CS255884B2 - Process for preparing derivatives of substituted 3-phenyliminothiazolidine - Google Patents

Process for preparing derivatives of substituted 3-phenyliminothiazolidine Download PDF

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Publication number
CS255884B2
CS255884B2 CS853049A CS304985A CS255884B2 CS 255884 B2 CS255884 B2 CS 255884B2 CS 853049 A CS853049 A CS 853049A CS 304985 A CS304985 A CS 304985A CS 255884 B2 CS255884 B2 CS 255884B2
Authority
CS
Czechoslovakia
Prior art keywords
formula
amino
pharmaceutically acceptable
acid addition
thiazolidine
Prior art date
Application number
CS853049A
Other languages
Czech (cs)
English (en)
Other versions
CS304985A2 (en
Inventor
Karoly Lempert
Gyula Hornyak
Ferenc Bartha
Gabor Doleschall
Jozsef Fetter
Jozsef Nyitrai
Gyula Simig
Karoly Zauer
Peter Huszthy
Antal Feller
Lujza Petoecz
Enikoe Szirt
Katalin Grasser
Edit Berenyi
Zsuzsanna Orr
Etelka Pjeczka
Original Assignee
Egyt Gyogyszervegyeszeti Gyar
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Egyt Gyogyszervegyeszeti Gyar filed Critical Egyt Gyogyszervegyeszeti Gyar
Priority to CS863927A priority Critical patent/CS255873B2/cs
Priority to CS863928A priority patent/CS255874B2/cs
Publication of CS304985A2 publication Critical patent/CS304985A2/cs
Publication of CS255884B2 publication Critical patent/CS255884B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/18—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
CS853049A 1984-04-25 1985-04-25 Process for preparing derivatives of substituted 3-phenyliminothiazolidine CS255884B2 (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
CS863927A CS255873B2 (cs) 1984-04-25 1986-05-29 Způsob výroby derivátů substituovaného 3~fenyliminothiazolidinu
CS863928A CS255874B2 (cs) 1984-04-25 1986-05-29 Způsob výroby derivátů substituovaného 3-fenyliminothiazolidinu

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU841581A HU191408B (en) 1984-04-25 1984-04-25 Process for preparing new imino-thiazolidine derivatives

Publications (2)

Publication Number Publication Date
CS304985A2 CS304985A2 (en) 1987-07-16
CS255884B2 true CS255884B2 (en) 1988-03-15

Family

ID=10955127

Family Applications (1)

Application Number Title Priority Date Filing Date
CS853049A CS255884B2 (en) 1984-04-25 1985-04-25 Process for preparing derivatives of substituted 3-phenyliminothiazolidine

Country Status (24)

Country Link
US (1) US4665083A (da)
JP (1) JPS6127974A (da)
AT (1) AT394555B (da)
BE (1) BE902249A (da)
CA (1) CA1246086A (da)
CH (1) CH664564A5 (da)
CS (1) CS255884B2 (da)
DD (1) DD231790A5 (da)
DE (1) DE3514843A1 (da)
DK (1) DK183585A (da)
ES (3) ES8608499A1 (da)
FI (1) FI82454C (da)
FR (1) FR2563519B1 (da)
GB (1) GB2159814B (da)
GR (1) GR851006B (da)
HU (1) HU191408B (da)
IT (1) IT1208532B (da)
NL (1) NL8501184A (da)
NO (1) NO164417C (da)
PH (1) PH20995A (da)
PL (3) PL144860B1 (da)
PT (1) PT80336B (da)
SE (1) SE464813B (da)
SU (3) SU1366058A3 (da)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3442757A1 (de) * 1984-11-23 1986-05-28 Wella Ag, 6100 Darmstadt Verwendung von 2-nitroanilinderivaten in haarfaerbemitteln und neue 2-nitroanilinderivate
US5266701A (en) * 1988-07-01 1993-11-30 Ici Americas Inc. Process for production of 2-iminothiazolidines and oxazolidines
US4867782A (en) * 1988-07-01 1989-09-19 Ici Americas Inc. Novel herbicidal 2-sulfonyliminothiazolidines
US5240918A (en) * 1992-03-24 1993-08-31 Egis Gyogyszergyar 2-(substituted imino)-thiazolidines and process for the preparation thereof
EP0600489B1 (en) * 1992-12-04 1996-11-06 Sumitomo Chemical Company Limited Process for producing 2-iminothiazoline derivatives and process for producing their intermediates
US20090156644A1 (en) * 2005-07-21 2009-06-18 Jacob Westman Use of thiazole derivatives and analogues in the treatment of cancer
WO2010086613A1 (en) 2009-01-30 2010-08-05 Betagenon Ab Compounds useful as inhibitors as ampk
CN105722830B (zh) 2013-06-20 2019-06-04 拜耳作物科学股份公司 作为杀螨剂和杀昆虫剂的芳基硫醚衍生物和芳基亚砜衍生物

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB690238A (en) * 1949-08-23 1953-04-15 Knoll Ag Process of producing 3, 4-dimethyl-5-phenyl-2-iminothiazolidine
DE841149C (de) * 1949-11-01 1952-06-13 Knoll Ag Verfahren zur Herstellung von 3, 4-Dimethyl-5-phenyl-2-iminothiazolidin
DE910650C (de) * 1951-09-14 1954-05-03 Knoll Ag Verfahren zur Herstellung von 2-Amino-í¸ -thiazolinen bzw. Thiazolidon-(2)-imiden undderen Salzen
US3297708A (en) * 1965-10-06 1967-01-10 American Cyanamid Co Method of preparing thiazolidines
FR1510014A (fr) * 1966-12-05 1968-01-19 Aquitaine Petrole Préparation de dithiolannes
SU465792A3 (ru) * 1968-11-06 1975-03-30 Хиноин Гиогисцер-Ес Вегиесцети Термекек Гиара Рт (Фирма) Способ получени гетероциклических соединений
US3671537A (en) * 1969-06-05 1972-06-20 Gyogyszerkutato Intezet Certain 3-(2,6-dichlorophenyl)-2-iminothiazolidines
US3898340A (en) * 1970-04-15 1975-08-05 Bayer Ag Aryliminothiazolidine compositions and methods
CH533420A (de) * 1970-06-23 1973-02-15 Agripat Sa Mittel zur Regulierung des Pflanzenwachstums und zur Erhöhung des Zuckergehaltes in Zuckerrohr
US4029803A (en) * 1976-05-03 1977-06-14 Merck & Co., Inc. Method of treatment with 2-iminothiazolidines and thiazolines
DE2655369A1 (de) * 1976-12-03 1978-06-08 Schering Ag 5-(subst. phenyl)-oxazolidinone und deren schwefelanaloga sowie verfahren zu deren herstellung
HU180240B (en) * 1978-04-21 1983-02-28 Gyogyszerkutato Intezet Process for producing new,substituted 1,3-diaryl-2-iminoimidasolidines and 2-imino-hexahydro-pyrimidines
US4348393A (en) * 1978-06-09 1982-09-07 Delalande S.A. N-Aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones
JPS59227870A (ja) * 1983-06-07 1984-12-21 Yamanouchi Pharmaceut Co Ltd 新規２−グアニジノチアゾリン誘導体ならびにその製造法

Also Published As

Publication number Publication date
AT394555B (de) 1992-05-11
PH20995A (en) 1987-06-18
HUT37928A (en) 1986-03-28
IT1208532B (it) 1989-07-10
GB8510457D0 (en) 1985-05-30
NO164417B (no) 1990-06-25
ES551481A0 (es) 1986-12-16
PL144821B1 (en) 1988-07-30
BE902249A (fr) 1985-10-22
FI82454C (fi) 1991-03-11
ES8702391A1 (es) 1987-01-16
PL253089A1 (en) 1985-12-17
FI82454B (fi) 1990-11-30
FR2563519A1 (fr) 1985-10-31
CS304985A2 (en) 1987-07-16
ATA124285A (de) 1991-10-15
JPH0466478B2 (da) 1992-10-23
FR2563519B1 (fr) 1988-06-10
CA1246086A (en) 1988-12-06
SU1375132A3 (ru) 1988-02-15
PL145084B1 (en) 1988-08-31
HU191408B (en) 1987-02-27
GB2159814B (en) 1987-09-16
ES8701741A1 (es) 1986-12-16
PT80336B (pt) 1987-06-17
SU1549480A3 (ru) 1990-03-07
GB2159814A (en) 1985-12-11
SE464813B (sv) 1991-06-17
FI851606A0 (fi) 1985-04-23
IT8520482A0 (it) 1985-04-24
SE8501988D0 (sv) 1985-04-24
PT80336A (en) 1985-05-01
JPS6127974A (ja) 1986-02-07
ES542469A0 (es) 1986-07-16
NO851638L (no) 1985-10-28
CH664564A5 (de) 1988-03-15
DE3514843C2 (da) 1992-11-05
FI851606L (fi) 1985-10-26
US4665083A (en) 1987-05-12
ES551480A0 (es) 1987-01-16
ES8608499A1 (es) 1986-07-16
DD231790A5 (de) 1986-01-08
NL8501184A (nl) 1985-11-18
GR851006B (da) 1985-11-25
SU1366058A3 (ru) 1988-01-07
PL144860B1 (en) 1988-07-30
DE3514843A1 (de) 1985-10-31
NO164417C (no) 1990-10-10
DK183585A (da) 1985-10-26
SE8501988L (sv) 1985-10-26
DK183585D0 (da) 1985-04-24

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