CO6541539A2 - Procesos para preparar las formas cristalinas a y b de ilaprazol y proceso para convertir las formas cristalinas - Google Patents
Procesos para preparar las formas cristalinas a y b de ilaprazol y proceso para convertir las formas cristalinasInfo
- Publication number
- CO6541539A2 CO6541539A2 CO12097489A CO12097489A CO6541539A2 CO 6541539 A2 CO6541539 A2 CO 6541539A2 CO 12097489 A CO12097489 A CO 12097489A CO 12097489 A CO12097489 A CO 12097489A CO 6541539 A2 CO6541539 A2 CO 6541539A2
- Authority
- CO
- Colombia
- Prior art keywords
- crystal forms
- crystalline form
- ilaprazole
- preparing
- ilaprazol
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR1020090121209A KR101144600B1 (ko) | 2009-12-08 | 2009-12-08 | 일라프라졸의 결정형 a, b의 제조방법 및 이들 결정형의 변환방법 |
Publications (1)
Publication Number | Publication Date |
---|---|
CO6541539A2 true CO6541539A2 (es) | 2012-10-16 |
Family
ID=44146052
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CO12097489A CO6541539A2 (es) | 2009-12-08 | 2012-06-08 | Procesos para preparar las formas cristalinas a y b de ilaprazol y proceso para convertir las formas cristalinas |
Country Status (7)
Country | Link |
---|---|
KR (1) | KR101144600B1 (ru) |
BR (1) | BR112012012212A2 (ru) |
CO (1) | CO6541539A2 (ru) |
EA (1) | EA019058B1 (ru) |
IN (1) | IN2012DN03176A (ru) |
UA (1) | UA102787C2 (ru) |
WO (1) | WO2011071314A2 (ru) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN103204842B (zh) * | 2012-01-13 | 2014-10-15 | 丽珠医药集团股份有限公司 | 结晶型艾普拉唑钠水合物及其制备方法 |
CN103204843B (zh) * | 2012-01-13 | 2014-12-31 | 丽珠医药集团股份有限公司 | 结晶型艾普拉唑钠乙醇化物及其制备方法 |
WO2013114232A1 (en) | 2012-02-02 | 2013-08-08 | Lupin Limited | Process for preparation of crystalline form l of ilaprazole |
CN102746277B (zh) * | 2012-06-21 | 2014-05-14 | 丽珠医药集团股份有限公司 | 一种结晶形式的艾普拉唑钠及其制备方法 |
CN102746275B (zh) * | 2012-06-21 | 2014-07-16 | 丽珠医药集团股份有限公司 | 结晶型艾普拉唑钠及其制备方法 |
CN102746276B (zh) * | 2012-06-21 | 2014-07-02 | 丽珠医药集团股份有限公司 | 一种艾普拉唑钠晶型及其制备方法 |
CN113045544A (zh) * | 2014-09-04 | 2021-06-29 | 江苏奥赛康药业有限公司 | 艾普拉唑钠化合物及其药物组合物 |
CN115403560A (zh) * | 2017-11-06 | 2022-11-29 | 丽珠医药集团股份有限公司 | 一种艾普拉唑镁晶型及其制备方法 |
KR102027388B1 (ko) * | 2017-11-15 | 2019-10-01 | 주식회사 다산제약 | 고순도 일라프라졸 결정형 b의 제조방법 |
CN111187255B (zh) * | 2020-01-13 | 2021-07-20 | 丽珠医药集团股份有限公司 | 右旋艾普拉唑钾盐的制备方法和右旋艾普拉唑的制备方法 |
KR20220065235A (ko) | 2020-11-13 | 2022-05-20 | 주식회사 파마코스텍 | 일라프라졸 혼형 결정의 신규한 제조방법 |
KR102250509B1 (ko) * | 2020-12-09 | 2021-05-11 | 유니셀랩 주식회사 | 새로운 일라프라졸/자일리톨 공결정 |
KR20210019469A (ko) | 2021-02-02 | 2021-02-22 | 주식회사 파마코스텍 | 일라프라졸 나트륨 결정형 및 신규한 제조방법 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR20090086121A (ko) * | 2006-12-29 | 2009-08-10 | 일양약품주식회사 | 용매화 일라프라졸의 결정형 |
WO2008083319A1 (en) * | 2006-12-29 | 2008-07-10 | Il Yang Pharmaceutical Company, Ltd. | Solid state forms of enantiopure ilaprazole |
-
2009
- 2009-12-08 KR KR1020090121209A patent/KR101144600B1/ko active IP Right Grant
-
2010
- 2010-12-08 WO PCT/KR2010/008767 patent/WO2011071314A2/en active Application Filing
- 2010-12-08 BR BR112012012212A patent/BR112012012212A2/pt not_active Application Discontinuation
- 2010-12-08 UA UAA201207006A patent/UA102787C2/ru unknown
- 2010-12-08 EA EA201200716A patent/EA019058B1/ru not_active IP Right Cessation
- 2010-12-08 IN IN3176DEN2012 patent/IN2012DN03176A/en unknown
-
2012
- 2012-06-08 CO CO12097489A patent/CO6541539A2/es unknown
Also Published As
Publication number | Publication date |
---|---|
EA019058B1 (ru) | 2013-12-30 |
WO2011071314A3 (en) | 2011-11-10 |
BR112012012212A2 (pt) | 2015-09-08 |
IN2012DN03176A (ru) | 2015-09-25 |
KR101144600B1 (ko) | 2012-05-16 |
WO2011071314A2 (en) | 2011-06-16 |
EA201200716A1 (ru) | 2012-10-30 |
KR20110064545A (ko) | 2011-06-15 |
UA102787C2 (ru) | 2013-08-12 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CO6541539A2 (es) | Procesos para preparar las formas cristalinas a y b de ilaprazol y proceso para convertir las formas cristalinas | |
AR076974A1 (es) | Metodo para sintetizar pirfenidona | |
AR098260A2 (es) | Polimorfo cristalino de una sal de bisulfato de un antagonista del receptor de trombina, proceso para su preparación, composición y forma purificada | |
EA201000147A1 (ru) | Способ выделения и очистки монтелукаста | |
MY167395A (en) | Method for producing glufosinate p free acid | |
AR076027A1 (es) | Metodos e intermediarios para la preparacion de agentes farmaceuticos | |
AR076891A1 (es) | Metodo para la preparacion de clorhidrato de nalmefeno | |
PE20061014A1 (es) | Clorhidrato de lercanidipina amorfo | |
CU20120137A7 (es) | Hidrato del hidrocloruro de agomelatina y preparación de éste | |
CL2011000296A1 (es) | Proceso de preparación del ester metílico del ácido 4-oxo-octahidro-indol-1-carboxílico y compuestos intermediarios utilizados. | |
CO6700138A1 (es) | Procedimiento de preparación de sal de l-arginina de perindoprilo | |
ES2571043T3 (es) | Preparación de dihidropiridinas | |
MX2014004823A (es) | Colorantes acidos de trisazo. | |
AR081659A1 (es) | Procedimiento de obtencion de la forma cristalina ii del febuxostat | |
AR087344A1 (es) | Formas polimorficas del acido 5-(3,3-dimetil-but-1-inil)-3-[(trans-4-hidroxi-ciclohexil)-(trans-4-metil-ciclohexancarbonil)-amino]-tiofen-2-carboxilico y su uso en el tratamiento de la hepatitis c | |
AR104145A1 (es) | Método de producción de epirrubicina, intermediario y sal farmacéutica | |
CL2012001528A1 (es) | Proceso para preparar la forma cristalina a de ilaprazol a partir de una sal inorganica de ilaprazol y posterior neutralizacion de la sal con un acido en un solvente de reaccion; y proceso para preparar la forma cristalina b de ilaprazol en la forma cristalina a de ilaprazol. | |
MX2010007923A (es) | Forma cristalina de abacavir que esta esencialmente libre de disolvente. | |
CU20120136A7 (es) | Hidrato del hidrobromuro de agomelatina y preparación de éste | |
AR094240A1 (es) | Proceso para producir cristal de compuesto de pirazol | |
AR071804A1 (es) | Cristales de sucralosa enjuagados con regulador (buffer) | |
TH137478B (th) | กระบวนการสำหรับจัดเตรียมรูปแบบผลึก a และ b ของไอลาพราโซล และกระบวนการสำหรับการเปลี่ยนรูปแบบผลึก | |
CO6280533A2 (es) | Proceso para preparar un compuesto intermedio para sintetizar un antiulcerante | |
BR112016006628A2 (pt) | forma polimórfica de hiodesoxicolato de sódio (nahdc) e seu processo de preparação | |
TH137478A (th) | กระบวนการสำหรับจัดเตรียมรูปแบบผลึก a และ b ของไอลาพราโซล และกระบวนการสำหรับการเปลี่ยนรูปแบบผลึก |