CS266597B2 - Method of pregnale-21-acid's 16,17-acetal-substituted derivatives production - Google Patents

Method of pregnale-21-acid's 16,17-acetal-substituted derivatives production Download PDF

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Publication number
CS266597B2
CS266597B2 CS869604A CS960486A CS266597B2 CS 266597 B2 CS266597 B2 CS 266597B2 CS 869604 A CS869604 A CS 869604A CS 960486 A CS960486 A CS 960486A CS 266597 B2 CS266597 B2 CS 266597B2
Authority
CS
Czechoslovakia
Prior art keywords
alpha
formula
compound
acid
prepared
Prior art date
Application number
CS869604A
Other languages
Czech (cs)
English (en)
Other versions
CS960486A2 (en
Inventor
Paul H Andersson
Per T Andersson
Bengt I Axelsson
Ralph L Brattsand
Bror A Thalen
Jan W Trofast
Original Assignee
Draco Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Draco Ab filed Critical Draco Ab
Publication of CS960486A2 publication Critical patent/CS960486A2/cs
Publication of CS266597B2 publication Critical patent/CS266597B2/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/0026—Oxygen-containing hetero ring cyclic ketals
    • C07J71/0031—Oxygen-containing hetero ring cyclic ketals at positions 16, 17
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CS869604A 1985-12-19 1986-12-19 Method of pregnale-21-acid's 16,17-acetal-substituted derivatives production CS266597B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE8506015A SE8506015D0 (sv) 1985-12-19 1985-12-19 Novel 16,17-acetalsubstituted pregnane 21-oic acid derivatives

Publications (2)

Publication Number Publication Date
CS960486A2 CS960486A2 (en) 1989-04-14
CS266597B2 true CS266597B2 (en) 1990-01-12

Family

ID=20362521

Family Applications (1)

Application Number Title Priority Date Filing Date
CS869604A CS266597B2 (en) 1985-12-19 1986-12-19 Method of pregnale-21-acid's 16,17-acetal-substituted derivatives production

Country Status (31)

Country Link
EP (1) EP0232690B1 (zh)
JP (1) JPH0780900B2 (zh)
KR (1) KR940004067B1 (zh)
CN (1) CN1016508B (zh)
AR (1) AR242797A1 (zh)
AT (1) ATE57935T1 (zh)
AU (1) AU591950B2 (zh)
CA (1) CA1318664C (zh)
CS (1) CS266597B2 (zh)
DD (1) DD256703A5 (zh)
DE (1) DE3675378D1 (zh)
DK (1) DK168601B1 (zh)
ES (1) ES2018656B3 (zh)
FI (1) FI84488C (zh)
GR (1) GR3001052T3 (zh)
HU (1) HU196831B (zh)
IE (1) IE59241B1 (zh)
IL (1) IL80679A (zh)
IS (1) IS1559B (zh)
JO (1) JO1499B1 (zh)
LT (1) LT3912B (zh)
LV (1) LV10959B (zh)
MY (1) MY100750A (zh)
NO (1) NO164243C (zh)
NZ (1) NZ218614A (zh)
PH (1) PH23237A (zh)
PL (1) PL151627B1 (zh)
PT (1) PT83984B (zh)
RU (1) RU1839673C (zh)
SE (1) SE8506015D0 (zh)
ZA (1) ZA868750B (zh)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU203769B (en) * 1989-03-09 1991-09-30 Richter Gedeon Vegyeszet Process for producing new steroide derivatives and pharmaceutical compositions containing them
SE8903914D0 (sv) 1989-11-22 1989-11-22 Draco Ab Oral composition for the treatment of inflammatory bowel diseases
US5643602A (en) * 1989-11-22 1997-07-01 Astra Aktiebolag Oral composition for the treatment of inflammatory bowel disease
US6166024A (en) * 1995-03-30 2000-12-26 Mayo Foundation For Medical Education And Research Use of topical azathioprine and thioguanine to treat colorectal adenomas
CA2936748C (en) 2014-10-31 2017-08-08 Purdue Pharma Methods and compositions particularly for treatment of attention deficit disorder
US10722473B2 (en) 2018-11-19 2020-07-28 Purdue Pharma L.P. Methods and compositions particularly for treatment of attention deficit disorder

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DD95565B1 (de) * 1971-10-04 1986-10-29 Schering Ag Verfahren zur herstellung neuer pregnansaeurederivate
DE2150268C3 (de) * 1971-10-04 1980-11-06 Schering Ag, 1000 Berlin Und 4619 Bergkamen Pregnansäure-Derivate, Verfahren zu ihrer Herstellung sowie diese enthaltende Arzneimittel
DE2204360C2 (de) * 1972-01-27 1982-11-04 Schering Ag, 1000 Berlin Und 4619 Bergkamen Neue Pregnansäure-Derivate, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Präparate
SE378109B (zh) * 1972-05-19 1975-08-18 Bofors Ab
DE2264003C2 (de) * 1972-12-22 1982-11-04 Schering Ag, 1000 Berlin Und 4619 Bergkamen Neue Pregnansäure-Derivate, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Präparate
IE38659B1 (en) * 1972-12-22 1978-05-10 Schering Ag New pregnane acid derivatives
SE8403905D0 (sv) * 1984-07-30 1984-07-30 Draco Ab Liposomes and steroid esters

Also Published As

Publication number Publication date
PT83984B (pt) 1989-07-31
DE3675378D1 (de) 1990-12-06
ZA868750B (en) 1987-08-26
CA1318664C (en) 1993-06-01
PH23237A (en) 1989-06-06
DK605186D0 (da) 1986-12-16
FI84488C (fi) 1991-12-10
AU591950B2 (en) 1989-12-21
AR242797A1 (es) 1993-05-31
GR3001052T3 (en) 1992-03-20
IL80679A (en) 1992-03-29
CN1016508B (zh) 1992-05-06
LTIP1682A (en) 1995-07-25
EP0232690A1 (en) 1987-08-19
KR940004067B1 (ko) 1994-05-11
MY100750A (en) 1991-02-14
LV10959B (en) 1996-06-20
NO164243B (no) 1990-06-05
PL263041A1 (en) 1988-07-21
IE863245L (en) 1987-06-19
CN86108634A (zh) 1987-07-22
NO164243C (no) 1990-09-19
HU196831B (en) 1989-01-30
JPS62155296A (ja) 1987-07-10
IE59241B1 (en) 1994-01-26
NZ218614A (en) 1989-02-24
EP0232690B1 (en) 1990-10-31
FI865128A0 (fi) 1986-12-16
PL151627B1 (en) 1990-09-28
KR870006081A (ko) 1987-07-09
NO865004L (no) 1987-06-22
FI84488B (fi) 1991-08-30
ES2018656B3 (es) 1991-05-01
IL80679A0 (en) 1987-02-27
NO865004D0 (no) 1986-12-11
LV10959A (lv) 1995-12-20
ATE57935T1 (de) 1990-11-15
DD256703A5 (de) 1988-05-18
CS960486A2 (en) 1989-04-14
JO1499B1 (en) 1988-03-10
RU1839673C (ru) 1993-12-30
IS1559B (is) 1994-10-05
JPH0780900B2 (ja) 1995-08-30
DK605186A (da) 1987-06-20
DK168601B1 (da) 1994-05-02
FI865128A (fi) 1987-06-20
HUT44273A (en) 1988-02-29
IS3179A7 (is) 1987-06-20
LT3912B (en) 1996-04-25
AU6644886A (en) 1987-06-25
PT83984A (en) 1987-01-01
SE8506015D0 (sv) 1985-12-19

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