990-11-22 Duphar International Research B.V "3,4-dehydropiperidine derivatives having psychotropic activity
US5296497A (en) * 1989-05-16 1994-03-22 Duphar International Research B.V. 3,4-dehydropiperidine derivatives having psychotropic activity
EP0404721A3 (de) * 1989-06-20 1991-12-27 Ciba-Geigy Ag Mikrobizide Mittel
DE4017211A1 (de) * 1990-05-29 1991-12-05 Merck Patent Gmbh Oxazolidinone
TW222631B (ja) * 1991-07-15 1994-04-21 Duphar Int Res
ATE180780T1 (de) * 1993-08-05 1999-06-15 Hoechst Marion Roussel Inc 2-(piperidin-4-yl, pyridin-4-yl und tetrahydropyridin-4-yl)-benzofuran-7-carbamat derivate, ihre herstellung und verwendung als acetylcholinesterase inhibitoren
JPH07320652A (ja) * 1994-05-27 1995-12-08 Toshiba Corp カラー受像管及びシャドウマスクの製造方法
EP0891358A1 (fr) * 1995-10-11 1999-01-20 Synthelabo Composes derives d'oxazolidin-2-one, leur procede de preparation et leur application en therapeutique
FR2751653B1 (fr) * 1996-07-25 1998-09-04 Synthelabo Derives de 3-benzofuranyloxazolidin-2-one, leur procede de preparation et leur application en therapeutique
FR2739856B1 (fr) * 1995-10-11 1997-11-14 Synthelabo Derives de 3-benzofuranyloxazolidin-2-one, leur procede de preparation et leur application en therapeutique
FR2741071B1 (fr) * 1995-11-09 1997-12-12 Synthelabo Derives de 3-(benzofuran-5-yl)oxazolidin-2-one, leur preparation et leur application en therapeutique
FR2741072B1 (fr) * 1995-11-09 1997-12-12 Synthelabo Derives d'oxazolidin-2-one, leur preparation et leur application en therapeutique
US6436964B1 (en) 1998-06-30 2002-08-20 Eli Lilly And Company Piperidine derivatives having effects on serotonin related systems
EP1204658B1 (en) * 1999-07-29 2003-05-07 Eli Lilly And Company Benzofurylpiperazine serotonin agonists
US6881733B1 (en) 1999-07-29 2005-04-19 Eli Lilly And Company Serotonergic benzofurans
MXPA02000914A (es) * 1999-07-29 2002-07-30 Lilly Co Eli Benzofuranos serotonergicos.
ES2203498T3 (es) 1999-07-29 2004-04-16 Eli Lilly And Company Benzofurilpiperazinas: agonistas de receptor 5-ht2c de la serotonina.
JP2005008631A (ja) * 2003-05-29 2005-01-13 New Industry Research Organization ベンゾフラン化合物、およびそれを含有してなる医薬組成物
WO2004106317A1 (ja) * 2003-05-29 2004-12-09 The New Industry Research Organization ベンゾフラン化合物、およびそれを含有してなる医薬組成物
EP2110374A1 (en) * 2008-04-18 2009-10-21 Merck Sante Benzofurane, benzothiophene, benzothiazol derivatives as FXR modulators
CN101810606A (zh) * 2010-03-12 2010-08-25 南方医科大学 2-(6-羟基-2′,3′-二甲氧基苯基)-6-羟基-7-甲氧基苯骈呋喃在制备单胺氧化酶抑制剂中的应用
CN102381961B (zh) * 2011-09-03 2014-01-15 四川大学 3-苯基戊二酸类化合物、其制备方法和用途
CN118460017B (zh) * 2024-05-11 2024-11-05 广州豫顺新材料科技有限公司 一种覆铜板用改性球形硅微粉及其制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2633468A (en) * 1951-07-26 1953-03-31 Lilly Co Eli Benzooxaheterocyclic bases and acid addition salts thereof
GB1041525A (en) * 1964-11-11 1966-09-07 Belge Produits Chimiques Sa Benzofuran derivatives and processes for preparing the same
US3751390A (en) * 1971-05-19 1973-08-07 Aldrich Chem Co Inc Substituted dibenzofuran
BE794630A (fr) * 1972-01-26 1973-07-26 Beecham Group Ltd Composes polycycliques antihypertenseurs
CH592656A5 (ja) * 1973-03-02 1977-10-31 Ciba Geigy Ag
IE39264B1 (en) * 1973-05-25 1978-08-30 Ciba Geigy Ag New pharmaceutical preparations
CH609054A5 (en) * 1975-11-26 1979-02-15 Ciba Geigy Ag Process for the preparation of a novel piperidine derivative
CH605925A5 (ja) * 1974-08-30 1978-10-13 Ciba Geigy Ag
LU76756A1 (ja) * 1977-02-11 1978-10-18

Also Published As

Publication number Publication date
CA1119601A (en) 1982-03-09
ES489627A0 (es) 1981-04-01
AU4825779A (en) 1980-01-03
ES481714A1 (es) 1980-06-16
US4259338A (en) 1981-03-31
DK259879A (da) 1979-12-23
EP0006524A1 (de) 1980-01-09
JPS552697A (en) 1980-01-10
ZA793091B (en) 1980-06-25
ES8104281A1 (es) 1981-04-01
AU523656B2 (en) 1982-08-05
NZ190784A (en) 1982-03-16
ES8104280A1 (es) 1981-04-01
ES489628A0 (es) 1981-04-01

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