CS226008B2 - Method of preparing piperidinopropyl derivatives - Google Patents

Method of preparing piperidinopropyl derivatives Download PDF

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Publication number
CS226008B2
CS226008B2 CS801056A CS105680A CS226008B2 CS 226008 B2 CS226008 B2 CS 226008B2 CS 801056 A CS801056 A CS 801056A CS 105680 A CS105680 A CS 105680A CS 226008 B2 CS226008 B2 CS 226008B2
Authority
CS
Czechoslovakia
Prior art keywords
group
carbon atoms
hydrogen
formula
optionally
Prior art date
Application number
CS801056A
Other languages
Czech (cs)
English (en)
Inventor
Walter Gunar Dr Friebe
Helmut Michel
Carl H Dr Ross
Fritz Dr Wiedemann
Gisbert Dr Sponer
Wolfgang Prof Dr Schaumann
Original Assignee
Boehringer Mannheim Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Mannheim Gmbh filed Critical Boehringer Mannheim Gmbh
Priority to CS807703A priority Critical patent/CS226022B2/cs
Priority to CS814585A priority patent/CS226029B2/cs
Publication of CS226008B2 publication Critical patent/CS226008B2/cs

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
    • C07D211/22Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/49Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups
    • C07C205/56Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups bound to carbon atoms of six-membered aromatic rings and carboxyl groups bound to acyclic carbon atoms of the carbon skeleton

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CS801056A 1979-02-16 1980-02-15 Method of preparing piperidinopropyl derivatives CS226008B2 (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
CS807703A CS226022B2 (cs) 1979-02-16 1980-11-13 Způsob přípravy piperidinopropylových derivátů
CS814585A CS226029B2 (cs) 1979-02-16 1981-06-18 Způsob přípravy piperidinopropylových derivátů

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19792905876 DE2905876A1 (de) 1979-02-16 1979-02-16 Neue piperidinopropylderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Publications (1)

Publication Number Publication Date
CS226008B2 true CS226008B2 (en) 1984-03-19

Family

ID=6063043

Family Applications (2)

Application Number Title Priority Date Filing Date
CS801056A CS226008B2 (en) 1979-02-16 1980-02-15 Method of preparing piperidinopropyl derivatives
CS807704A CS226021B2 (en) 1979-02-16 1980-02-15 Method of presparing piperidine propylderivatives

Family Applications After (1)

Application Number Title Priority Date Filing Date
CS807704A CS226021B2 (en) 1979-02-16 1980-02-15 Method of presparing piperidine propylderivatives

Country Status (16)

Country Link
US (1) US4288442A (fi)
EP (1) EP0014928B1 (fi)
JP (1) JPS55113777A (fi)
AT (1) ATE968T1 (fi)
AU (1) AU529849B2 (fi)
CA (1) CA1115703A (fi)
CS (2) CS226008B2 (fi)
DD (1) DD149069A5 (fi)
DE (2) DE2905876A1 (fi)
DK (1) DK65780A (fi)
ES (1) ES8102719A1 (fi)
FI (1) FI66370C (fi)
HU (1) HU184238B (fi)
IL (1) IL59351A (fi)
SU (2) SU1021342A3 (fi)
ZA (1) ZA80787B (fi)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2901336A1 (de) 1979-01-15 1980-07-24 Boehringer Mannheim Gmbh Neue arylether, verfahren zu deren herstellung sowie diese verbindungen enthaltende arzneimittel
BE883069A (fr) 1979-05-04 1980-08-18 Continental Pharma Derives de phenylethylamine, leur preparation et utilisation ainsi que composition contenant ces derives.
DE3200304A1 (de) * 1981-01-16 1982-08-26 Sandoz-Patent-GmbH, 7850 Lörrach 3-aminopropoxyaryl-derivate, ihre herstellung und sie enthaltende arzneimittel
DE3209271A1 (de) * 1982-03-13 1983-09-15 Boehringer Mannheim Gmbh, 6800 Mannheim Bicyclische phenolether, verfahren zu deren herstellung sowie diese verbindungen enthaltende arzneimittel
ZA848275B (en) * 1983-12-28 1985-08-28 Degussa New piridine-2-ethers or pyridine-2-thioethers having a nitrogen-containing cycloaliphatic ring
US5231184A (en) * 1987-11-23 1993-07-27 Janssen Pharmaceutica N.V. Pridazinamine derivatives
DE3839743A1 (de) * 1988-11-25 1990-05-31 Hoechst Ag Verfahren zur herstellung von benzimidazolonen
US5082847A (en) * 1990-07-18 1992-01-21 Syntex (U.S.A.) Inc. Carbostyril compounds connected via an oxyalkyl group with a piperidine ring and having pharmaceutical utility
US5614523A (en) * 1995-01-17 1997-03-25 Eli Lilly And Company Compounds having effects on serotonin-related systems
US5627196A (en) * 1995-01-17 1997-05-06 Eli Lilly And Company Compounds having effects on serotonin-related systems
US5576321A (en) * 1995-01-17 1996-11-19 Eli Lilly And Company Compounds having effects on serotonin-related systems
US5789402A (en) * 1995-01-17 1998-08-04 Eli Lilly Company Compounds having effects on serotonin-related systems
US5741789A (en) * 1995-01-17 1998-04-21 Eli Lilly And Company Compounds having effects on serotonin-related systems

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE255000C (fi) *
DE2550001A1 (de) 1975-11-07 1977-05-12 Boehringer Mannheim Gmbh Neue indol-derivate und verfahren zu ihrer herstellung
DE2701794A1 (de) * 1976-01-21 1977-07-28 Ciba Geigy Ag Oxigenierte n-aryl-diazacyclen
US4126687A (en) * 1976-05-17 1978-11-21 Janssen Pharmaceutica N.V. Antiemetic, 1-(benzimidazolyl-alkyl)-piperidine derivatives
US4146630A (en) * 1976-11-12 1979-03-27 Boehringer Mannheim Gmbh Blood pressure lowering and adrenergic β-receptor inhibiting 3-(4-phenoxymethylpiperidino)-propyl-phenyl ethers
DE2737630A1 (de) * 1977-08-20 1979-03-01 Boehringer Mannheim Gmbh Neue aminopropanolderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
US4200641A (en) * 1976-12-21 1980-04-29 Janssen Pharmaceutica, N.V. 1-[(Heterocyclyl)-alkyl]-4-diarylmethoxy piperidine derivatives

Also Published As

Publication number Publication date
FI66370C (fi) 1984-10-10
FI800407A (fi) 1980-08-17
US4288442A (en) 1981-09-08
ATE968T1 (de) 1982-05-15
EP0014928A1 (de) 1980-09-03
ZA80787B (en) 1981-03-25
EP0014928B1 (de) 1982-05-05
DK65780A (da) 1980-08-17
SU1021342A3 (ru) 1983-05-30
CA1115703A (en) 1982-01-05
ES488401A0 (es) 1981-02-16
JPS55113777A (en) 1980-09-02
DD149069A5 (de) 1981-06-24
SU1241987A3 (ru) 1986-06-30
CS226021B2 (en) 1984-03-19
IL59351A (en) 1984-01-31
DE2905876A1 (de) 1980-08-28
IL59351A0 (en) 1980-05-30
ES8102719A1 (es) 1981-02-16
FI66370B (fi) 1984-06-29
DE3060353D1 (en) 1982-06-24
HU184238B (en) 1984-07-30
AU5540980A (en) 1980-08-21
AU529849B2 (en) 1983-06-23

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