BR112012012212A2 - processos de preparo de formas cristalinas a e b de ilaprazol e processo para conversão das formas cristalinas - Google Patents

processos de preparo de formas cristalinas a e b de ilaprazol e processo para conversão das formas cristalinas

Info

Publication number
BR112012012212A2
BR112012012212A2 BR112012012212A BR112012012212A BR112012012212A2 BR 112012012212 A2 BR112012012212 A2 BR 112012012212A2 BR 112012012212 A BR112012012212 A BR 112012012212A BR 112012012212 A BR112012012212 A BR 112012012212A BR 112012012212 A2 BR112012012212 A2 BR 112012012212A2
Authority
BR
Brazil
Prior art keywords
crystalline forms
ilaprazole
processes
converting
preparing
Prior art date
Application number
BR112012012212A
Other languages
English (en)
Inventor
Dong Yeon Kim
Hee Yun Kim
Jae Soo Shin
Jun Yeoun Lee
Jung Woo Kim
Kwi Hyung Cho
Sang Don Nam
Sung Tae Park
Original Assignee
Il Yang Pharm Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Il Yang Pharm Co Ltd filed Critical Il Yang Pharm Co Ltd
Publication of BR112012012212A2 publication Critical patent/BR112012012212A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Saccharide Compounds (AREA)
BR112012012212A 2009-12-08 2010-12-08 processos de preparo de formas cristalinas a e b de ilaprazol e processo para conversão das formas cristalinas BR112012012212A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR1020090121209A KR101144600B1 (ko) 2009-12-08 2009-12-08 일라프라졸의 결정형 a, b의 제조방법 및 이들 결정형의 변환방법
PCT/KR2010/008767 WO2011071314A2 (en) 2009-12-08 2010-12-08 Processes for preparing crystalline forms a and b of ilaprazole and process for converting the crystalline forms

Publications (1)

Publication Number Publication Date
BR112012012212A2 true BR112012012212A2 (pt) 2015-09-08

Family

ID=44146052

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112012012212A BR112012012212A2 (pt) 2009-12-08 2010-12-08 processos de preparo de formas cristalinas a e b de ilaprazol e processo para conversão das formas cristalinas

Country Status (7)

Country Link
KR (1) KR101144600B1 (pt)
BR (1) BR112012012212A2 (pt)
CO (1) CO6541539A2 (pt)
EA (1) EA019058B1 (pt)
IN (1) IN2012DN03176A (pt)
UA (1) UA102787C2 (pt)
WO (1) WO2011071314A2 (pt)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103204843B (zh) * 2012-01-13 2014-12-31 丽珠医药集团股份有限公司 结晶型艾普拉唑钠乙醇化物及其制备方法
CN103204842B (zh) * 2012-01-13 2014-10-15 丽珠医药集团股份有限公司 结晶型艾普拉唑钠水合物及其制备方法
WO2013114232A1 (en) 2012-02-02 2013-08-08 Lupin Limited Process for preparation of crystalline form l of ilaprazole
CN102746276B (zh) * 2012-06-21 2014-07-02 丽珠医药集团股份有限公司 一种艾普拉唑钠晶型及其制备方法
CN102746277B (zh) * 2012-06-21 2014-05-14 丽珠医药集团股份有限公司 一种结晶形式的艾普拉唑钠及其制备方法
CN102746275B (zh) * 2012-06-21 2014-07-16 丽珠医药集团股份有限公司 结晶型艾普拉唑钠及其制备方法
CN113045544A (zh) * 2014-09-04 2021-06-29 江苏奥赛康药业有限公司 艾普拉唑钠化合物及其药物组合物
CN107857756B (zh) * 2017-11-06 2022-08-30 丽珠医药集团股份有限公司 一种艾普拉唑镁晶型及其制备方法
KR102027388B1 (ko) * 2017-11-15 2019-10-01 주식회사 다산제약 고순도 일라프라졸 결정형 b의 제조방법
CN111187255B (zh) * 2020-01-13 2021-07-20 丽珠医药集团股份有限公司 右旋艾普拉唑钾盐的制备方法和右旋艾普拉唑的制备方法
KR20220065235A (ko) 2020-11-13 2022-05-20 주식회사 파마코스텍 일라프라졸 혼형 결정의 신규한 제조방법
KR102250509B1 (ko) * 2020-12-09 2021-05-11 유니셀랩 주식회사 새로운 일라프라졸/자일리톨 공결정
KR20210019469A (ko) 2021-02-02 2021-02-22 주식회사 파마코스텍 일라프라졸 나트륨 결정형 및 신규한 제조방법

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008083319A1 (en) * 2006-12-29 2008-07-10 Il Yang Pharmaceutical Company, Ltd. Solid state forms of enantiopure ilaprazole
MY146462A (en) * 2006-12-29 2012-08-15 Il Yang Pharmaceutical Company Ltd Crystalline forms of solvated ilaprazole

Also Published As

Publication number Publication date
CO6541539A2 (es) 2012-10-16
KR101144600B1 (ko) 2012-05-16
WO2011071314A2 (en) 2011-06-16
KR20110064545A (ko) 2011-06-15
WO2011071314A3 (en) 2011-11-10
IN2012DN03176A (pt) 2015-09-25
UA102787C2 (ru) 2013-08-12
EA201200716A1 (ru) 2012-10-30
EA019058B1 (ru) 2013-12-30

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B06T Formal requirements before examination [chapter 6.20 patent gazette]
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: AS CLASSIFICACOES ANTERIORES ERAM: C07D 401/14 , C07D 403/14 , C07D 235/24

Ipc: C07D 401/14 (2006.01), C07D 403/14 (2006.01), C07D

B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]
B12B Appeal against refusal [chapter 12.2 patent gazette]