CN85104471B - 双—三唑衍生物的制备方法 - Google Patents

双—三唑衍生物的制备方法

Info

Publication number
CN85104471B
CN85104471B CN85104471A CN85104471A CN85104471B CN 85104471 B CN85104471 B CN 85104471B CN 85104471 A CN85104471 A CN 85104471A CN 85104471 A CN85104471 A CN 85104471A CN 85104471 B CN85104471 B CN 85104471B
Authority
CN
China
Prior art keywords
compound
formula
salt
ether
milliliters
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CN85104471A
Other languages
English (en)
Chinese (zh)
Other versions
CN85104471A (zh
Inventor
巴斯
库珀
理查森
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of CN85104471A publication Critical patent/CN85104471A/zh
Publication of CN85104471B publication Critical patent/CN85104471B/zh
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Zoology (AREA)
  • Pest Control & Pesticides (AREA)
  • Environmental Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Epoxy Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CN85104471A 1984-06-07 1985-06-11 双—三唑衍生物的制备方法 Expired CN85104471B (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB848414519A GB8414519D0 (en) 1984-06-07 1984-06-07 Triazole antifungal agents

Publications (2)

Publication Number Publication Date
CN85104471A CN85104471A (zh) 1986-12-10
CN85104471B true CN85104471B (zh) 1987-10-21

Family

ID=10562061

Family Applications (1)

Application Number Title Priority Date Filing Date
CN85104471A Expired CN85104471B (zh) 1984-06-07 1985-06-11 双—三唑衍生物的制备方法

Country Status (25)

Country Link
US (1) US4618616A (enExample)
EP (1) EP0164246B1 (enExample)
JP (1) JPS611672A (enExample)
KR (1) KR870001829B1 (enExample)
CN (1) CN85104471B (enExample)
AT (1) ATE36328T1 (enExample)
AU (1) AU554476B2 (enExample)
CA (1) CA1287059C (enExample)
DD (1) DD235641A5 (enExample)
DE (1) DE3564266D1 (enExample)
DK (1) DK170301B1 (enExample)
ES (1) ES8604170A1 (enExample)
FI (1) FI86176C (enExample)
GB (1) GB8414519D0 (enExample)
GR (1) GR851382B (enExample)
HU (1) HU195647B (enExample)
IE (1) IE57804B1 (enExample)
IL (1) IL75410A (enExample)
NO (1) NO852287L (enExample)
NZ (1) NZ212317A (enExample)
PH (1) PH22870A (enExample)
PL (1) PL144920B1 (enExample)
PT (1) PT80598B (enExample)
YU (1) YU94985A (enExample)
ZA (1) ZA854250B (enExample)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3440114A1 (de) * 1984-11-02 1986-05-07 Bayer Ag, 5090 Leverkusen Antimykotische mittel
EP0180850A3 (de) * 1984-11-02 1987-05-27 Bayer Ag Antimykotische Azolylmethyl-cyclopropyl-carbinol Derivate
DE3440117A1 (de) * 1984-11-02 1986-05-15 Bayer Ag, 5090 Leverkusen Substituierte azolylcyclopropyl-azolylmethyl-carbinol-derivate
GB8429932D0 (en) * 1984-11-27 1985-01-03 Pfizer Ltd Triazole antifungal agents
DE3608792A1 (de) * 1986-03-15 1987-09-24 Hoechst Ag 1,1-disubstituierte cyclopropanderivate, verfahren zu ihrer herstellung und ihre verwendung
DE3608727A1 (de) * 1986-03-15 1987-09-17 Hoechst Ag 1,1-disubstituierte cyclopropanderivate, verfahren zu ihrer herstellung sowie ihre verwendung als antimykotika oder als zwischenprodukte
DE3837463A1 (de) * 1988-11-04 1990-05-10 Bayer Ag Substituierte bisazole, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
DE3921162A1 (de) * 1989-06-28 1991-01-10 Bayer Ag Verwendung von substituierten bis-azolyl-derivaten zur bekaempfung von pilzen im pflanzenschutz
US5247094A (en) * 1990-01-24 1993-09-21 Bayer Aktiengesellschaft 1-(3- or 5-halo-1,2,4-triazol-1-yl)ethyl phenyl ketone intermediates
US5039676A (en) * 1990-05-11 1991-08-13 Schering Corporation Tri- and tetra-substituted-oxetanes and tetrahydrofurans and intermediates thereof
US5488035A (en) * 1991-12-06 1996-01-30 Pioneer Hi-Bred International, Inc. Peptide with inhibitory activity towards plant pathogenic fungi
JPH06340636A (ja) * 1993-05-31 1994-12-13 Ss Pharmaceut Co Ltd トリアゾール誘導体又はその塩、及びこれを含有する抗真菌剤
RU2141955C1 (ru) * 1997-06-04 1999-11-27 Санкт-Петербургский государственный университет технологии и дизайна Способ получения бис-1,2-(1,2,4-триазол-1-ил)этана
BR112015018547A2 (pt) * 2013-02-04 2017-07-18 Syngenta Participations Ag microbiocidas

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0051565A1 (de) * 1980-11-03 1982-05-12 Ciba-Geigy Ag 1-N,N-Dimethylcarbamoyl-3(5)-cyclopropyl-1,2,4-triazole, Verfahren zu ihrer Herstellung und ihre Verwendung in der Schädlingsbekämpfung
DE3337937A1 (de) * 1982-10-28 1984-05-03 Sandoz-Patent-GmbH, 7850 Lörrach Neue azolderivate
GB8302500D0 (en) * 1983-01-29 1983-03-02 Pfizer Ltd Antifungal agents
DE3305834A1 (de) * 1983-02-19 1984-08-23 Bayer Ag, 5090 Leverkusen Mikrobizides mittel zum schutz technischer mineralien
DE3440114A1 (de) * 1984-11-02 1986-05-07 Bayer Ag, 5090 Leverkusen Antimykotische mittel
EP0180850A3 (de) * 1984-11-02 1987-05-27 Bayer Ag Antimykotische Azolylmethyl-cyclopropyl-carbinol Derivate
GB8429932D0 (en) * 1984-11-27 1985-01-03 Pfizer Ltd Triazole antifungal agents

Also Published As

Publication number Publication date
PL144920B1 (en) 1988-07-30
PT80598A (en) 1985-07-01
US4618616A (en) 1986-10-21
CA1287059C (en) 1991-07-30
IL75410A (en) 1989-02-28
FI852223A0 (fi) 1985-06-03
NZ212317A (en) 1988-04-29
KR860000288A (ko) 1986-01-27
FI86176C (fi) 1992-07-27
DE3564266D1 (en) 1988-09-15
ATE36328T1 (de) 1988-08-15
AU554476B2 (en) 1986-08-21
HUT38326A (en) 1986-05-28
EP0164246A3 (en) 1987-01-28
YU94985A (en) 1987-10-31
HU195647B (en) 1988-06-28
DK170301B1 (da) 1995-07-31
GR851382B (enExample) 1985-11-25
JPS611672A (ja) 1986-01-07
FI852223L (fi) 1985-12-08
GB8414519D0 (en) 1984-07-11
AU4334885A (en) 1985-12-12
FI86176B (fi) 1992-04-15
ZA854250B (en) 1987-01-28
DK253685A (da) 1985-12-08
IE57804B1 (en) 1993-04-07
CN85104471A (zh) 1986-12-10
ES543998A0 (es) 1986-01-16
DD235641A5 (de) 1986-05-14
DK253685D0 (da) 1985-06-06
EP0164246A2 (en) 1985-12-11
ES8604170A1 (es) 1986-01-16
PT80598B (en) 1987-04-23
EP0164246B1 (en) 1988-08-10
JPH0521108B2 (enExample) 1993-03-23
KR870001829B1 (ko) 1987-10-15
IE851416L (en) 1985-12-07
NO852287L (no) 1985-12-09
PH22870A (en) 1989-01-19
PL253666A1 (en) 1986-06-17

Similar Documents

Publication Publication Date Title
US4616027A (en) Antifungal 1-aryl-1-fluoroalkyl-2-(1H-1,2,4-triazol-1-yl)ethanols
JPH0543701B2 (enExample)
EP0096569A2 (en) Triazole antifungal agents
EP0106515A2 (en) Triazole anti-fungal agents
EP0164246B1 (en) Triazole antifungal agents
EP0183494B1 (en) Triazole antifungal agents
EP0117100A1 (en) Triazole antifungal agents
EP0126581B1 (en) Antifungal triazole derivatives
JPS59181266A (ja) トリアゾ−ル抗真菌剤
JPS5998073A (ja) トリアゾ−ル系抗真菌剤
US4483862A (en) 2-(1H-1,2,4-triazol-1-yl)-1,1-bis-(perfluoro-alkyl)ethanol antifungal agents
EP0133805B1 (en) Triazole antifungal agents
US4529799A (en) Bis-pyridyl containing triazoles
JPS5993062A (ja) トリアゾ−ル系抗真菌剤
JPS5948468A (ja) トリアゾ−ル系抗真菌薬
CS235346B2 (cs) Fungicidní prostředek k ošetřování rostlin nebo semen a způsob výroby účinných látek
CS246097B2 (cs) Fungicidní prostředek pro použití v zemědělství a způsob výroby účinných látek
DD232044A5 (de) Verfahren zur herstellung von triazol-derivaten

Legal Events

Date Code Title Description
C10 Entry into substantive examination
SE01 Entry into force of request for substantive examination
PB01 Publication
C06 Publication
C13 Decision
GR02 Examined patent application
C14 Grant of patent or utility model
GR01 Patent grant