CO5180587A1 - Composicion farmaceutica de orlistat que contiene tensoactivos y dispersantes - Google Patents

Composicion farmaceutica de orlistat que contiene tensoactivos y dispersantes

Info

Publication number
CO5180587A1
CO5180587A1 CO00068859A CO00068859A CO5180587A1 CO 5180587 A1 CO5180587 A1 CO 5180587A1 CO 00068859 A CO00068859 A CO 00068859A CO 00068859 A CO00068859 A CO 00068859A CO 5180587 A1 CO5180587 A1 CO 5180587A1
Authority
CO
Colombia
Prior art keywords
dispersant
pharmaceutical composition
tensoactive
composition containing
orlistat
Prior art date
Application number
CO00068859A
Other languages
English (en)
Spanish (es)
Inventor
Smidt Passchier Christiaan De
Paul Hadvary
Hans Lengsfeld
Thomas Rades
Hans Steffen
Joseph Tardio
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8238990&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO5180587(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of CO5180587A1 publication Critical patent/CO5180587A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365—Lactones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/485—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0007—Effervescent

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Biophysics (AREA)
  • Diabetes (AREA)
  • Molecular Biology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Inorganic Chemistry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Plant Substances (AREA)
CO00068859A 1999-09-13 2000-09-12 Composicion farmaceutica de orlistat que contiene tensoactivos y dispersantes CO5180587A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP99118180 1999-09-13

Publications (1)

Publication Number Publication Date
CO5180587A1 true CO5180587A1 (es) 2002-07-30

Family

ID=8238990

Family Applications (1)

Application Number Title Priority Date Filing Date
CO00068859A CO5180587A1 (es) 1999-09-13 2000-09-12 Composicion farmaceutica de orlistat que contiene tensoactivos y dispersantes

Country Status (38)

Country Link
US (3) US20030181512A1 (cs)
EP (1) EP1216025B1 (cs)
JP (1) JP4217016B2 (cs)
KR (1) KR100572434B1 (cs)
CN (1) CN1197551C (cs)
AR (1) AR025587A1 (cs)
AT (1) ATE333866T1 (cs)
AU (1) AU769415B2 (cs)
BR (2) BR0013939A (cs)
CA (1) CA2383916C (cs)
CO (1) CO5180587A1 (cs)
CY (1) CY1106180T1 (cs)
CZ (1) CZ301901B6 (cs)
DE (1) DE60029602T2 (cs)
DK (1) DK1216025T3 (cs)
EG (1) EG24117A (cs)
ES (1) ES2267563T3 (cs)
HR (1) HRP20020205B1 (cs)
HU (1) HU228858B1 (cs)
IL (1) IL148494A0 (cs)
JO (1) JO2386B1 (cs)
MA (1) MA26818A1 (cs)
ME (1) ME00674B (cs)
MX (1) MXPA02002034A (cs)
MY (1) MY130200A (cs)
NO (1) NO331906B1 (cs)
NZ (1) NZ517545A (cs)
PE (1) PE20010595A1 (cs)
PL (1) PL199870B1 (cs)
PT (1) PT1216025E (cs)
RS (1) RS50422B (cs)
RU (1) RU2239428C2 (cs)
SI (1) SI1216025T1 (cs)
TR (1) TR200200606T2 (cs)
TW (1) TWI243060B (cs)
UY (1) UY26338A1 (cs)
WO (1) WO2001019340A1 (cs)
ZA (1) ZA200201518B (cs)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2001289699B2 (en) 2000-07-28 2006-06-01 Cheplapharm Arzneimittel Gmbh New pharmaceutical composition
US6730319B2 (en) * 2001-06-06 2004-05-04 Hoffmann-La Roche Inc. Pharmaceutical compositions having depressed melting points
US20030027786A1 (en) 2001-06-06 2003-02-06 Karsten Maeder Lipase inhibiting composition
US8372430B2 (en) 2002-12-17 2013-02-12 The Procter & Gamble Company Compositions, methods, and kits useful for the alleviation of gastrointestinal effects
FI20045076A7 (fi) * 2004-03-15 2005-09-16 Bioferme Oy Funktionaalinen elintarvike
BRPI0607549A2 (pt) * 2005-04-15 2009-09-15 Clarus Therapeutics Inc sistemas de distribuição farmacêutica para fármacos hidrófobos e composições compreendendo os mesmos
KR100910000B1 (ko) * 2005-05-13 2009-07-29 씨제이제일제당 (주) 리파아제 저해제 함유 약학 조성물
US20090208584A1 (en) * 2005-06-09 2009-08-20 Tomohiro Yoshinari Solid preparation
KR100669497B1 (ko) * 2005-08-17 2007-01-16 보람제약주식회사 안정성과 용출률이 뛰어난 약리학적 조성물 및 그 제조방법
WO2007033522A1 (fr) * 2005-09-21 2007-03-29 Shenzhen Tys R & D Co., Ltd. Formulation de gélule contenant de la moxifloxacine et son procédé de préparation
KR101252635B1 (ko) 2006-04-20 2013-04-10 (주)아모레퍼시픽 리파아제 저해제 및 친유성 오일흡수제를 포함하는 약학조성물 및 이로부터 제조된 경구 투여용 제제
TR200607613A2 (tr) * 2006-12-29 2008-07-21 NOBEL İLAÇ SAN.ve TiC.A.Ş. Lipaz inhibitörü içeren farmasötik formülasyonlar
EP1970051A1 (en) * 2007-03-14 2008-09-17 Merz Pharma GmbH & Co.KGaA Use of an aqueous micro-emulsion for the preparation of a formulation for the treatment of adipose diseases
KR101439470B1 (ko) * 2007-05-22 2014-09-16 한미사이언스 주식회사 오를리스타트 및 대변 연화제를 포함하는 비만의 예방 또는치료용 조성물
EP2036575B1 (en) * 2007-09-12 2010-08-18 Mader S.r.l. Pharmaceutical compositions for oral use for treating patients affected by obesity
EP2044930A1 (en) * 2007-10-01 2009-04-08 Nestec S.A. Composition for controlling lipase catalyzed reactions
PL216542B1 (pl) 2008-03-20 2014-04-30 Zakłady Farmaceutyczne POLPHARMA Spółka Akcyjna Sposób wytwarzania stabilnej kompozycji orlistatu w postaci kapsułkowanego proszku
WO2010042499A1 (en) * 2008-10-06 2010-04-15 Banner Pharmacaps, Inc. Stable solutions of orlistat for pharmaceutical dosage forms
KR20100075260A (ko) * 2008-12-24 2010-07-02 주식회사종근당 리파아제 저해제의 부작용 개선을 위한 신규한 약제학적 조성물
BRPI0901602B8 (pt) 2009-04-03 2021-05-25 Ems S/A formulação farmacêuticas
RU2441654C2 (ru) * 2010-02-17 2012-02-10 Лабораториос Баго С.А. Фармацевтическая композиция с активностью против ожирения, включающая премикс чистого орлистата, и способ ее изготовления
ITRM20120331A1 (it) 2012-07-12 2014-01-13 Guidotti & C Spa Labor Composizioni pediatriche orali liquide contenenti nepadutant.
BR112017021995A2 (pt) * 2015-04-14 2018-07-10 Zim Laboratories Ltd formulação farmacêutica compreendendo drogas de baixa fusão e altamente lipofílicas e método de melhora da dissolução
CN106310287B (zh) * 2015-06-25 2019-03-19 山东省药学科学院 新利司他药用组合物及其制备方法
MY196635A (en) * 2018-06-22 2023-04-25 Sime Darby Plantation Intellectual Property Sdn Bhd Method For Reducing Formation of Free Fatty Acids in Plants
CN115105476B (zh) * 2021-03-23 2023-11-14 山东新时代药业有限公司 一种奥利司他冻干口服制剂及其制备工艺
CN114983938A (zh) * 2022-05-19 2022-09-02 广东嘉博制药有限公司 一种奥利司他口服复合乳液及其制备方法

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1247547A (en) 1983-06-22 1988-12-28 Paul Hadvary Leucine derivatives
EP0281200B1 (en) * 1987-03-02 1994-01-19 Yamanouchi Europe B.V. Pharmaceutical composition, pharmaceutical granulate and process for their preparation
SU1510148A1 (ru) * 1988-01-26 1995-04-30 Всесоюзный научно-исследовательский институт химии и технологии лекарственных средств Способ получения ингибитора липазы
TW381025B (en) * 1993-08-05 2000-02-01 Hoffmann La Roche Pharmaceutical composition containing a glucosidase inhibitor and a lipase inhibitor
IT1282673B1 (it) 1996-02-23 1998-03-31 Ist Naz Stud Cura Dei Tumori Derivati della camptotecina e loro uso come agenti antitumorali
US5891469A (en) * 1997-04-02 1999-04-06 Pharmos Corporation Solid Coprecipitates for enhanced bioavailability of lipophilic substances
EP1017366A4 (en) 1996-09-01 2006-03-22 Pharmos Corp SOLID COPARCIPITATES FOR IMPROVED BIOVERABILITY OF LIPOPHILIC SUBSTANCES
HU230834B1 (hu) * 1997-02-05 2018-07-30 F.Hoffmann-La Roche Ag Tetrahidrolipsztatin felhasználása
US6004996A (en) * 1997-02-05 1999-12-21 Hoffman-La Roche Inc. Tetrahydrolipstatin containing compositions
US6267952B1 (en) 1998-01-09 2001-07-31 Geltex Pharmaceuticals, Inc. Lipase inhibiting polymers
DK1105123T3 (da) 1998-08-14 2004-08-09 Hoffmann La Roche Farmaceutiske præparater indeholdende lipase-inhibitorer og chitosan
ES2242413T3 (es) 1998-08-14 2005-11-01 F. Hoffmann-La Roche Ag Composiciones farmaceuticas que contienen inhibidores de lipasa.
US6368622B2 (en) * 1999-01-29 2002-04-09 Abbott Laboratories Process for preparing solid formulations of lipid regulating agents with enhanced dissolution and absorption

Also Published As

Publication number Publication date
PL199870B1 (pl) 2008-11-28
MA26818A1 (fr) 2004-12-20
US20040175420A1 (en) 2004-09-09
BRPI0013939B1 (pt) 2017-07-18
HK1049966A1 (en) 2003-06-06
HU228858B1 (en) 2013-06-28
US20030181512A1 (en) 2003-09-25
MEP90808A (en) 2011-12-20
EG24117A (en) 2008-07-06
US8012494B2 (en) 2011-09-06
ES2267563T3 (es) 2007-03-16
JP2003509357A (ja) 2003-03-11
PL356174A1 (en) 2004-06-14
AU7286300A (en) 2001-04-17
IL148494A0 (en) 2002-09-12
NO331906B1 (no) 2012-04-30
AR025587A1 (es) 2002-12-04
EP1216025B1 (en) 2006-07-26
CZ20021276A3 (cs) 2003-04-16
JP4217016B2 (ja) 2009-01-28
ZA200201518B (en) 2003-07-30
HRP20020205B1 (hr) 2011-06-30
MY130200A (en) 2007-06-29
TR200200606T2 (tr) 2002-07-22
CA2383916A1 (en) 2001-03-22
SI1216025T1 (sl) 2006-12-31
HRP20020205A2 (en) 2004-04-30
CA2383916C (en) 2009-01-20
KR20020063852A (ko) 2002-08-05
UY26338A1 (es) 2000-10-31
WO2001019340A1 (en) 2001-03-22
HUP0202737A2 (hu) 2003-01-28
EP1216025A1 (en) 2002-06-26
ME00674B (me) 2011-12-20
DK1216025T3 (da) 2006-10-30
DE60029602D1 (de) 2006-09-07
NZ517545A (en) 2003-11-28
PT1216025E (pt) 2006-12-29
ATE333866T1 (de) 2006-08-15
BR0013939A (pt) 2002-05-14
CN1197551C (zh) 2005-04-20
DE60029602T2 (de) 2007-07-26
NO20021204D0 (no) 2002-03-12
HUP0202737A3 (en) 2005-01-28
JO2386B1 (en) 2007-06-17
RU2239428C2 (ru) 2004-11-10
AU769415B2 (en) 2004-01-29
CN1373656A (zh) 2002-10-09
PE20010595A1 (es) 2001-05-26
TWI243060B (en) 2005-11-11
KR100572434B1 (ko) 2006-04-18
YU17202A (sh) 2006-01-16
RS50422B (sr) 2009-12-31
MXPA02002034A (es) 2002-08-20
CY1106180T1 (el) 2011-06-08
CZ301901B6 (cs) 2010-07-28
US20110275706A1 (en) 2011-11-10
NO20021204L (no) 2002-03-12

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