CZ286789B6 - Pyridazine derivative, process of its preparation, use and pharmaceutical preparation based thereon - Google Patents

Pyridazine derivative, process of its preparation, use and pharmaceutical preparation based thereon Download PDF

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Publication number
CZ286789B6
CZ286789B6 CZ19981380A CZ138098A CZ286789B6 CZ 286789 B6 CZ286789 B6 CZ 286789B6 CZ 19981380 A CZ19981380 A CZ 19981380A CZ 138098 A CZ138098 A CZ 138098A CZ 286789 B6 CZ286789 B6 CZ 286789B6
Authority
CZ
Czechia
Prior art keywords
diazo
formula
pyridazine
hexahydro
hexahydrophenanthrene
Prior art date
Application number
CZ19981380A
Other languages
Czech (cs)
English (en)
Other versions
CZ138098A3 (cs
Inventor
Donald W Combs
Original Assignee
Ortho Mcneil Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ortho Mcneil Pharm Inc filed Critical Ortho Mcneil Pharm Inc
Publication of CZ138098A3 publication Critical patent/CZ138098A3/cs
Publication of CZ286789B6 publication Critical patent/CZ286789B6/cs

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50Pyridazines; Hydrogenated pyridazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/06Antiabortive agents; Labour repressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/26Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/26Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
    • C07D237/36Benzo-cinnolines

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Gynecology & Obstetrics (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Pregnancy & Childbirth (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CZ19981380A 1995-11-06 1996-10-10 Pyridazine derivative, process of its preparation, use and pharmaceutical preparation based thereon CZ286789B6 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US790095P 1995-11-06 1995-11-06

Publications (2)

Publication Number Publication Date
CZ138098A3 CZ138098A3 (cs) 1998-09-16
CZ286789B6 true CZ286789B6 (en) 2000-07-12

Family

ID=21728709

Family Applications (1)

Application Number Title Priority Date Filing Date
CZ19981380A CZ286789B6 (en) 1995-11-06 1996-10-10 Pyridazine derivative, process of its preparation, use and pharmaceutical preparation based thereon

Country Status (17)

Country Link
JP (1) JP2000501073A (no)
KR (1) KR100360614B1 (no)
CN (1) CN1110485C (no)
AU (1) AU704507B2 (no)
BR (1) BR9611407A (no)
CZ (1) CZ286789B6 (no)
HU (1) HU225162B1 (no)
IL (1) IL124320A (no)
MX (1) MX9803605A (no)
NO (1) NO310460B1 (no)
NZ (1) NZ319979A (no)
PL (1) PL185618B1 (no)
RU (1) RU2175969C2 (no)
TW (1) TW460467B (no)
UA (1) UA48989C2 (no)
WO (1) WO1997017332A1 (no)
ZA (1) ZA969298B (no)

Also Published As

Publication number Publication date
AU704507B2 (en) 1999-04-22
BR9611407A (pt) 1999-12-28
CN1110485C (zh) 2003-06-04
KR100360614B1 (ko) 2003-06-02
CZ138098A3 (cs) 1998-09-16
PL326669A1 (en) 1998-10-12
CN1207091A (zh) 1999-02-03
TW460467B (en) 2001-10-21
HU225162B1 (en) 2006-07-28
PL185618B1 (pl) 2003-06-30
JP2000501073A (ja) 2000-02-02
AU7263796A (en) 1997-05-29
NO982030D0 (no) 1998-05-05
IL124320A (en) 2001-10-31
HUP0201305A2 (hu) 2002-12-28
MX9803605A (es) 1998-09-30
NO310460B1 (no) 2001-07-09
HUP0201305A3 (en) 2003-02-28
NO982030L (no) 1998-06-23
IL124320A0 (en) 1998-12-06
NZ319979A (en) 1999-11-29
UA48989C2 (uk) 2002-09-16
ZA969298B (en) 1998-05-05
WO1997017332A1 (en) 1997-05-15
KR19990067340A (ko) 1999-08-16
RU2175969C2 (ru) 2001-11-20

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Legal Events

Date Code Title Description
IF00 In force as of 2000-06-30 in czech republic
MM4A Patent lapsed due to non-payment of fee

Effective date: 20071010