CU20110106A7 - Nuevos compuestos 578 - Google Patents

Nuevos compuestos 578

Info

Publication number
CU20110106A7
CU20110106A7 CU20110106A CU20110106A CU20110106A7 CU 20110106 A7 CU20110106 A7 CU 20110106A7 CU 20110106 A CU20110106 A CU 20110106A CU 20110106 A CU20110106 A CU 20110106A CU 20110106 A7 CU20110106 A7 CU 20110106A7
Authority
CU
Cuba
Prior art keywords
dementia
disease
alzheimer
taxatively
amyloid angiopathy
Prior art date
Application number
CU20110106A
Other languages
English (en)
Spanish (es)
Inventor
Sofia Karlstroem
Berg Stefan Von
Britt-Marie Swahn
Peter Soederman
Didier Rotticci
Laszlo Rakos
Johan Lindstroem
Karin Kolmodin
Joerg Holenz
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42170158&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CU20110106(A7) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of CU20110106A7 publication Critical patent/CU20110106A7/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CU20110106A 2008-11-14 2011-05-13 Nuevos compuestos 578 CU20110106A7 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US11463408P 2008-11-14 2008-11-14
US13976708P 2008-12-22 2008-12-22
US22165309P 2009-06-30 2009-06-30

Publications (1)

Publication Number Publication Date
CU20110106A7 true CU20110106A7 (es) 2012-01-31

Family

ID=42170158

Family Applications (1)

Application Number Title Priority Date Filing Date
CU20110106A CU20110106A7 (es) 2008-11-14 2011-05-13 Nuevos compuestos 578

Country Status (24)

Country Link
US (2) US8030500B2 (OSRAM)
EP (1) EP2367814A4 (OSRAM)
JP (1) JP2012508734A (OSRAM)
KR (1) KR20110091540A (OSRAM)
CN (1) CN102282140A (OSRAM)
AR (1) AR074341A1 (OSRAM)
AU (1) AU2009314664A1 (OSRAM)
BR (1) BRPI0921879A2 (OSRAM)
CA (1) CA2743938A1 (OSRAM)
CL (1) CL2011001098A1 (OSRAM)
CO (1) CO6362004A2 (OSRAM)
CR (1) CR20110255A (OSRAM)
CU (1) CU20110106A7 (OSRAM)
DO (1) DOP2011000138A (OSRAM)
EA (1) EA201190020A1 (OSRAM)
EC (1) ECSP11011051A (OSRAM)
IL (1) IL212590A0 (OSRAM)
MX (1) MX2011004918A (OSRAM)
NI (1) NI201100099A (OSRAM)
PE (1) PE20110875A1 (OSRAM)
TW (1) TW201020244A (OSRAM)
UY (1) UY32241A (OSRAM)
WO (1) WO2010056196A1 (OSRAM)
ZA (1) ZA201104396B (OSRAM)

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JP2016501827A (ja) 2012-10-24 2016-01-21 塩野義製薬株式会社 Ｂａｃｅ１阻害作用を有するジヒドロオキサジンまたはオキサゼピン誘導体
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Also Published As

Publication number Publication date
KR20110091540A (ko) 2011-08-11
AR074341A1 (es) 2011-01-12
CA2743938A1 (en) 2010-05-20
ECSP11011051A (es) 2011-06-30
CR20110255A (es) 2011-07-04
AU2009314664A1 (en) 2011-06-23
CO6362004A2 (es) 2012-01-20
BRPI0921879A2 (pt) 2018-10-16
PE20110875A1 (es) 2012-01-11
EA201190020A1 (ru) 2012-02-28
JP2012508734A (ja) 2012-04-12
CL2011001098A1 (es) 2012-02-24
MX2011004918A (es) 2011-05-30
WO2010056196A1 (en) 2010-05-20
US20100125082A1 (en) 2010-05-20
US20110319426A1 (en) 2011-12-29
EP2367814A4 (en) 2012-07-04
DOP2011000138A (es) 2011-06-30
TW201020244A (en) 2010-06-01
UY32241A (es) 2010-06-30
ZA201104396B (en) 2012-03-28
EP2367814A1 (en) 2011-09-28
US8030500B2 (en) 2011-10-04
CN102282140A (zh) 2011-12-14
NI201100099A (es) 2012-03-19
IL212590A0 (en) 2011-07-31

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