CY1112324T1 - Φαρμακευτικες συνθεσεις αναστολεων της πρωτεϊνης μεταφορας εστερων χοληστερολης (cετρ) - Google Patents

Φαρμακευτικες συνθεσεις αναστολεων της πρωτεϊνης μεταφορας εστερων χοληστερολης (cετρ)

Info

Publication number
CY1112324T1
CY1112324T1 CY20121100126T CY121100126T CY1112324T1 CY 1112324 T1 CY1112324 T1 CY 1112324T1 CY 20121100126 T CY20121100126 T CY 20121100126T CY 121100126 T CY121100126 T CY 121100126T CY 1112324 T1 CY1112324 T1 CY 1112324T1
Authority
CY
Cyprus
Prior art keywords
pharmaceutical compositions
cetp
transfer composition
stock transfer
protein cholesterol
Prior art date
Application number
CY20121100126T
Other languages
English (en)
Inventor
Yoshifumi Uemoto
Original Assignee
Japan Tobacco, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33033290&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1112324(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Japan Tobacco, Inc. filed Critical Japan Tobacco, Inc.
Publication of CY1112324T1 publication Critical patent/CY1112324T1/el

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/70—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/82—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton with the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/095—Sulfur, selenium, or tellurium compounds, e.g. thiols
    • A61K31/10—Sulfides; Sulfoxides; Sulfones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/265—Esters, e.g. nitroglycerine, selenocyanates of carbonic, thiocarbonic, or thiocarboxylic acids, e.g. thioacetic acid, xanthogenic acid, trithiocarbonic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Steroid Compounds (AREA)

Abstract

Η εφεύρεση παρέχει φαρμακευτικές συνθέσεις που περιλαμβάνουν έναν αναστολέα της πρωτεΐνης μεταφοράς εστέρων της χοληστερόλης (CΕΤΡ) και ένα αδιάλυτο στο νερό πρόσθετο που αυξάνει τη συγκέντρωση, οι οποίες επιδεικνύουν βελτιωμένη βιοδιαθεσιμότητα. Η εφεύρεση προσφέρει επίσης μεθόδους για την αντιμετώπιση καρδιαγγειακών διαταραχών που περιλαμβάνουν τη χορήγηση των φαρμακευτικών συνθέσεων που περιλαμβάνουν έναν αναστολέα της CΕΤΡ.
CY20121100126T 2003-03-17 2012-02-06 Φαρμακευτικες συνθεσεις αναστολεων της πρωτεϊνης μεταφορας εστερων χοληστερολης (cετρ) CY1112324T1 (el)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US45529303P 2003-03-17 2003-03-17
US46052103P 2003-04-04 2003-04-04
US47720203P 2003-06-10 2003-06-10
US49364903P 2003-08-08 2003-08-08
EP04721345A EP1603553B9 (en) 2003-03-17 2004-03-17 Pharmaceutical compositions of cetp inhibitors

Publications (1)

Publication Number Publication Date
CY1112324T1 true CY1112324T1 (el) 2015-12-09

Family

ID=33033290

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20121100126T CY1112324T1 (el) 2003-03-17 2012-02-06 Φαρμακευτικες συνθεσεις αναστολεων της πρωτεϊνης μεταφορας εστερων χοληστερολης (cετρ)

Country Status (21)

Country Link
US (2) US20040225018A1 (el)
EP (2) EP2289507A1 (el)
JP (2) JP5546715B2 (el)
KR (2) KR20080008440A (el)
AT (1) ATE534381T1 (el)
AU (1) AU2004222434B2 (el)
BR (1) BRPI0408466B8 (el)
CA (1) CA2519432C (el)
CO (1) CO5640101A2 (el)
CY (1) CY1112324T1 (el)
DK (1) DK1603553T3 (el)
ES (1) ES2377121T3 (el)
HK (1) HK1084882A1 (el)
IL (1) IL170749A (el)
MX (1) MXPA05009848A (el)
NO (1) NO336891B1 (el)
NZ (1) NZ542852A (el)
PL (1) PL1603553T3 (el)
PT (1) PT1603553E (el)
SI (1) SI1603553T1 (el)
WO (1) WO2004082593A2 (el)

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JP6539661B2 (ja) 2013-12-19 2019-07-03 エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ 眼疾患の処置において使用するためのｃｅｔｐモデュレーター
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JP2006520808A (ja) 2006-09-14
WO2004082593A3 (en) 2005-02-24
KR100857759B1 (ko) 2008-09-09
CA2519432A1 (en) 2004-09-30
HK1084882A1 (en) 2006-08-11
NO20054740L (no) 2005-12-13
US20140243414A1 (en) 2014-08-28
JP2011052006A (ja) 2011-03-17
EP1603553A2 (en) 2005-12-14
JP5546715B2 (ja) 2014-07-09
AU2004222434B2 (en) 2010-06-03
ES2377121T3 (es) 2012-03-22
PL1603553T3 (pl) 2012-04-30
WO2004082593A2 (en) 2004-09-30
BRPI0408466B1 (pt) 2018-11-21
AU2004222434A1 (en) 2004-09-30
KR20080008440A (ko) 2008-01-23
SI1603553T1 (sl) 2012-03-30
EP1603553B9 (en) 2012-06-20
EP2289507A1 (en) 2011-03-02
NZ542852A (en) 2008-09-26
PT1603553E (pt) 2012-02-03
ATE534381T1 (de) 2011-12-15
IL170749A (en) 2012-08-30
KR20050110019A (ko) 2005-11-22
CO5640101A2 (es) 2006-05-31
BRPI0408466B8 (pt) 2021-05-25
BRPI0408466A (pt) 2006-04-04
ES2377121T9 (es) 2012-08-21
IL170749A0 (en) 2009-02-11
NO336891B1 (no) 2015-11-23
MXPA05009848A (es) 2005-12-06
CA2519432C (en) 2009-06-09
NO20054740D0 (no) 2005-10-14
US20040225018A1 (en) 2004-11-11
DK1603553T3 (da) 2012-01-30
EP1603553B1 (en) 2011-11-23

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