CS9692A3 - Process for preparing 3-fluoropyrimidine nucleosides - Google Patents

Process for preparing 3-fluoropyrimidine nucleosides Download PDF

Info

Publication number
CS9692A3
CS9692A3 CS9296A CS9692A CS9692A3 CS 9692 A3 CS9692 A3 CS 9692A3 CS 9296 A CS9296 A CS 9296A CS 9692 A CS9692 A CS 9692A CS 9692 A3 CS9692 A3 CS 9692A3
Authority
CS
Czechoslovakia
Prior art keywords
apos
methanesulfonyl
compound
deoxy
nucleoside
Prior art date
Application number
CS9296A
Other languages
Czech (cs)
English (en)
Inventor
Antuono Joseph D Iii
Donald Carl Boop
Steven L Clauss
John Leo Considine Jr
Thurairajah Padmanathan
Carl J Rizzo
John Robert Andrade
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of CS9692A3 publication Critical patent/CS9692A3/cs

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06Pyrimidine radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CS9296A 1991-01-15 1992-01-14 Process for preparing 3-fluoropyrimidine nucleosides CS9692A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US64121391A 1991-01-15 1991-01-15

Publications (1)

Publication Number Publication Date
CS9692A3 true CS9692A3 (en) 1992-08-12

Family

ID=24571422

Family Applications (1)

Application Number Title Priority Date Filing Date
CS9296A CS9692A3 (en) 1991-01-15 1992-01-14 Process for preparing 3-fluoropyrimidine nucleosides

Country Status (16)

Country Link
EP (1) EP0495225A1 (ja)
JP (1) JPH07165785A (ja)
KR (1) KR920014825A (ja)
CN (1) CN1063287A (ja)
AU (1) AU647231B2 (ja)
CA (1) CA2059249A1 (ja)
CS (1) CS9692A3 (ja)
FI (1) FI920158A (ja)
HU (1) HUT60279A (ja)
IE (1) IE920106A1 (ja)
IL (1) IL100480A0 (ja)
NO (1) NO920180L (ja)
NZ (1) NZ241274A (ja)
PL (1) PL293172A1 (ja)
TW (1) TW199155B (ja)
ZA (1) ZA92274B (ja)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9309787D0 (en) * 1993-05-12 1993-06-23 Rhone Poulenc Chemicals Purification of fluoronucleosides
EP0698032B1 (en) * 1993-05-12 1998-07-29 Rhodia Limited Preparation of fluoro-nucleosides and intermediates for use therein
GB9309795D0 (en) * 1993-05-12 1993-06-23 Rhone Poulenc Chemicals Preparation of flouro-compounds
JP2002293792A (ja) * 1998-12-25 2002-10-09 Ajinomoto Co Inc ヌクレオシド又は糖のフッ素化誘導体の製造方法
CN116120262A (zh) * 2023-02-24 2023-05-16 宁德时代新能源科技股份有限公司 氟代环状醚的制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3775397A (en) * 1969-11-12 1973-11-27 Akad Wissenschaften Ddr Novel cytostatic 2',3'-dideoxy-3'-fluoropyrimidine-nucleosides
DD103241A1 (ja) * 1972-12-12 1974-01-12
DK0470355T3 (da) * 1990-08-06 1996-07-15 American Cyanamid Co Fremgangsmåde til fremstilling af deoxynucleosider

Also Published As

Publication number Publication date
CA2059249A1 (en) 1992-07-16
IL100480A0 (en) 1992-09-06
HUT60279A (en) 1992-08-28
PL293172A1 (en) 1993-04-05
EP0495225A1 (en) 1992-07-22
NO920180D0 (no) 1992-01-14
AU1023992A (en) 1992-07-23
ZA92274B (en) 1992-10-28
HU9200117D0 (en) 1992-04-28
AU647231B2 (en) 1994-03-17
NO920180L (no) 1992-07-16
FI920158A (fi) 1992-07-16
NZ241274A (en) 1994-04-27
JPH07165785A (ja) 1995-06-27
FI920158A0 (fi) 1992-01-14
KR920014825A (ko) 1992-08-25
TW199155B (ja) 1993-02-01
IE920106A1 (en) 1992-07-15
CN1063287A (zh) 1992-08-05

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