ES489628A0 - Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina - Google Patents

Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina

Info

Publication number
ES489628A0
ES489628A0 ES489628A ES489628A ES489628A0 ES 489628 A0 ES489628 A0 ES 489628A0 ES 489628 A ES489628 A ES 489628A ES 489628 A ES489628 A ES 489628A ES 489628 A0 ES489628 A0 ES 489628A0
Authority
ES
Spain
Prior art keywords
piperidina
piridina
tetrahidro
derivatives
procedure
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES489628A
Other languages
English (en)
Other versions
ES8104281A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of ES8104281A1 publication Critical patent/ES8104281A1/es
Publication of ES489628A0 publication Critical patent/ES489628A0/es
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/86Benzo [b] furans; Hydrogenated benzo [b] furans with an oxygen atom directly attached in position 7
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/91Dibenzofurans; Hydrogenated dibenzofurans
ES489628A 1978-06-22 1980-03-17 Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina Granted ES489628A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH682378 1978-06-22

Publications (2)

Publication Number Publication Date
ES8104281A1 ES8104281A1 (es) 1981-04-01
ES489628A0 true ES489628A0 (es) 1981-04-01

Family

ID=4315581

Family Applications (3)

Application Number Title Priority Date Filing Date
ES481714A Expired ES481714A1 (es) 1978-06-22 1979-06-20 Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina.
ES489628A Granted ES489628A0 (es) 1978-06-22 1980-03-17 Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina
ES489627A Granted ES489627A0 (es) 1978-06-22 1980-03-17 Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES481714A Expired ES481714A1 (es) 1978-06-22 1979-06-20 Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina.

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES489627A Granted ES489627A0 (es) 1978-06-22 1980-03-17 Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina

Country Status (10)

Country Link
US (1) US4259338A (es)
EP (1) EP0006524A1 (es)
JP (1) JPS552697A (es)
AU (1) AU523656B2 (es)
CA (1) CA1119601A (es)
DD (1) DD144545A5 (es)
DK (1) DK259879A (es)
ES (3) ES481714A1 (es)
NZ (1) NZ190784A (es)
ZA (1) ZA793091B (es)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4490531A (en) * 1981-07-01 1984-12-25 The Upjohn Company Pyridyl-substituted-benzofurans
US4495357A (en) * 1981-07-01 1985-01-22 The Upjohn Company Pyridyl-substituted-benzofurans
US4455427A (en) * 1981-07-01 1984-06-19 The Upjohn Company Pyridyl-substituted-benzofurans
US4452986A (en) * 1982-06-08 1984-06-05 The Upjohn Company Imidazolyl-substituted benzofurans
US4447620A (en) * 1982-06-08 1984-05-08 The Upjohn Company Imidazolyl-substituted benzothiophenes
GB2128993B (en) * 1982-10-08 1986-01-15 Ciba Geigy Ag Benzofurans
US4611059A (en) * 1982-10-12 1986-09-09 The Upjohn Company Pyridyl-substituted benzothiophenes
US4855435A (en) * 1982-10-12 1989-08-08 The Upjohn Company Pyridyl-substituted benzothiophenes
EP0398413A1 (en) * 1989-05-16 1990-11-22 Duphar International Research B.V "3,4-dehydropiperidine derivatives having psychotropic activity
US5296497A (en) * 1989-05-16 1994-03-22 Duphar International Research B.V. 3,4-dehydropiperidine derivatives having psychotropic activity
US5068359A (en) * 1989-06-20 1991-11-26 Ciba-Geigy Corporation Microbicidal compositions
DE4017211A1 (de) * 1990-05-29 1991-12-05 Merck Patent Gmbh Oxazolidinone
TW222631B (es) * 1991-07-15 1994-04-21 Duphar Int Res
EP0637586B1 (en) * 1993-08-05 1999-06-02 HOECHST MARION ROUSSEL, Inc. 2-(Piperidin-4-yl, pyridin-4-yl and tetrahydropyridin-4-yl)-benzofuran-7-carbamate derivatives, their preparation and their use as acetylcholinesterase inhibitors
JPH07320652A (ja) * 1994-05-27 1995-12-08 Toshiba Corp カラー受像管及びシャドウマスクの製造方法
FR2739856B1 (fr) * 1995-10-11 1997-11-14 Synthelabo Derives de 3-benzofuranyloxazolidin-2-one, leur procede de preparation et leur application en therapeutique
AU7135996A (en) * 1995-10-11 1997-04-30 Synthelabo Oxazolidin-2-one derivatives, preparation method therefor and therapeutical use thereof
FR2751653B1 (fr) * 1996-07-25 1998-09-04 Synthelabo Derives de 3-benzofuranyloxazolidin-2-one, leur procede de preparation et leur application en therapeutique
FR2741071B1 (fr) * 1995-11-09 1997-12-12 Synthelabo Derives de 3-(benzofuran-5-yl)oxazolidin-2-one, leur preparation et leur application en therapeutique
FR2741072B1 (fr) * 1995-11-09 1997-12-12 Synthelabo Derives d'oxazolidin-2-one, leur preparation et leur application en therapeutique
AU4726699A (en) * 1998-06-30 2000-01-17 Eli Lilly And Company Piperidine derivatives having effects on serotonin related systems
US6881733B1 (en) 1999-07-29 2005-04-19 Eli Lilly And Company Serotonergic benzofurans
DE60002583T2 (de) * 1999-07-29 2004-03-25 Eli Lilly And Co., Indianapolis Benzofurylpiperazine als serotonin-agonisten
ES2209951T3 (es) * 1999-07-29 2004-07-01 Eli Lilly And Company Benzofuranos serotoninergicos.
JP2003506365A (ja) 1999-07-29 2003-02-18 イーライ・リリー・アンド・カンパニー ベンゾフリルピペラジンおよびベンゾフリルホモピペラジン:セロトニンアゴニスト
JP2005008631A (ja) * 2003-05-29 2005-01-13 New Industry Research Organization ベンゾフラン化合物、およびそれを含有してなる医薬組成物
US7638540B2 (en) 2003-05-29 2009-12-29 The New Industry Research Organization Benzofuran compound and medicinal composition containing the same
EP2110374A1 (en) * 2008-04-18 2009-10-21 Merck Sante Benzofurane, benzothiophene, benzothiazol derivatives as FXR modulators
CN101810606A (zh) * 2010-03-12 2010-08-25 南方医科大学 2-(6-羟基-2′,3′-二甲氧基苯基)-6-羟基-7-甲氧基苯骈呋喃在制备单胺氧化酶抑制剂中的应用
CN102381961B (zh) * 2011-09-03 2014-01-15 四川大学 3-苯基戊二酸类化合物、其制备方法和用途

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2633468A (en) * 1951-07-26 1953-03-31 Lilly Co Eli Benzooxaheterocyclic bases and acid addition salts thereof
GB1041525A (en) * 1964-11-11 1966-09-07 Belge Produits Chimiques Sa Benzofuran derivatives and processes for preparing the same
US3751390A (en) * 1971-05-19 1973-08-07 Aldrich Chem Co Inc Substituted dibenzofuran
BE794630A (fr) * 1972-01-26 1973-07-26 Beecham Group Ltd Composes polycycliques antihypertenseurs
CH592656A5 (es) * 1973-03-02 1977-10-31 Ciba Geigy Ag
IE39264B1 (en) * 1973-05-25 1978-08-30 Ciba Geigy Ag New pharmaceutical preparations
CH609054A5 (en) * 1975-11-26 1979-02-15 Ciba Geigy Ag Process for the preparation of a novel piperidine derivative
CH605925A5 (es) * 1974-08-30 1978-10-13 Ciba Geigy Ag
LU76756A1 (es) * 1977-02-11 1978-10-18

Also Published As

Publication number Publication date
JPS552697A (en) 1980-01-10
DD144545A5 (de) 1980-10-22
DK259879A (da) 1979-12-23
AU4825779A (en) 1980-01-03
CA1119601A (en) 1982-03-09
ZA793091B (en) 1980-06-25
ES8104280A1 (es) 1981-04-01
ES8104281A1 (es) 1981-04-01
AU523656B2 (en) 1982-08-05
EP0006524A1 (de) 1980-01-09
NZ190784A (en) 1982-03-16
US4259338A (en) 1981-03-31
ES489627A0 (es) 1981-04-01
ES481714A1 (es) 1980-06-16

Similar Documents

Publication Publication Date Title
ES489628A0 (es) Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina
AR220704A1 (es) Procedimiento para la preparacion de derivados de indanil y tetrahidronaftil octatrieno
MX6749E (es) Procedimiento para la preparacion de derivados de tetrazolilalcoxicarboestirilo
ES494634A0 (es) Procedimiento para la preparacion de compuestos de cefem y cefam
MX5631E (es) Procedimiento para la preparacion de acil-anilinas
MX5793E (es) Procedimiento para la preparacion de 4-amino-5-alquilsulfonil-orto-anisamidas
MX5676E (es) Procedimiento mejorado para la preparacion de cicloalcanoles y cicloalcanonas
ES482499A0 (es) Procedimiento para la preparacion de 2-cloro-6-nitroanilinas
AR221355A1 (es) Procedimiento para la preparacion de derivados de pirrolidinil y pirrolidinilmetil-benzamidas
AR227379A1 (es) Procedimiento para la preparacion de 1-aril-2-imidazolil vinileteres
MX5509E (es) Procedimiento para la preparacion de n-halogenoacetil-fenilaminocarboniloximas
MX5898E (es) Procedimiento para la preparacion de 2-amino-4-pirimidonas
AR224784A1 (es) Procedimiento para la preparacion de nuevos derivados de 4-amino-2-piperidinoquinazolina
MX5594E (es) Procedimiento mejorado para la preparacion de derivados de n-trifluoroacetil-n-fosfonometilglicinatos
ES485567A0 (es) Procedimiento para la preparacion de azolilcetales
MX5826E (es) Procedimiento para la obtencion de derivados de fenilimino metil-piridina
MX5672E (es) Procedimiento para la preparacion de acidos 2-piridil y 2-pirimidil-aminobenzoicos
MX5738E (es) Procedimiento para la obtencion de compuestos de iminoeter de benzotiazolina y benzoxazolina-n-substituidos
MX149694A (es) Procedimiento para la preparacion de trialcoxisilanos de fenoxialquilo
ES484342A0 (es) Procedimiento para la preparacion de propenilensulfona
ES480637A0 (es) Procedimiento para la obtencion de nuevos derivados de la piperacina metanimina
MX5955E (es) Procedimiento para la preparacion de derivados de piridoxina
AR227629A1 (es) Procedimiento para la preparacion esteroespecifica o esteroselectiva de derivados de imidazolil-oxi-meteres y derivados de imidazoliloximas
MX5674E (es) Procedimiento para la preparacion de derivados de la butenofenona
MX5445E (es) Procedimiento para la preparacion de derivados de isotiocianobenzotiazol