CS411291A3 - Pilocarpine derivatives, process of their preparation and a pharmaceutical comprising thereof - Google Patents

Pilocarpine derivatives, process of their preparation and a pharmaceutical comprising thereof Download PDF

Info

Publication number
CS411291A3
CS411291A3 CS914112A CS411291A CS411291A3 CS 411291 A3 CS411291 A3 CS 411291A3 CS 914112 A CS914112 A CS 914112A CS 411291 A CS411291 A CS 411291A CS 411291 A3 CS411291 A3 CS 411291A3
Authority
CS
Czechoslovakia
Prior art keywords
methyl
acid addition
compound
formula
imidazol
Prior art date
Application number
CS914112A
Other languages
Czech (cs)
English (en)
Inventor
Rene Amstutz
Georg Dr Bolliger
Gideon Dr Shapiro
Original Assignee
Sandoz Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ltd filed Critical Sandoz Ltd
Publication of CS411291A3 publication Critical patent/CS411291A3/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CS914112A 1987-01-31 1991-12-27 Pilocarpine derivatives, process of their preparation and a pharmaceutical comprising thereof CS411291A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3702940 1987-01-31

Publications (1)

Publication Number Publication Date
CS411291A3 true CS411291A3 (en) 1992-06-17

Family

ID=6319976

Family Applications (1)

Application Number Title Priority Date Filing Date
CS914112A CS411291A3 (en) 1987-01-31 1991-12-27 Pilocarpine derivatives, process of their preparation and a pharmaceutical comprising thereof

Country Status (27)

Country Link
US (1) US4835174A (da)
JP (1) JPS63201185A (da)
KR (1) KR880009013A (da)
AT (1) AT395852B (da)
AU (1) AU607966B2 (da)
BE (1) BE1001005A3 (da)
CA (1) CA1327805C (da)
CH (1) CH675721A5 (da)
CS (1) CS411291A3 (da)
DK (1) DK46288A (da)
ES (1) ES2008421A6 (da)
FI (1) FI90080C (da)
FR (1) FR2610322B1 (da)
GB (1) GB2200910B (da)
GR (1) GR880100042A (da)
HU (1) HU204047B (da)
IE (1) IE61989B1 (da)
IL (1) IL85252A (da)
IT (1) IT1219827B (da)
LU (1) LU87122A1 (da)
MY (1) MY102415A (da)
NL (1) NL8800099A (da)
NZ (1) NZ223359A (da)
PH (1) PH24837A (da)
PT (1) PT86666B (da)
SE (1) SE466150B (da)
ZA (1) ZA88665B (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4882343A (en) * 1987-08-28 1989-11-21 G. D. Searle & Co. Biarylalkylimidazole derivatives as anti-depressants
US5861431A (en) * 1995-06-07 1999-01-19 Iotek, Inc. Incontinence treatment
RU2761436C1 (ru) 2017-11-17 2021-12-08 Целликс Био Прайвет Лимитед Композиции и способы лечения нарушений со стороны органа зрения

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2457047A (en) * 1946-02-13 1948-12-21 Monsanto Chemicals 2-(2'-thenyl)-4, 5-dihydroimidazoles and process for making the same
GB1601310A (en) * 1978-05-23 1981-10-28 Lilly Industries Ltd Aryl hydantoins
JPS56131579A (en) * 1980-03-17 1981-10-15 Kissei Pharmaceut Co Ltd Novel 1-substituted imidazole derivative
JPS58150566A (ja) * 1982-03-03 1983-09-07 Yoshitomi Pharmaceut Ind Ltd 新規イミダゾ−ル誘導体
DE3228266A1 (de) * 1982-07-29 1984-02-02 A. Nattermann & Cie GmbH, 5000 Köln Imidazolylalkylthiophene, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
DE3329028A1 (de) * 1983-08-11 1985-02-28 Cassella Ag, 6000 Frankfurt Substituierte (2-amino-2-imidazolin-1-yl)-essigsaeurederivate, verfahren zu ihrer herstellung, ihre verwendung und sie enthaltende pharmazeutische zubereitungen

Also Published As

Publication number Publication date
IT1219827B (it) 1990-05-24
IT8847578A0 (it) 1988-01-29
LU87122A1 (fr) 1988-08-23
SE8800293L (sv) 1988-08-01
ATA18288A (de) 1992-08-15
AU607966B2 (en) 1991-03-21
NL8800099A (nl) 1988-08-16
HU204047B (en) 1991-11-28
MY102415A (en) 1992-06-17
PH24837A (en) 1990-10-30
SE8800293D0 (sv) 1988-01-29
FI90080B (fi) 1993-09-15
BE1001005A3 (fr) 1989-06-06
GB8801804D0 (en) 1988-02-24
NZ223359A (en) 1991-03-26
FI880430A0 (fi) 1988-01-29
GB2200910A (en) 1988-08-17
ES2008421A6 (es) 1989-07-16
FR2610322A1 (fr) 1988-08-05
GR880100042A (el) 1988-12-16
PT86666A (pt) 1988-02-01
DK46288D0 (da) 1988-01-29
PT86666B (pt) 1992-04-30
FI880430A (fi) 1988-08-01
US4835174A (en) 1989-05-30
IL85252A (en) 1992-03-29
IE880244L (en) 1988-07-31
IE61989B1 (en) 1994-12-14
FR2610322B1 (fr) 1990-02-16
CA1327805C (en) 1994-03-15
KR880009013A (ko) 1988-09-13
ZA88665B (en) 1989-09-27
JPS63201185A (ja) 1988-08-19
HUT50168A (en) 1989-12-28
IL85252A0 (en) 1988-07-31
AT395852B (de) 1993-03-25
SE466150B (sv) 1992-01-07
AU1096088A (en) 1988-08-04
FI90080C (fi) 1993-12-27
CH675721A5 (da) 1990-10-31
DK46288A (da) 1988-08-01
GB2200910B (en) 1991-01-16

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