CZ302461B6 - Cyklický hexapeptid, zpusob jeho výroby, farmaceutický prípravek tento cyklický hexapeptid obsahující a použití tohoto cyklického hexapeptidu pro výrobu léciva - Google Patents
Cyklický hexapeptid, zpusob jeho výroby, farmaceutický prípravek tento cyklický hexapeptid obsahující a použití tohoto cyklického hexapeptidu pro výrobu léciva Download PDFInfo
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- CZ302461B6 CZ302461B6 CZ20030288A CZ2003288A CZ302461B6 CZ 302461 B6 CZ302461 B6 CZ 302461B6 CZ 20030288 A CZ20030288 A CZ 20030288A CZ 2003288 A CZ2003288 A CZ 2003288A CZ 302461 B6 CZ302461 B6 CZ 302461B6
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Classifications
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- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
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Landscapes
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- Organic Chemistry (AREA)
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| Application Number | Priority Date | Filing Date | Title |
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| GBGB0018891.2A GB0018891D0 (en) | 2000-08-01 | 2000-08-01 | Organic compounds |
Publications (2)
| Publication Number | Publication Date |
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| CZ2003288A3 CZ2003288A3 (cs) | 2003-05-14 |
| CZ302461B6 true CZ302461B6 (cs) | 2011-06-01 |
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| Application Number | Title | Priority Date | Filing Date |
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| CZ20030288A CZ302461B6 (cs) | 2000-08-01 | 2001-07-30 | Cyklický hexapeptid, zpusob jeho výroby, farmaceutický prípravek tento cyklický hexapeptid obsahující a použití tohoto cyklického hexapeptidu pro výrobu léciva |
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| US7189856B2 (en) | 2001-12-28 | 2007-03-13 | Gideon Shapiro | Non-peptide somatostatin receptor ligands |
| ATE461173T1 (de) * | 2002-12-12 | 2010-04-15 | Novartis Pharma Gmbh | Prozess für die herstellung von peptiden, die eine 4-hydorxy-prolin substruktur enthalten |
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| US7697338B2 (en) * | 2006-11-16 | 2010-04-13 | Sandisk Corporation | Systems for controlled boosting in non-volatile memory soft programming |
| CN101553728B (zh) * | 2006-11-28 | 2013-02-06 | 香港大学 | 颗粒体蛋白-上皮素前体(gep)抗体用于检测和抑制肝细胞癌(hcc)的用途 |
| EP1941902A1 (en) * | 2007-01-02 | 2008-07-09 | Novartis AG | Use of Somatostatin analogs in cluster headache |
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| US8592377B2 (en) | 2007-03-28 | 2013-11-26 | President And Fellows Of Harvard College | Stitched polypeptides |
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| EP2067786A1 (en) | 2007-12-07 | 2009-06-10 | ITALFARMACO S.p.A. | Novel non selective analogs of somatostatin |
| US8937152B2 (en) * | 2007-12-03 | 2015-01-20 | Italfarmaco Spa | Non-selective somatostatin analogues |
| US20090325863A1 (en) * | 2008-06-13 | 2009-12-31 | Kleinberg David L | Somatostatin analogs and IGF-I inhibition for breast cancer prevention |
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| EP2172189A1 (en) | 2008-10-01 | 2010-04-07 | Novartis AG | Pharmaceutical Compositions |
| EP2213307A1 (en) | 2009-02-03 | 2010-08-04 | Novartis AG | Injectable depot formulations |
| KR101814186B1 (ko) | 2008-09-17 | 2018-03-14 | 키아스마 인코포레이티드 | 약제학적 조성물 및 연관된 투여방법 |
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| ES2711526T3 (es) | 2010-08-13 | 2019-05-06 | Aileron Therapeutics Inc | Macrociclos peptidomiméticos |
| US8629103B2 (en) | 2010-12-02 | 2014-01-14 | New York University | Treatment of non-proliferative cystic disease of the breast |
| EP2651917A1 (en) | 2010-12-13 | 2013-10-23 | Novartis AG | Dimeric iap inhibitors |
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| US20130035054A1 (en) * | 2011-07-14 | 2013-02-07 | Faceon Mobile | Phone with multi-portal access for display during incoming and outgoing call |
| WO2013019923A2 (en) | 2011-08-02 | 2013-02-07 | New York University | Methods for detecting progenitor cells and uses thereof |
| BR112014007310A2 (pt) | 2011-09-27 | 2017-04-04 | Novartis Ag | 3-pirimidin-4-il-oxazolidin-2-onas como inibidores de idh mutante |
| TW201806968A (zh) | 2011-10-18 | 2018-03-01 | 艾利倫治療公司 | 擬肽巨環化合物 |
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| MX350929B (es) | 2011-12-05 | 2017-09-26 | Camurus Ab | Formulaciones peptidicas robustas de liberación controlada. |
| EP2802658A2 (en) | 2012-01-09 | 2014-11-19 | Novartis AG | Rnai agents to treat beta-catenin related diseases |
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| EP2819688A4 (en) | 2012-02-15 | 2015-10-28 | Aileron Therapeutics Inc | TRIAZOL AND THIOETHER-COUPLED PEPTIDOMIMETIC MACROCYCLES |
| BR112014020103A2 (pt) | 2012-02-15 | 2018-10-09 | Aileron Therapeutics, Inc. | macrociclos peptidomiméticos |
| BR112014029425A2 (pt) * | 2012-05-25 | 2017-06-27 | Camurus Ab | pré-formulação, dispositivo de administração pré-cheio, kit, processo para a formação de uma pré-formulação, usos de mistura e de um solvente polar, e, método para o tratamento de um sujeito |
| TWI704919B (zh) | 2012-05-31 | 2020-09-21 | 日商大塚製藥股份有限公司 | 用於預防及/或治療多囊性腎臟病之藥物 |
| WO2014071241A1 (en) | 2012-11-01 | 2014-05-08 | Aileron Therapeutics, Inc. | Disubstituted amino acids and methods of preparation and use thereof |
| US9480759B2 (en) | 2012-11-21 | 2016-11-01 | Serene, Llc | Tin-117m somatostatin receptor binding compounds and methods |
| ES2671516T3 (es) | 2013-02-19 | 2018-06-06 | Novartis Ag | Derivados de benzotiofeno y composiciones de los mismos como degradantes selectivos de los receptores de estrógeno |
| AU2014229283B2 (en) | 2013-03-14 | 2016-07-28 | Novartis Ag | 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant IDH |
| JP6387360B2 (ja) | 2013-03-14 | 2018-09-05 | ノバルティス アーゲー | 変異ｉｄｈの阻害薬としての３−ピリミジン−４−イル−オキサゾリジン−２−オン |
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- 2001-07-30 AU AU8977801A patent/AU8977801A/xx active Pending
- 2001-07-30 IL IL15392001A patent/IL153920A0/xx unknown
- 2001-07-30 SK SK121-2003A patent/SK287798B6/sk not_active IP Right Cessation
- 2001-07-30 DE DE60133823T patent/DE60133823T2/de not_active Expired - Lifetime
- 2001-07-30 CZ CZ20030288A patent/CZ302461B6/cs unknown
- 2001-07-30 NZ NZ523836A patent/NZ523836A/en not_active IP Right Cessation
- 2001-07-30 US US10/343,288 patent/US7473761B2/en active Active
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2003
- 2003-01-13 IL IL153920A patent/IL153920A/en active Protection Beyond IP Right Term
- 2003-01-15 ZA ZA200300406A patent/ZA200300406B/xx unknown
- 2003-01-29 EC EC2003004456A patent/ECSP034456A/es unknown
- 2003-01-30 NO NO20030484A patent/NO331093B1/no not_active IP Right Cessation
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2008
- 2008-07-29 CY CY20081100789T patent/CY1108547T1/el unknown
- 2008-11-05 US US12/265,135 patent/US7939625B2/en not_active Expired - Fee Related
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2011
- 2011-03-16 US US13/048,932 patent/US8822637B2/en not_active Expired - Lifetime
- 2011-03-16 US US13/048,935 patent/US9035021B2/en not_active Expired - Lifetime
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2012
- 2012-06-20 LU LU92024C patent/LU92024I2/fr unknown
- 2012-06-21 BE BE2012C026C patent/BE2012C026I2/fr unknown
- 2012-06-26 FR FR12C0041C patent/FR12C0041I2/fr active Active
- 2012-06-29 CY CY2012018C patent/CY2012018I1/el unknown
- 2012-06-29 NO NO2012012C patent/NO2012012I2/no not_active IP Right Cessation
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2015
- 2015-04-08 US US14/681,226 patent/US20150218223A1/en not_active Abandoned
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1997001579A2 (en) * | 1995-06-29 | 1997-01-16 | Novartis Ag | Somatostatin peptides |
| EP1307486A2 (en) * | 2000-08-01 | 2003-05-07 | Novartis AG | Somatostatin analogues |
Non-Patent Citations (1)
| Title |
|---|
| Huang a kol. (1992) J. Am. Chem. Soc. 114 (24), 9390-9401 * |
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