CO6160327A2 - Forma cristalina de la sal diclorhidrato de ((2s)-2-(5-(4`-(2((2s)-1-((2s)-2-((metoxicarbonil)amino)-3-metilbutaniol)-2-pirrolidinil)-1h-imidazol-5-il-4bifenilil)-1h-imidazol-2-il)-1-pirrolidinil)carbonil)-2-metilpropil)carbamato de metilo - Google Patents

Forma cristalina de la sal diclorhidrato de ((2s)-2-(5-(4`-(2((2s)-1-((2s)-2-((metoxicarbonil)amino)-3-metilbutaniol)-2-pirrolidinil)-1h-imidazol-5-il-4bifenilil)-1h-imidazol-2-il)-1-pirrolidinil)carbonil)-2-metilpropil)carbamato de metilo

Info

Publication number
CO6160327A2
CO6160327A2 CO10011972A CO10011972A CO6160327A2 CO 6160327 A2 CO6160327 A2 CO 6160327A2 CO 10011972 A CO10011972 A CO 10011972A CO 10011972 A CO10011972 A CO 10011972A CO 6160327 A2 CO6160327 A2 CO 6160327A2
Authority
CO
Colombia
Prior art keywords
imidazol
pirrolidinil
crystalline form
amino
methyl carbamate
Prior art date
Application number
CO10011972A
Other languages
English (en)
Spanish (es)
Inventor
Soojin Kim
Qi Gao
Fukang Yang
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39739413&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO6160327(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of CO6160327A2 publication Critical patent/CO6160327A2/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CO10011972A 2007-08-08 2010-02-04 Forma cristalina de la sal diclorhidrato de ((2s)-2-(5-(4`-(2((2s)-1-((2s)-2-((metoxicarbonil)amino)-3-metilbutaniol)-2-pirrolidinil)-1h-imidazol-5-il-4bifenilil)-1h-imidazol-2-il)-1-pirrolidinil)carbonil)-2-metilpropil)carbamato de metilo CO6160327A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US95459207P 2007-08-08 2007-08-08

Publications (1)

Publication Number Publication Date
CO6160327A2 true CO6160327A2 (es) 2010-05-20

Family

ID=39739413

Family Applications (1)

Application Number Title Priority Date Filing Date
CO10011972A CO6160327A2 (es) 2007-08-08 2010-02-04 Forma cristalina de la sal diclorhidrato de ((2s)-2-(5-(4`-(2((2s)-1-((2s)-2-((metoxicarbonil)amino)-3-metilbutaniol)-2-pirrolidinil)-1h-imidazol-5-il-4bifenilil)-1h-imidazol-2-il)-1-pirrolidinil)carbonil)-2-metilpropil)carbamato de metilo

Country Status (20)

Country Link
US (1) US8629171B2 (enExample)
EP (1) EP2183244B1 (enExample)
JP (1) JP5244179B2 (enExample)
KR (1) KR101508022B1 (enExample)
CN (1) CN101778840B (enExample)
AR (2) AR070016A1 (enExample)
AU (1) AU2008284100B2 (enExample)
BR (1) BRPI0815142B8 (enExample)
CA (1) CA2695729C (enExample)
CL (1) CL2008002354A1 (enExample)
CO (1) CO6160327A2 (enExample)
EA (1) EA018152B1 (enExample)
ES (1) ES2402791T3 (enExample)
IL (1) IL203684A (enExample)
MX (1) MX2010001368A (enExample)
NZ (1) NZ583148A (enExample)
PE (1) PE20090940A1 (enExample)
TW (1) TWI359813B (enExample)
WO (1) WO2009020828A1 (enExample)
ZA (1) ZA201000843B (enExample)

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US8236950B2 (en) 2006-12-20 2012-08-07 Abbott Laboratories Anti-viral compounds
US7728027B2 (en) * 2007-08-08 2010-06-01 Bristol-Myers Squibb Company Process for synthesizing compounds useful for treating hepatitis C

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AU2008284100A1 (en) 2009-02-12
MX2010001368A (es) 2010-03-01
CL2008002354A1 (es) 2009-01-02
EA201000196A1 (ru) 2010-06-30
ES2402791T3 (es) 2013-05-09
AR104566A2 (es) 2017-08-02
TWI359813B (en) 2012-03-11
IL203684A (en) 2014-12-31
BRPI0815142A2 (pt) 2015-02-03
EP2183244B1 (en) 2013-01-23
CA2695729A1 (en) 2009-02-12
EP2183244A1 (en) 2010-05-12
AU2008284100B2 (en) 2014-01-16
BRPI0815142B1 (pt) 2018-09-25
CN101778840A (zh) 2010-07-14
BRPI0815142B8 (pt) 2021-05-25
NZ583148A (en) 2011-04-29
AR070016A1 (es) 2010-03-10
US8629171B2 (en) 2014-01-14
JP5244179B2 (ja) 2013-07-24
PE20090940A1 (es) 2009-07-13
HK1144089A1 (en) 2011-01-28
CA2695729C (en) 2015-03-31
TW200911790A (en) 2009-03-16
US20090041716A1 (en) 2009-02-12
JP2010535785A (ja) 2010-11-25
WO2009020828A1 (en) 2009-02-12
KR20100042641A (ko) 2010-04-26
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